NanoBRETA Novel BRET Platform for the Analysis of Protein–Protein Interactions
Machleidt, Thomas, Woodroofe, Carolyn C, Schwinn, Marie K, Méndez, Jacqui, Robers, Matthew B, Zimmerman, Kris, Otto, Paul, Daniels, Danette L, Kirkland, Thomas A, Wood, Keith V
Published in ACS chemical biology (21.08.2015)
Published in ACS chemical biology (21.08.2015)
Get full text
Journal Article
Application of BRET to monitor ligand binding to GPCRs
Stoddart, Leigh A, Johnstone, Elizabeth K M, Wheal, Amanda J, Goulding, Joëlle, Robers, Matthew B, Machleidt, Thomas, Wood, Keith V, Hill, Stephen J, Pfleger, Kevin D G
Published in Nature methods (01.07.2015)
Published in Nature methods (01.07.2015)
Get full text
Journal Article
Engineered Luciferase Reporter from a Deep Sea Shrimp Utilizing a Novel Imidazopyrazinone Substrate
Hall, Mary P, Unch, James, Binkowski, Brock F, Valley, Michael P, Butler, Braeden L, Wood, Monika G, Otto, Paul, Zimmerman, Kristopher, Vidugiris, Gediminas, Machleidt, Thomas, Robers, Matthew B, Benink, Hélène A, Eggers, Christopher T, Slater, Michael R, Meisenheimer, Poncho L, Klaubert, Dieter H, Fan, Frank, Encell, Lance P, Wood, Keith V
Published in ACS chemical biology (16.11.2012)
Published in ACS chemical biology (16.11.2012)
Get full text
Journal Article
tracerDB: a crowdsourced fluorescent tracer database for target engagement analysis
Dopfer, Johannes, Vasta, James D., Müller, Susanne, Knapp, Stefan, Robers, Matthew B., Schwalm, Martin P.
Published in Nature communications (05.07.2024)
Published in Nature communications (05.07.2024)
Get full text
Journal Article
Selective JAK3 Inhibitors with a Covalent Reversible Binding Mode Targeting a New Induced Fit Binding Pocket
Forster, Michael, Chaikuad, Apirat, Bauer, Silke M., Holstein, Julia, Robers, Matthew B., Corona, Cesear R., Gehringer, Matthias, Pfaffenrot, Ellen, Ghoreschi, Kamran, Knapp, Stefan, Laufer, Stefan A.
Published in Cell chemical biology (17.11.2016)
Published in Cell chemical biology (17.11.2016)
Get full text
Journal Article
Quantifying CDK inhibitor selectivity in live cells
Wells, Carrow I., Vasta, James D., Corona, Cesear R., Wilkinson, Jennifer, Zimprich, Chad A., Ingold, Morgan R., Pickett, Julie E., Drewry, David H., Pugh, Kathryn M., Schwinn, Marie K., Hwang, Byounghoon (Brian), Zegzouti, Hicham, Huber, Kilian V. M., Cong, Mei, Meisenheimer, Poncho L., Willson, Timothy M., Robers, Matthew B.
Published in Nature communications (02.06.2020)
Published in Nature communications (02.06.2020)
Get full text
Journal Article
Potent and selective bivalent inhibitors of BET bromodomains
Waring, Michael J, Chen, Huawei, Rabow, Alfred A, Walker, Graeme, Bobby, Romel, Boiko, Scott, Bradbury, Rob H, Callis, Rowena, Clark, Edwin, Dale, Ian, Daniels, Danette L, Dulak, Austin, Flavell, Liz, Holdgate, Geoff, Jowitt, Thomas A, Kikhney, Alexey, McAlister, Mark, Méndez, Jacqui, Ogg, Derek, Patel, Joe, Petteruti, Philip, Robb, Graeme R, Robers, Matthew B, Saif, Sakina, Stratton, Natalie, Svergun, Dmitri I, Wang, Wenxian, Whittaker, David, Wilson, David M, Yao, Yi
Published in Nature chemical biology (01.12.2016)
Published in Nature chemical biology (01.12.2016)
Get full text
Journal Article
Exploiting an Asp-Glu "switch" in glycogen synthase kinase 3 to design paralog-selective inhibitors for use in acute myeloid leukemia
Wagner, Florence F, Benajiba, Lina, Campbell, Arthur J, Weïwer, Michel, Sacher, Joshua R, Gale, Jennifer P, Ross, Linda, Puissant, Alexandre, Alexe, Gabriela, Conway, Amy, Back, Morgan, Pikman, Yana, Galinsky, Ilene, DeAngelo, Daniel J, Stone, Richard M, Kaya, Taner, Shi, Xi, Robers, Matthew B, Machleidt, Thomas, Wilkinson, Jennifer, Hermine, Olivier, Kung, Andrew, Stein, Adam J, Lakshminarasimhan, Damodharan, Hemann, Michael T, Scolnick, Edward, Zhang, Yan-Ling, Pan, Jen Q, Stegmaier, Kimberly, Holson, Edward B
Published in Science translational medicine (07.03.2018)
Published in Science translational medicine (07.03.2018)
Get more information
Journal Article
Tetrahydroquinoline-Capped Histone Deacetylase 6 Inhibitor SW-101 Ameliorates Pathological Phenotypes in a Charcot–Marie–Tooth Type 2A Mouse Model
Shen, Sida, Picci, Cristina, Ustinova, Kseniya, Benoy, Veronick, Kutil, Zsófia, Zhang, Guiping, Tavares, Maurício T, Pavlíček, Jiří, Zimprich, Chad A, Robers, Matthew B, Van Den Bosch, Ludo, Bařinka, Cyril, Langley, Brett, Kozikowski, Alan P
Published in Journal of medicinal chemistry (22.04.2021)
