Search Results - "ROSSI Tino" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Discovery Process and Pharmacological Characterization of 2-(S)-(4-Fluoro-2-methylphenyl)piperazine-1-carboxylic Acid [1-(R)-(3,5-Bis-trifluoromethylphenyl)ethyl]methylamide (Vestipitant) as a Potent, Selective, and Orally Active NK1 Receptor Antagonist

Discovery Process and Pharmacological Characterization of 2-(S)-(4-Fluoro-2-methylphenyl)piperazine-1-carboxylic Acid [1-(R)-(3,5-Bis-trifluoromethylphenyl)ethyl]methylamide (Vestipitant) as a Potent, Selective, and Orally Active NK1 Receptor Antagonist

by Di Fabio, Romano, Griffante, Cristiana, Alvaro, Giuseppe, Pentassuglia, Giorgio, Pizzi, Domenica A, Donati, Daniele, Rossi, Tino, Guercio, Giuseppe, Mattioli, Mario, Cimarosti, Zadeo, Marchioro, Carla, Provera, Stefano, Zonzini, Laura, Montanari, Dino, Melotto, Sergio, Gerrard, Philip A, Trist, David G, Ratti, Emiliangelo, Corsi, Mauro
Published in Journal of medicinal chemistry (28.05.2009)

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Journal Article

Quality by Design in lead optimization: a new strategy to address productivity in drug discovery

Quality by Design in lead optimization: a new strategy to address productivity in drug discovery

by Rossi, Tino, Braggio, Simone
Published in Current opinion in pharmacology (01.10.2011)

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Journal Article

Stereoselective Synthesis of a Key Intermediate of Sanfetrinem by Means of a Chelated Tin(IV) Enolate

Stereoselective Synthesis of a Key Intermediate of Sanfetrinem by Means of a Chelated Tin(IV) Enolate

by Rossi, Tino, Marchioro, Carla, Paio, Alfredo, Thomas, Russell J, Zarantonello, Paola
Published in Journal of organic chemistry (21.03.1997)

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Journal Article

Solution phase library of perhydrooxazin-4-ones

Solution phase library of perhydrooxazin-4-ones

by Panunzio, Mauro, Villa, Marzia, Missio, Andrea, Rossi, Tino, Seneci, Pierfausto
Published in Tetrahedron letters (01.09.1998)

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Journal Article

The synthesis of a key intermediate of tricyclic beta-lactam antibiotics

The synthesis of a key intermediate of tricyclic beta-lactam antibiotics

by Bismara, Claudio, Di Fabio, Romano, Donati, Daniele, Rossi, Tino, Thomas, Russell J.
Published in Tetrahedron letters (12.06.1995)

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Journal Article

도파민-B-하이드록실라제 억제제

도파민-B-하이드록실라제 억제제

by BELIAEV ALEXANDER, KISS LASZLO, PINTO RUI, ROSSI TINO, CARDONA FRANCISCO, SOARES DA SILVA PATRICIO, PALMA NUNO
Year of Publication 07.04.2022

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Patent

Drug efficiency: a new concept to guide lead optimization programs towards the selection of better clinical candidates

Drug efficiency: a new concept to guide lead optimization programs towards the selection of better clinical candidates

by Braggio, Simone, Montanari, Dino, Rossi, Tino, Ratti, Emiliangelo
Published in Expert opinion on drug discovery (01.07.2010)

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Journal Article

Application of drug efficiency index in drug discovery: a strategy towards low therapeutic dose

Application of drug efficiency index in drug discovery: a strategy towards low therapeutic dose

by Montanari, Dino, Chiarparin, Elisabetta, Gleeson, Matthew Paul, Braggio, Simone, Longhi, Raffaele, Valko, Klara, Rossi, Tino
Published in Expert opinion on drug discovery (01.09.2011)

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Journal Article

1,2,4-Triazol-3-yl-thiopropyl-tetrahydrobenzazepines: A Series of Potent and Selective Dopamine D 3 Receptor Antagonists

