A miniaturized mode-of-action profiling platform enables high throughput characterization of the molecular and cellular dynamics of EZH2 inhibition
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Published in Scientific reports (19.01.2024)
Published in Scientific reports (19.01.2024)
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Published in Journal for immunotherapy of cancer (01.11.2023)
Published in Journal for immunotherapy of cancer (01.11.2023)
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Published in Journal for immunotherapy of cancer (01.11.2023)
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Discovery of BAY-298 and BAY-899: Tetrahydro-1,6-naphthyridine-Based, Potent, and Selective Antagonists of the Luteinizing Hormone Receptor Which Reduce Sex Hormone Levels in Vivo
Wortmann, Lars, Lindenthal, Bernhard, Muhn, Peter, Walter, Alexander, Nubbemeyer, Reinhard, Heldmann, Dieter, Sobek, Lothar, Morandi, Federica, Schrey, Anna K, Moosmayer, Dieter, Günther, Judith, Kuhnke, Joachim, Koppitz, Marcus, Lücking, Ulrich, Röhn, Ulrike, Schäfer, Martina, Nowak-Reppel, Katrin, Kühne, Ronald, Weinmann, Hilmar, Langer, Gernot
Published in Journal of medicinal chemistry (27.11.2019)
Published in Journal of medicinal chemistry (27.11.2019)
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Abstract 1288: Blocking tumor-associated immune suppression with BAY-218, a novel, selective aryl hydrocarbon receptor (AhR) inhibitor
Gutcher, Ilona, Kober, Christina, Roese, Lars, Roewe, Julian, Schmees, Norbert, Prinz, Florian, Gorjanacz, Matyas, Roehn, Ulrike, Bader, Benjamin, Irlbacher, Horst, Stoeckigt, Detlef, Carretero, Rafael, Sahm, Katharina, Oezen, Iris, Weinmann, Hilmar, Hartung, Ingo V., Kreft, Bertolt, Platten, Michael
Published in Cancer research (Chicago, Ill.) (01.07.2019)
Published in Cancer research (Chicago, Ill.) (01.07.2019)
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Abstract 4454: Identification of BAY-218, a potent and selective small-molecule AhR inhibitor, as a new modality to counteract tumor immunosuppression
Schmees, Norbert, Gutcher, Ilona, Roehn, Ulrike, Irlbacher, Horst, Stoeckigt, Detlef, Bader, Benjamin, Kober, Christina, Roese, Lars, Carretero, Rafael, Oezen, Iris, Zorn, Ludiwg, Platten, Michael, Hartung, Ingo Volker, Kreft, Bertolt, Weinmann, Hilmar
Published in Cancer research (Chicago, Ill.) (01.07.2019)
Published in Cancer research (Chicago, Ill.) (01.07.2019)
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Abstract ND04: BAY 2965501: A highly selective DGK- ζ inhibitor for cancer immuno-therapy with first-in-class potential
Offringa, Rienk, Olesch, Catherine, Cichon, Frederik, Grees, Mareike, Schmees, Norbert, Roehn, Ulrike, Prinz, Florian, Guenther, Judith, Stoeckigt, Detlef, Erkelenz, Michael, Nguyen, Thi Thanh Uyen, Boemer, Ulf, Werbeck, Nicolas, Kunze, Marc, Petersen, Kirstin, Kirchhoff, Dennis
Published in Cancer research (Chicago, Ill.) (29.05.2023)
Published in Cancer research (Chicago, Ill.) (29.05.2023)
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Published in Journal of fluorine chemistry (01.10.2009)
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Year of Publication 22.06.2011
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Year of Publication 22.06.2011
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Year of Publication 23.04.2024
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Year of Publication 04.05.2023
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Year of Publication 08.09.2021
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Year of Publication 08.09.2021
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SUBSTITUTED AMINOTHIAZOLES AS DGKZETA INHIBITORS FOR IMMUNE ACTIVATION
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Year of Publication 01.06.2023
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Year of Publication 01.06.2023
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SUBSTITUTED AMINOTHIAZOLES AS DGKZETA INHIBITORS FOR IMMUNE ACTIVATION
OFFRINGA, Rienk, LINK, Corinna, WERBECK, Nicolas, STOECKIGT, Detlef, BOEMER, Ulf, NGUYEN, Thi Thanh Uyen, BADER, Benjamin, PETERSEN, Kirstin, SCHMEES, Norbert, ROEHN, Ulrike, GREES, Mareike, TESTOLIN, Giambattista, NOWAK-REPPEL, Katrin, KIRCHHOFF, Dennis
Year of Publication 01.06.2023
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Year of Publication 01.06.2023
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