Published in Journal of medicinal chemistry (22.04.2021)
Get full text
Journal Article
Development of Cell Permeable NanoBRET Probes for the Measurement of PLK1 Target Engagement in Live Cells
Yang, Xuan, Smith, Jeffery L, Beck, Michael T, Wilkinson, Jennifer M, Michaud, Ani, Vasta, James D, Robers, Matthew B, Willson, Timothy M
Published in Molecules (Basel, Switzerland) (25.03.2023)
Published in Molecules (Basel, Switzerland) (25.03.2023)
Get full text
Journal Article
Brain Penetrable Histone Deacetylase 6 Inhibitor SW-100 Ameliorates Memory and Learning Impairments in a Mouse Model of Fragile X Syndrome
Kozikowski, Alan P, Shen, Sida, Pardo, Marta, Tavares, Maurício T, Szarics, Dora, Benoy, Veronick, Zimprich, Chad A, Kutil, Zsófia, Zhang, Guiping, Bařinka, Cyril, Robers, Matthew B, Van Den Bosch, Ludo, Eubanks, James H, Jope, Richard S
Published in ACS chemical neuroscience (20.03.2019)
Published in ACS chemical neuroscience (20.03.2019)
Get full text
Journal Article
Design, Synthesis and Characterization of Covalent KDM5 Inhibitors
Vazquez‐Rodriguez, Saleta, Wright, Miranda, Rogers, Catherine M., Cribbs, Adam P., Velupillai, Srikannathasan, Philpott, Martin, Lee, Henry, Dunford, James E., Huber, Kilian V. M., Robers, Matthew B., Vasta, James D., Thezenas, Marie‐Laetitia, Bonham, Sarah, Kessler, Benedikt, Bennett, James, Fedorov, Oleg, Raynaud, Florence, Donovan, Adam, Blagg, Julian, Bavetsias, Vassilios, Oppermann, Udo, Bountra, Chas, Kawamura, Akane, Brennan, Paul E.
Published in Angewandte Chemie International Edition (08.01.2019)
Published in Angewandte Chemie International Edition (08.01.2019)
Get full text
Journal Article
Dual targeting of the androgen receptor and PI3K/AKT/mTOR pathways in prostate cancer models improves antitumor efficacy and promotes cell apoptosis
Sugawara, Tatsuo, Nevedomskaya, Ekaterina, Heller, Simon, Böhme, Annika, Lesche, Ralf, Ahsen, Oliver, Grünewald, Sylvia, Nguyen, Holly M., Corey, Eva, Baumgart, Simon J., Georgi, Victoria, Pütter, Vera, Fernández‐Montalván, Amaury, Vasta, James D., Robers, Matthew B., Politz, Oliver, Mumberg, Dominik, Haendler, Bernard
Published in Molecular oncology (01.03.2024)
Published in Molecular oncology (01.03.2024)
Get full text
Journal Article
Resistance to kinase inhibition through shortened target engagement
Rangwala, Aziz M., Berger, Benedict-Tilman, Robers, Matthew B., Knapp, Stefan, Seeliger, Markus A.
Published in Molecular & cellular oncology (31.12.2022)
Published in Molecular & cellular oncology (31.12.2022)
Get full text
Journal Article
A Toolbox for the Generation of Chemical Probes for Baculovirus IAP Repeat Containing Proteins
Schwalm, Martin P., Berger, Lena M., Meuter, Maximilian N., Vasta, James D., Corona, Cesear R., Röhm, Sandra, Berger, Benedict-Tilman, Farges, Frederic, Beinert, Sebastian M., Preuss, Franziska, Morasch, Viktoria, Rogov, Vladimir V., Mathea, Sebastian, Saxena, Krishna, Robers, Matthew B., Müller, Susanne, Knapp, Stefan
Published in Frontiers in cell and developmental biology (26.05.2022)
Published in Frontiers in cell and developmental biology (26.05.2022)
Get full text
Journal Article
Real-time analysis of the binding of fluorescent VEGF 165 a to VEGFR2 in living cells: Effect of receptor tyrosine kinase inhibitors and fate of internalized agonist-receptor complexes
Kilpatrick, Laura E, Friedman-Ohana, Rachel, Alcobia, Diana C, Riching, Kristin, Peach, Chloe J, Wheal, Amanda J, Briddon, Stephen J, Robers, Matthew B, Zimmerman, Kris, Machleidt, Thomas, Wood, Keith V, Woolard, Jeanette, Hill, Stephen J
Published in Biochemical pharmacology (01.07.2017)
Published in Biochemical pharmacology (01.07.2017)
Get full text
Journal Article
Quantitative Live-Cell Kinetic Degradation and Mechanistic Profiling of PROTAC Mode of Action
Riching, Kristin M, Mahan, Sarah, Corona, Cesear R, McDougall, Mark, Vasta, James D, Robers, Matthew B, Urh, Marjeta, Daniels, Danette L
Published in ACS chemical biology (21.09.2018)
Published in ACS chemical biology (21.09.2018)
Get full text
Journal Article
KRAS is vulnerable to reversible switch-II pocket engagement in cells
Vasta, James D., Peacock, D. Matthew, Zheng, Qinheng, Walker, Joel A., Zhang, Ziyang, Zimprich, Chad A., Thomas, Morgan R., Beck, Michael T., Binkowski, Brock F., Corona, Cesear R., Robers, Matthew B., Shokat, Kevan M.
Published in Nature chemical biology (01.06.2022)
Published in Nature chemical biology (01.06.2022)
Get full text
Journal Article