New Benzylureas as a Novel Series of Potent, Nonpeptidic Vasopressin V2 Receptor Agonists
Yea, Christopher M, Allan, Christine E, Ashworth, Doreen M, Barnett, James, Baxter, Andy J, Broadbridge, Janice D, Franklin, Richard J, Hampton, Sally L, Hudson, Peter, Horton, John A, Jenkins, Paul D, Penson, Andy M, Pitt, Gary R. W, Rivière, Pierre, Robson, Peter A, Rooker, David P, Semple, Graeme, Sheppard, Andy, Haigh, Robert M, Roe, Michael B
Published in Journal of medicinal chemistry (25.12.2008)
Published in Journal of medicinal chemistry (25.12.2008)
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(3R)-N-(1-(tert-Butylcarbonylmethyl)-2,3-dihydro-2-oxo-5-(2-pyridyl)-1H- 1,4-benzodiazepin-3-yl)-N‘-(3-(methylamino)phenyl)urea (YF476): A Potent and Orally Active Gastrin/CCK-B Antagonist
Semple, Graeme, Ryder, Hamish, Rooker, David P, Batt, Andrzej R, Kendrick, David A, Szelke, Michael, Ohta, Mitsuaki, Satoh, Masato, Nishida, Akito, Akuzawa, Shinobu, Miyata, Keiji
Published in Journal of medicinal chemistry (31.01.1997)
Published in Journal of medicinal chemistry (31.01.1997)
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PYRIDONE-BASED PEPTIDOMIMETIC INHIBITORS OF INTERLEUKIN-1β-CONVERTING ENZYME (ICE)
Semple, Graeme, Ashworth, Doreen M, Baker, Graham R, Batt, Andrzej R, Baxter, Andrew J, Benzies, David W.M, Elliot, Lucy H, Evans, D.Michael, Franklin, Richard J, Hudson, Peter, Jenkins, Paul D, Pitt, Gary R, Rooker, David P, Sheppard, Andrew, Szelke, Michael, Yamamoto, Satoshi, Isomura, Yasuo
Published in Bioorganic & medicinal chemistry letters (20.05.1997)
Published in Bioorganic & medicinal chemistry letters (20.05.1997)
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Non-peptide oxytocin agonists
PITT, Gary R. W, BATT, Andrzej R, HAIGH, Robert M, PENSON, Andrew M, ROBSON, Peter A, ROOKER, David P, TARTAR, André L, TRIM, Julie E, YEA, Christopher M, ROE, Michael B
Published in Bioorganic & medicinal chemistry letters (06.09.2004)
Published in Bioorganic & medicinal chemistry letters (06.09.2004)
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Peptidomimetic aminomethylene ketone inhibitors of interleukin-1β-converting enzyme (ICE)
Semple, Graeme, Ashworth, Doreen M., Batt, Andrzej R., Baxter, Andrew J., Benzies, David W.M., Elliot, Lucy H., Evans, D.Michael, Franklin, Richard J., Hudson, Peter, Jenkins, Paul D., Pitt, Gary R., Rooker, David P., Yamamoto, Satoshi, Isomura, Yasuo
Published in Bioorganic & medicinal chemistry letters (21.04.1998)
Published in Bioorganic & medicinal chemistry letters (21.04.1998)
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(3 R )- N -(1-( tert -Butylcarbonylmethyl)-2,3-dihydro-2-oxo-5-(2-pyridyl)-1 H - 1,4-benzodiazepin-3-yl)- N ‘-(3-(methylamino)phenyl)urea (YF476): A Potent and Orally Active Gastrin/CCK-B Antagonist
Semple, Graeme, Ryder, Hamish, Rooker, David P., Batt, Andrzej R., Kendrick, David A., Szelke, Michael, Ohta, Mitsuaki, Satoh, Masato, Nishida, Akito, Akuzawa, Shinobu, Miyata, Keiji
Published in Journal of medicinal chemistry (01.01.1997)
Published in Journal of medicinal chemistry (01.01.1997)
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Identification and biological activity of novel peptidomimetic gastrin/CCK-B receptor agonists
Semple, Graeme, Ryder, Hamish, Kendrick, David A., Batt, Andrzej R., Mathews, Elizabeth, Rooker, David P., Szelke, Michael, Nishida, Akito, Miyata, Keiji
Published in Bioorganic & medicinal chemistry letters (17.12.1996)
Published in Bioorganic & medicinal chemistry letters (17.12.1996)
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Non-peptide gnrh antagonists
ROOKER DAVID P, ROE MICHAEL B, BATT ANDRZEJ R, PITT GARY R.W, EVANS DAVID M
Year of Publication 06.10.2005
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Year of Publication 06.10.2005
Patent
Non-Peptide Oxytocin Agonists
Pitt, Gary R. W., Batt, Andrzej R., Haigh, Robert M., Penson, Andrew M, Robson, Peter A., Rooker, David P., Tartar, Andre L., Trim, Julie E., Yea, Christopher M., Roe, Michael B.
Published in ChemInform (28.12.2004)
Published in ChemInform (28.12.2004)
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