Search Results - "RIDGILL, Mark" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

3-[[4-(4-Chlorophenyl)piperazin-1-yl]methyl]-1H-pyrrolo[2,3-b]pyridine: An Antagonist with High Affinity and Selectivity for the Human Dopamine D4 Receptor

3-[[4-(4-Chlorophenyl)piperazin-1-yl]methyl]-1H-pyrrolo[2,3-b]pyridine: An Antagonist with High Affinity and Selectivity for the Human Dopamine D4 Receptor

by Kulagowski, Janusz J, Broughton, Howard B, Curtis, Neil R, Mawer, Ian M, Ridgill, Mark P, Baker, Raymond, Emms, Frances, Freedman, Stephen B, Marwood, Rosemarie, Patel, Shil, Patel, Smita, Ragan, C. Ian, Leeson, Paul D
Published in Journal of medicinal chemistry (10.05.1996)

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Journal Article

Biological Profile of L-745,870, a Selective Antagonist with High Affinity for the Dopamine D4 Receptor

by Patel, S, Freedman, S, Chapman, K L, Emms, F, Fletcher, A E, Knowles, M, Marwood, R, Mcallister, G, Myers, J, Curtis, N, Kulagowski, J J, Leeson, P D, Ridgill, M, Graham, M, Matheson, S, Rathbone, D, Watt, A P, Bristow, L J, Rupniak, N M, Baskin, E, Lynch, J J, Ragan, C I
Published in The Journal of pharmacology and experimental therapeutics (01.11.1997)

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Journal Article

L-745,870, a Subtype Selective Dopamine D4 Receptor Antagonist, Does Not Exhibit a Neuroleptic-Like Profile in Rodent Behavioral Tests

by Bristow, L J, Collinson, N, Cook, G P, Curtis, N, Freedman, S B, Kulagowski, J J, Leeson, P D, Patel, S, Ragan, C I, Ridgill, M, Saywell, K L, Tricklebank, M D
Published in The Journal of pharmacology and experimental therapeutics (01.12.1997)

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Journal Article

2-Aryl indole NK1 receptor antagonists : Optimisation of the 2-aryl ring and the indole nitrogen substituent

2-Aryl indole NK1 receptor antagonists : Optimisation of the 2-aryl ring and the indole nitrogen substituent

by DINNELL, Kevin, CHICCHI, Gary G, SWAIN, Christopher J, DHAR, Madhumeeta J, ELLIOTT, Jason M, HOLLINGWORTH, Gregory J, KURTZ, Marc M, RIDGILL, Mark P, RYCROFT, Wayne, TSAO, Kwei-Lan, WILLIAMS, Angela R
Published in Bioorganic & medicinal chemistry letters (07.05.2001)

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4,4-Disubstituted cyclohexylamine NK1 receptor antagonists II

4,4-Disubstituted cyclohexylamine NK1 receptor antagonists II

by COOPER, Laura C, CARLSON, Emma J, RYCROFT, Wayne, TSAO, Kwei-Lan, SWAIN, Christopher J, CASTRO, Jose L, CHICCHI, Gary G, DINNELL, Kevin, DI SALVO, Jerry, ELLIOTT, Jason M, HOLLINGWORTH, Gregory J, KURTZ, Marc M, RIDGILL, Mark P
Published in Bioorganic & medicinal chemistry letters (08.07.2002)

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Journal Article

3'-(Arylmethyl)- and 3'-(Aryloxy)-3-phenyl-4-hydroxyquinolin- 2(1H)-ones: Orally Active Antagonists of the Glycine Site on the NMDA Receptor

3'-(Arylmethyl)- and 3'-(Aryloxy)-3-phenyl-4-hydroxyquinolin- 2(1H)-ones: Orally Active Antagonists of the Glycine Site on the NMDA Receptor

by Kulagowski, Janusz J, Baker, Raymond, Curtis, Neil R, Mawer, Ian M, Moseley, Angela M, Ridgill, Mark P, Rowley, Michael, Stansfield, Ian, Leeson, Paul D
Published in Journal of medicinal chemistry (01.05.1994)

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Journal Article

2-aryl indole NK1 antagonists : Optimisation of the amide substituent

2-aryl indole NK1 antagonists : Optimisation of the amide substituent

by SHAW, Duncan, CHICCHI, Gary G, ELLIOTT, Jason M, KURTZ, Marc, MORRISON, Denise, RIDGILL, Mark P, SZETO, Nicola, WATT, Alan P, WILLIAMS, Angela R, SWAIN, Christopher J
Published in Bioorganic & medicinal chemistry letters (03.12.2001)

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Journal Article

4,4-Disubstituted cyclohexylamine NK1 receptor antagonists I

4,4-Disubstituted cyclohexylamine NK1 receptor antagonists I

by ELLIOTT, Jason M, CASTRO, Jose L, SWAIN, Christopher J, TSAO, Kwei-Lan, LIHU YANG, CHICCHI, Gary G, COOPER, Laura C, DINNELL, Kevin, HOLLINGWORTH, Gregory J, RIDGILL, Mark P, RYCROFT, Wayne, KURTZ, Marc M, SHAW, Duncan E
Published in Bioorganic & medicinal chemistry letters (08.07.2002)

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Journal Article

METTL3 저해제로서의 폴리헤테로환식 화합물

METTL3 저해제로서의 폴리헤테로환식 화합물

by SHEPHERD JON, THOMAS ELIZABETH JANE, BLACKABY WESLEY PETER, BUBERT CHRISTIAN, BROOKFIELD FREDERICK ARTHUR, HARDICK DAVID JAMES, RIDGILL MARK PETER
Year of Publication 12.08.2022

