Pharmacological characterization of 1-(5-chloro-6-(trifluoromethoxy)-1H-benzoimidazol-2-yl)-1H-pyrazole-4-carboxylic acid (JNJ-42041935), a potent and selective hypoxia-inducible factor prolyl hydroxylase inhibitor
Barrett, Terrance D, Palomino, Heather L, Brondstetter, Theresa I, Kanelakis, Kimon C, Wu, Xiaodong, Haug, Peter V, Yan, Wen, Young, Andrew, Hua, Hong, Hart, Juliet C, Tran, Da-Thao, Venkatesan, Hariharan, Rosen, Mark D, Peltier, Hillary M, Sepassi, Kia, Rizzolio, Michele C, Bembenek, Scott D, Mirzadegan, Tara, Rabinowitz, Michael H, Shankley, Nigel P
Published in Molecular pharmacology (01.06.2011)
Published in Molecular pharmacology (01.06.2011)
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Leonard, Kristi A, Madge, Lisa A, Krawczuk, Paul J, Wang, Aihua, Kreutter, Kevin D, Bacani, Genesis M, Chai, Wenying, Smith, Russell C, Tichenor, Mark S, Harris, Michael C, Malaviya, Ravi, Seierstad, Mark, Johnson, Marguerite E, Venable, Jennifer D, Kim, Suzie, Hirst, Gavin C, Mathur, Ashok S, Rao, Tadimeti S, Edwards, James P, Rizzolio, Michele C, Koudriakova, Tatiana
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Published in Journal of medicinal chemistry (26.03.2020)
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Published in Journal of biomolecular screening (01.07.2009)
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JNJ-26070109 [(R)4-bromo-N-[1-(2,4-difluoro-phenyl)-ethyl]-2-(quinoxaline-5-sulfonylamino)-benzamide]: a novel, potent, and selective cholecystokinin 2 receptor antagonist with good oral bioavailability
Morton, Magda F, Barrett, Terrance D, Freedman, Jamie, Li, Lina, Rizzolio, Michele C, Prendergast, Clodagh E, Wu, Xiaodong, Moreno, Veronica, Pyati, Jayashree, Figueroa, Katherine, Cagnon, Laurence, Lagaud, Guy, Ver Donck, Luc, Ghoos, Etienne, Allison, Brett, Rabinowitz, Michael H, Shankley, Nigel P
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Identification and Optimization of Anthranilic Sulfonamides as Novel, Selective Cholecystokinin-2 Receptor Antagonists
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Published in Journal of medicinal chemistry (19.10.2006)
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Design of Selective and Soluble Inhibitors of Tumor Necrosis Factor-α Converting Enzyme (TACE)
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Published in Journal of medicinal chemistry (22.11.2001)
Published in Journal of medicinal chemistry (22.11.2001)
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JAK 패밀리의 키나제의 소분자 억제제
LEONARD KRISTI, KREUTTER KEVIN D, KOUDRIAKOVA TATIANA, TICHENOR MARK S, RIZZOLIO MICHELE C, WANG AIHUA, SMITH RUSSELL C
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Year of Publication 23.07.2019
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JAK 패밀리의 키나제의 억제제로서의 이미다조피롤로피리딘
LEONARD KRISTI, KREUTTER KEVIN D, CHAI WENYING, SEIERSTAD MARK, BACANI GENESIS M, KOUDRIAKOVA TATIANA, TICHENOR MARK S, VENABLE JENNIFER D, RIZZOLIO MICHELE C, SMITH RUSSEL C, KRAWCZUK PAUL J, WANG AIHUA
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Year of Publication 07.08.2019
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Pharmacological Characterization of 1-(5-Chloro-6-(trifluoromethoxy)-1 H -benzoimidazol-2-yl)-1 H -pyrazole-4-carboxylic Acid (JNJ-42041935), a Potent and Selective Hypoxia-Inducible Factor Prolyl Hydroxylase Inhibitor
Barrett, Terrance D., Palomino, Heather L., Brondstetter, Theresa I., Kanelakis, Kimon C., Wu, Xiaodong, Haug, Peter V., Yan, Wen, Young, Andrew, Hua, Hong, Hart, Juliet C., Tran, Da-Thao, Venkatesan, Hariharan, Rosen, Mark D., Peltier, Hillary M., Sepassi, Kia, Rizzolio, Michele C., Bembenek, Scott D., Mirzadegan, Tara, Rabinowitz, Michael H., Shankley, Nigel P.
Published in Molecular pharmacology (01.06.2011)
Published in Molecular pharmacology (01.06.2011)
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Small molecule inhibitors of the JAK family of kinases
WANG, Aihua, TICHENOR, Mark S, KOUDRIAKOVA, Tatiana, RIZZOLIO, Michele C, SMITH, Russell C, KREUTTER, Kevin D, LEONARD, Kristi
Year of Publication 05.10.2023
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Year of Publication 05.10.2023
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