Search Results - "RICHARD D. CALDWELL" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Discovery of Evobrutinib: An Oral, Potent, and Highly Selective, Covalent Bruton’s Tyrosine Kinase (BTK) Inhibitor for the Treatment of Immunological Diseases

Discovery of Evobrutinib: An Oral, Potent, and Highly Selective, Covalent Bruton’s Tyrosine Kinase (BTK) Inhibitor for the Treatment of Immunological Diseases

by Caldwell, Richard D, Qiu, Hui, Askew, Ben C, Bender, Andrew T, Brugger, Nadia, Camps, Montserrat, Dhanabal, Mohanraj, Dutt, Vikram, Eichhorn, Thomas, Gardberg, Anna S, Goutopoulos, Andreas, Grenningloh, Roland, Head, Jared, Healey, Brian, Hodous, Brian L, Huck, Bayard R, Johnson, Theresa L, Jones, Christopher, Jones, Reinaldo C, Mochalkin, Igor, Morandi, Federica, Nguyen, Ngan, Meyring, Michael, Potnick, Justin R, Santos, Dusica Cvetinovic, Schmidt, Ralf, Sherer, Brian, Shutes, Adam, Urbahns, Klaus, Follis, Ariele Viacava, Wegener, Ansgar A, Zimmerli, Simone C, Liu-Bujalski, Lesley
Published in Journal of medicinal chemistry (12.09.2019)

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Journal Article

Conformationally constrained farnesoid X receptor (FXR) agonists: Naphthoic acid-based analogs of GW 4064

Conformationally constrained farnesoid X receptor (FXR) agonists: Naphthoic acid-based analogs of GW 4064

by Akwabi-Ameyaw, Adwoa, Bass, Jonathan Y., Caldwell, Richard D., Caravella, Justin A., Chen, Lihong, Creech, Katrina L., Deaton, David N., Jones, Stacey A., Kaldor, Istvan, Liu, Yaping, Madauss, Kevin P., Marr, Harry B., McFadyen, Robert B., Miller, Aaron B., III, Frank Navas, Parks, Derek J., Spearing, Paul K., Todd, Dan, Williams, Shawn P., Wisely, G. Bruce
Published in Bioorganic & medicinal chemistry (01.08.2008)

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Journal Article

FXR agonist activity of conformationally constrained analogs of GW 4064

FXR agonist activity of conformationally constrained analogs of GW 4064

by Akwabi-Ameyaw, Adwoa, Bass, Jonathan Y., Caldwell, Richard D., Caravella, Justin A., Chen, Lihong, Creech, Katrina L., Deaton, David N., Madauss, Kevin P., Marr, Harry B., McFadyen, Robert B., Miller, Aaron B., Navas, Frank, Parks, Derek J., Spearing, Paul K., Todd, Dan, Williams, Shawn P., Bruce Wisely, G.
Published in Bioorganic & medicinal chemistry letters (15.08.2009)

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Journal Article

Substituted isoxazole analogs of farnesoid X receptor (FXR) agonist GW4064

Substituted isoxazole analogs of farnesoid X receptor (FXR) agonist GW4064

by Bass, Jonathan Y., Caldwell, Richard D., Caravella, Justin A., Chen, Lihong, Creech, Katrina L., Deaton, David N., Madauss, Kevin P., Marr, Harry B., McFadyen, Robert B., Miller, Aaron B., Parks, Derek J., Todd, Dan, Williams, Shawn P., Wisely, G. Bruce
Published in Bioorganic & medicinal chemistry letters (01.06.2009)

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Journal Article

Discovery of potent, highly selective covalent irreversible BTK inhibitors from a fragment hit

Discovery of potent, highly selective covalent irreversible BTK inhibitors from a fragment hit

by Qiu, Hui, Liu-Bujalski, Lesley, Caldwell, Richard D, Follis, Ariele Viacava, Gardberg, Anna, Goutopoulos, Andreas, Grenningloh, Roland, Head, Jared, Johnson, Theresa, Jones, Reinaldo, Mochalkin, Igor, Morandi, Federica, Neagu, Constantin, Sherer, Brian
Published in Bioorganic & medicinal chemistry letters (15.09.2018)

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Journal Article

Optimization of the efflux ratio and permeability of covalent irreversible BTK inhibitors

Optimization of the efflux ratio and permeability of covalent irreversible BTK inhibitors

by Qiu, Hui, Liu-Bujalski, Lesley, Caldwell, Richard D., Viacava Follis, Ariele, Gardberg, Anna, Goutopoulos, Andreas, Grenningloh, Roland, Head, Jared, Johnson, Theresa, Jones, Christopher C.V., Jones, Reinaldo, Mochalkin, Igor, Morandi, Federica, Neagu, Constantin, Potnick, Justin, Sherer, Brian
Published in Bioorganic & medicinal chemistry letters (01.11.2018)

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Journal Article

Discovery of 6,7-Dihydro‑5H‑pyrrolo[2,3‑a]pyrimidines as Orally Available G Protein-Coupled Receptor 119 Agonists