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Patent

PAD4의 헤테로아릴 억제제

PAD4의 헤테로아릴 억제제

by RIDGILL MARK, KUMARAVEL GNANASAMBANDAM, LECCI CRISTINA, LOKE PUI, DEVRAJ RAJESH, NORTH CARL, MENICONI MIRCO, TYE HEATHER, MONCK NAT
Year of Publication 02.05.2019

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Patent

Regioselective rapid analogue syntheses of 1-methyl-3,5-diarylpyrazoles via palladium-catalysed coupling to 3(5)-pyrazolyl nonaflates

Regioselective rapid analogue syntheses of 1-methyl-3,5-diarylpyrazoles via palladium-catalysed coupling to 3(5)-pyrazolyl nonaflates

by Bourrain, S, Ridgill, M, Collins
Published in Synlett (02.04.2004)

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Journal Article

PAD4의 비시클릭 억제제

PAD4의 비시클릭 억제제

by PARROTT SHELLEY, BROMBRIDGE STEVE, LECCI CRISTINA, LOKE PUI, COOPER SOPHIE, DEVRAJ RAJESH, BOWLES LEE, NORTH CARL, MENICONI MIRCO, PALFREY JORDAN, MONCK NAT, PARKER MICHAEL F, BEAUMONT EDWARD, GADOULEAU ELISE, KOTEY ADRIAN, GLEAVE LAURA, RIDGILL MARK, KUMARAVEL GNANASAMBANDAM, TYE HEATHER, KRULLE THOMAS, KERRY PHILIP
Year of Publication 04.09.2018

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Patent

Amino acid bioisosteres: design of 2-quinolone derivatives as glycine-site N-methyl-D-aspartate receptor antagonists

Amino acid bioisosteres: design of 2-quinolone derivatives as glycine-site N-methyl-D-aspartate receptor antagonists

by Leeson, Paul D., Baker, Raymond, Carling, Robert W., Kulagowski, Janusz J., Mawer, Ian M., Ridgill, Mark P., Rowley, Michael, Smith, Julian D., Stansfield, Ian, Stevenson, Graeme I., Foster, Alan C., Kemp, John A.
Published in Bioorganic & medicinal chemistry letters (01.02.1993)

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Journal Article

PROCESSES FOR THE PREPARATION OF INHIBITORY COMPOUNDS

PROCESSES FOR THE PREPARATION OF INHIBITORY COMPOUNDS

by Ridgill, Mark Peter, Bubert, Christian, Canelli, Tommaso, Hardick, David James
Year of Publication 22.08.2024

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Patent

PROCESSES FOR THE PREPARATION OF INHIBITORY COMPOUNDS

PROCESSES FOR THE PREPARATION OF INHIBITORY COMPOUNDS

by RIDGILL, Mark Peter, BUBERT, Christian, CANELLI, Tommaso, HARDICK, David James
Year of Publication 08.12.2022

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Patent

NOVEL SULFONAMINOQUINOLINE HEPCIDIN ANTAGONISTS

NOVEL SULFONAMINOQUINOLINE HEPCIDIN ANTAGONISTS

by DAWSON GRAHAM, DUERRENBERGER FRANZ, ELLENBROEK ALBERTUS ANTONIUS, GEISSER PETER OTTO, BOYCE SUSAN, RIDGILL MARK PETER, BUHR WILM, BURCKHARDT SUSANNA, DAVENPORT TARA, YARNOLD CHRISTOPHER JOHN, CORDEN VINCENT ANTHONY, COURTNEY STEPHEN MARTIN, FUNK FELIX, SLACK MARK
Year of Publication 22.01.2014

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Patent

NOVEL PYRIMIDINE AND TRIAZINE HEPCIDINE ANTAGONISTS

NOVEL PYRIMIDINE AND TRIAZINE HEPCIDINE ANTAGONISTS

by YAU WEI TSUNG, DUERRENBERGER FRANZ, JAEGER STEFAN, GEISSER PETER OTTO, RIDGILL MARK PETER, BUHR WILM, BURCKHARDT SUSANNA, BAINBRIDGE JULIA MARIE, DAVENPORT TARA, YARNOLD CHRISTOPHER JOHN, CORDEN VINCENT ANTHONY, COURTNEY STEPHEN MARTIN, FUNK FELIX, SLACK MARK
Year of Publication 12.06.2012

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Patent

INHIBITORS OF METTL3

INHIBITORS OF METTL3

by Blackaby, Wesley Peter, Shepherd, Jon, HARDICK, DAVID JAMES, Ridgill, Mark Peter, Bubert, Christian, Brookfield, Frederick Arthur, Thomas, Elizabeth Jane
Year of Publication 28.03.2024

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Patent

METTL3 INHIBITORY COMPOUNDS

METTL3 INHIBITORY COMPOUNDS

by Blackaby, Wesley Peter, Shepherd, Jon, Ridgill, Mark Peter, Bubert, Christian, Hardick, David James, Brookfield, Frederick Arthur, Thomas, Elizabeth Jane
Year of Publication 07.12.2023

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Patent

Polyheterocyclic compounds as METTL3 inhibitors

Polyheterocyclic compounds as METTL3 inhibitors

by Blackaby, Wesley Peter, Shepherd, Jon, Ridgill, Mark Peter, Bubert, Christian, Hardick, David James, Brookfield, Frederick Arthur, Thomas, Elizabeth Jane
Year of Publication 15.08.2023

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Patent

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