1,2,4-Triazol-3-yl-thiopropyl-tetrahydrobenzazepines: A Series of Potent and Selective Dopamine D 3 Receptor Antagonists

by Micheli, Fabrizio, Bonanomi, Giorgio, Blaney, Frank E., Braggio, Simone, Capelli, Anna Maria, Checchia, Anna, Curcuruto, Ornella, Damiani, Federica, Di Fabio, Romano, Donati, Daniele, Gentile, Gabriella, Gribble, Andy, Hamprecht, Dieter, Tedesco, Giovanna, Terreni, Silvia, Tarsi, Luca, Lightfoot, Andrew, Stemp, Geoff, MacDonald, Gregor, Smith, Alex, Pecoraro, Michela, Petrone, Marcella, Perini, Ornella, Piner, Jacqui, Rossi, Tino, Worby, Angela, Pilla, Maria, Valerio, Enzo, Griffante, Cristiana, Mugnaini, Manolo, Wood, Martyn, Scott, Claire, Andreoli, Michela, Lacroix, Laurent, Schwarz, Adam, Gozzi, Alessandro, Bifone, Angelo, Ashby, Charles R., Hagan, Jim J., Heidbreder, Christian
Published in Journal of medicinal chemistry (18.10.2007)

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Journal Article

도파민-B-하이드록실라제 억제제

도파민-B-하이드록실라제 억제제

by PALMA PEDRO NUNO LEAL, KISS LASZLO ERNO, BELIAEV ALEXANDER, PINTO RUI, SOARES DA SILVA PATRICIO MANUEL VIEIRA ARAUJO, ROSSI TINO, CARDONA FRANCISCO
Year of Publication 12.08.2020

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Patent

혈액-뇌 장벽-투과성 도파민-β-하이드록실라제 저해제

혈액-뇌 장벽-투과성 도파민-β-하이드록실라제 저해제

by KISS LASZLO ERNO, BELIAEV ALEXANDER, LEAL PALMA PEDRO NUNO, ROSSI TINO, SOARES DA SILVA PATRICIO
Year of Publication 08.07.2019

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Patent

도파민-β-하이드록실라제 저해제

도파민-β-하이드록실라제 저해제

by KISS LASZLO ERNO, BELIAEV ALEXANDER, LEAL PALMA PEDRO NUNO, ROSSI TINO, SOARES DA SILVA PATRICIO
Year of Publication 02.07.2019

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Patent

Analogues of 4,5-bis(3,5-dichlorophenyl)-2-trifluoromethyl-1H-imidazole as potential antibacterial agents

Analogues of 4,5-bis(3,5-dichlorophenyl)-2-trifluoromethyl-1H-imidazole as potential antibacterial agents

by ANTOLINI, M, BOZZOLI, A, GHIRON, C, KENNEDY, G, ROSSI, T, URSINI, A
Published in Bioorganic & medicinal chemistry letters (05.04.1999)

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Journal Article

Californians Reject New Taxes and Borrowing

Californians Reject New Taxes and Borrowing

by Rossi, Tino
Published in Fox & Hounds [BLOG] (12.03.2020)

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Web Resource

Saying ‘Goodbye’ to California

Saying ‘Goodbye’ to California

by Rossi, Tino
Published in Fox & Hounds [BLOG] (12.03.2020)

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Web Resource

A Brief Note on Being the Envy of the World

A Brief Note on Being the Envy of the World

by Rossi, Tino
Published in Fox & Hounds [BLOG] (12.03.2020)

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Web Resource

Exempt All Small Businesses Under AB 5

Exempt All Small Businesses Under AB 5

by Rossi, Tino
Published in Fox & Hounds [BLOG] (12.03.2020)

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Web Resource

Dopamine D 3 receptor antagonists: The quest for a potentially selective PET ligand. Part 3: Radiosynthesis and in vivo studies

Dopamine D 3 receptor antagonists: The quest for a potentially selective PET ligand. Part 3: Radiosynthesis and in vivo studies

by Bennacef, Idriss, Salinas, Cristian A., Bonasera, Thomas A., Gunn, Roger N., Audrain, Hélène, Jakobsen, Steen, Nabulsi, Nabeel, Weinzimmer, David, Carson, Richard E., Huang, Yiyun, Holmes, Ian, Micheli, Fabrizio, Heidbreder, Christian, Gentile, Gabriella, Rossi, Tino, Laruelle, Marc
Published in Bioorganic & medicinal chemistry letters (01.09.2009)

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Journal Article

Application of LC-NMR to the identification of bulk drug impurities in NK1 antagonist GW597599 (vestipitant)

Application of LC-NMR to the identification of bulk drug impurities in NK1 antagonist GW597599 (vestipitant)

by Provera, Stefano, Guercio, Giuseppe, Turco, Lucilla, Curcuruto, Ornella, Alvaro, Giuseppe, Rossi, Tino, Marchioro, Carla
Published in Magnetic resonance in chemistry (01.07.2010)

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Journal Article

The Perils of Regulating Drugs by Sound Bite

The Perils of Regulating Drugs by Sound Bite

by Rossi, Tino
Published in Fox & Hounds [BLOG] (16.05.2019)

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Web Resource

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