Discovery of 6,7-Dihydro‑5H‑pyrrolo[2,3‑a]pyrimidines as Orally Available G Protein-Coupled Receptor 119 Agonists

by Katamreddy, Subba R, Carpenter, Andrew J, Ammala, Carina E, Boros, Eric E, Brashear, Ron L, Briscoe, Celia P, Bullard, Sarah R, Caldwell, Richard D, Conlee, Christopher R, Croom, Dallas K, Hart, Shane M, Heyer, Dennis O, Johnson, Paul R, Kashatus, Jennifer A, Minick, Doug J, Peckham, Gregory E, Ross, Sean A, Roller, Shane G, Samano, Vicente A, Sauls, Howard R, Tadepalli, Sarva M, Thompson, James B, Xu, Yun, Way, James M
Published in Journal of medicinal chemistry (27.12.2012)

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Journal Article

BICYCLIC ARYL SPHINGOSINE 1-PHOSPHATE ANALOGS

BICYCLIC ARYL SPHINGOSINE 1-PHOSPHATE ANALOGS

by BIN MA, GNANASAMBANDAM KUMARAVEL, JERMAINE THOMAS, KEVIN M GUCKIAN, ZHENG GUO ZHU, TAVERAS ARTHUR G, LIN EDWARD YIN-SHIANG, RICHARD D CALDWELL, LIU XIAOGAO
Year of Publication 09.08.2018

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Patent

BICYCLIC ARYL SPHINGOSINE 1-PHOSPHATE ANALOGS

BICYCLIC ARYL SPHINGOSINE 1-PHOSPHATE ANALOGS

by BIN MA, GNANASAMBANDAM KUMARAVEL, JERMAINE THOMAS, KEVIN M GUCKIAN, ZHENG GUO ZHU, TAVERAS ARTHUR G, LIN EDWARD YIN-SHIANG, RICHARD D CALDWELL, LIU XIAOGAO
Year of Publication 01.09.2016

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Patent

2-OXO-IMIDAZOPYRIDINES AS REVERSIBLE BTK INHIBITORS AND USES THEREOF

2-OXO-IMIDAZOPYRIDINES AS REVERSIBLE BTK INHIBITORS AND USES THEREOF

by CALDWELL, Richard D
Year of Publication 18.05.2022

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Patent

2-oxo-imidazopyridines and their use

2-oxo-imidazopyridines and their use

by CALDWELL Richard D
Year of Publication 01.05.2022

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Patent

Discovery of 6,7-Dihydro-5 H -pyrrolo[2,3- a ]pyrimidines as Orally Available G Protein-Coupled Receptor 119 Agonists

Discovery of 6,7-Dihydro-5 H -pyrrolo[2,3- a ]pyrimidines as Orally Available G Protein-Coupled Receptor 119 Agonists

by Katamreddy, Subba R., Carpenter, Andrew J., Ammala, Carina E., Boros, Eric E., Brashear, Ron L., Briscoe, Celia P., Bullard, Sarah R., Caldwell, Richard D., Conlee, Christopher R., Croom, Dallas K., Hart, Shane M., Heyer, Dennis O., Johnson, Paul R., Kashatus, Jennifer A., Minick, Doug J., Peckham, Gregory E., Ross, Sean A., Roller, Shane G., Samano, Vicente A., Sauls, Howard R., Tadepalli, Sarva M., Thompson, James B., Xu, Yun, Way, James M.
Published in Journal of medicinal chemistry (27.12.2012)

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Journal Article

2-oxo-imidazopyridines as reversible BTK inhibitors and uses thereof

2-oxo-imidazopyridines as reversible BTK inhibitors and uses thereof

by Caldwell, Richard D
Year of Publication 12.08.2021

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Patent

2-OXO-IMIDAZOPYRIDINES AS REVERSIBLE BTK INHIBITORS AND USES THEREOF

2-OXO-IMIDAZOPYRIDINES AS REVERSIBLE BTK INHIBITORS AND USES THEREOF

by CALDWELL, Richard D
Year of Publication 26.06.2019

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Patent

2-oxo-imidazopyridines as reversible BTK inhibitors and uses thereof

2-oxo-imidazopyridines as reversible BTK inhibitors and uses thereof

by Caldwell, Richard D
Year of Publication 23.04.2019

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Patent

2-oxo-imidazopyridines as reversible BTK inhibitors and uses thereof

2-oxo-imidazopyridines as reversible BTK inhibitors and uses thereof

by Caldwell, Richard D
Year of Publication 28.03.2019

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Patent

2-OXO-IMIDAZOPYRIDINES AS REVERSIBLE BTK INHIBITORS AND USES THEREOF

2-OXO-IMIDAZOPYRIDINES AS REVERSIBLE BTK INHIBITORS AND USES THEREOF

by CALDWELL Richard D
Year of Publication 22.02.2018

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Patent

2-OXO-IMIDAZOPYRIDINES AS REVERSIBLE BTK INHIBITORS AND USES THEREOF

2-OXO-IMIDAZOPYRIDINES AS REVERSIBLE BTK INHIBITORS AND USES THEREOF

by CALDWELL, RICHARD D
Year of Publication 22.02.2018

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Patent

2-OXO-IMIDAZOPYRIDINES AS REVERSIBLE BTK INHIBITORS AND USES THEREOF

2-OXO-IMIDAZOPYRIDINES AS REVERSIBLE BTK INHIBITORS AND USES THEREOF

by CALDWELL, Richard D
Year of Publication 22.02.2018

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Patent

2-oxo-imidazopiridinas como inhibidores de BTK reversibles y usos de las mismas

2-oxo-imidazopiridinas como inhibidores de BTK reversibles y usos de las mismas

by CALDWELL, Richard D
Year of Publication 14.10.2022

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Patent

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