Watson−Crick Base-Pairing Properties of Tricyclo-DNA
Renneberg, Dorte, Leumann, Christian J
Published in Journal of the American Chemical Society (29.05.2002)
Published in Journal of the American Chemical Society (29.05.2002)
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Journal Article
Scalable Synthesis of C5aR1 Antagonist ACT-1014-6470 via N 7‑Selective Reductive Amination of an Unprotected Pyrazole Starting Material and Intramolecular Urea Formation with 1,1′-Carbonyl-di(1,2,4-triazol) (CDT)
Reber, Stefan, Blumer, Nicole, Leuenberger, Daniel, Fleischer, Tony, Renneberg, Dorte, Abele, Stefan, Schäfer, Gabriel
Published in Organic process research & development (21.06.2024)
Published in Organic process research & development (21.06.2024)
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Journal Article
Discovery and Characterization of a New Class of C5aR1 Antagonists Showing In Vivo Activity
Hubler, Francis, Renneberg, Dorte, Siendt, Hervé, Stamm, Simon, Hilpert, Kurt, Caroff, Eva, Delahaye, Stephane, Froidevaux, Sylvie, Murphy, Mark J.
Published in Journal of medicinal chemistry (14.03.2024)
Published in Journal of medicinal chemistry (14.03.2024)
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Journal Article
4‑((R)‑2-{[6-((S)‑3-Methoxypyrrolidin-1-yl)-2-phenylpyrimidine-4-carbonyl]amino}-3-phosphonopropionyl)piperazine-1-carboxylic Acid Butyl Ester (ACT-246475) and Its Prodrug (ACT-281959), a Novel P2Y12 Receptor Antagonist with a Wider Therapeutic Window in the Rat Than Clopidogrel
Caroff, Eva, Hubler, Francis, Meyer, Emmanuel, Renneberg, Dorte, Gnerre, Carmela, Treiber, Alexander, Rey, Markus, Hess, Patrick, Steiner, Beat, Hilpert, Kurt, Riederer, Markus A
Published in Journal of medicinal chemistry (10.12.2015)
Published in Journal of medicinal chemistry (10.12.2015)
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Journal Article
Discovery of novel bridged tetrahydronaphthalene derivatives as potent T/L-type calcium channel blockers
Renneberg, Dorte, Hubler, Francis, Rey, Markus, Hess, Patrick, Delahaye, Stephane, Gatfield, John, Iglarz, Marc, Hilpert, Kurt
Published in Bioorganic & medicinal chemistry letters (15.09.2015)
Published in Bioorganic & medicinal chemistry letters (15.09.2015)
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Journal Article
혈관염 및 염증성 질환을 치료하기 위한 C5A 수용체 조절제로서의 2,4,6,7-테트라히드로-피라졸로[4,3-D]피리미딘-5-온 유도체 및 관련 화합물
RENNEBERG DORTE, MURPHY MARK, HUBLER FRANCIS, FROIDEVAUX SYLVIE, STAMM SIMON
Year of Publication 10.09.2020
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Year of Publication 10.09.2020
Patent
4-(( R )-2-{[6-(( S )-3-Methoxypyrrolidin-1-yl)-2-phenylpyrimidine-4-carbonyl]amino}-3-phosphonopropionyl)piperazine-1-carboxylic Acid Butyl Ester (ACT-246475) and Its Prodrug (ACT-281959), a Novel P2Y 12 Receptor Antagonist with a Wider Therapeutic Window in the Rat Than Clopidogrel
Caroff, Eva, Hubler, Francis, Meyer, Emmanuel, Renneberg, Dorte, Gnerre, Carmela, Treiber, Alexander, Rey, Markus, Hess, Patrick, Steiner, Beat, Hilpert, Kurt, Riederer, Markus A.
Published in Journal of medicinal chemistry (10.12.2015)
Published in Journal of medicinal chemistry (10.12.2015)
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Journal Article
Evolution of novel tricyclic CRTh2 receptor antagonists from a (E)-2-cyano-3-(1H-indol-3-yl)acrylamide scaffold
Valdenaire, Anja, Pothier, Julien, Renneberg, Dorte, Riederer, Markus A., Peter, Oliver, Leroy, Xavier, Gnerre, Carmela, Fretz, Heinz
Published in Bioorganic & medicinal chemistry letters (15.02.2013)
Published in Bioorganic & medicinal chemistry letters (15.02.2013)
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Journal Article
테트라히드로피라졸로피리미디논 화합물을 포함하는 약학 조성물
RENNEBERG DORTE, MURPHY MARK, FOURNIER ELVIRE, FRAICHARD AMANDINE, HUBLER FRANCIS, FROIDEVAUX SYLVIE, GEISELER OLIVER, AMBUEHL MICHAEL, HERRMANN CHARLYSE, VON RAUMER MARKUS, STAMM SIMON
Year of Publication 18.03.2022
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Year of Publication 18.03.2022
Patent
Imidazopyridine/Pyrrole and Hydroxybenzimidazole/Pyrrole Pairs for DNA Minor Groove Recognition
Renneberg, Dorte, Dervan, Peter B
Published in Journal of the American Chemical Society (14.05.2003)
Published in Journal of the American Chemical Society (14.05.2003)
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Journal Article
Corrigendum to “Evolution of novel tricyclic CRTh2 receptor antagonists from a (E)-2-cyano-3-(1H-indol-3-yl)acrylamide scaffold” [Bioorg. Med. Chem. Lett. 23 (2013) 944–948]
Valdenaire, Anja, Pothier, Julien, Renneberg, Dorte, Riederer, Markus A., Peter, Oliver, Leroy, Xavier, Gnerre, Carmela, Fretz, Heinz
Published in Bioorganic & medicinal chemistry letters (01.04.2013)
Published in Bioorganic & medicinal chemistry letters (01.04.2013)
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Journal Article
Synthesis of the Sugar Building Block of Bicyclo-RNA
Haziri, Arben I., Silhar, Peter, Renneberg, Dorte, Leumann, Christian J.
Published in Synthesis (Stuttgart) (01.03.2010)
Published in Synthesis (Stuttgart) (01.03.2010)
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Journal Article
INDOLE CARBOXAMIDE DERIVATIVES AS P2X7 RECEPTOR ANTAGONISTS
RENNEBERG DORTE, HUBLER FRANCIS, KIMMERLIN THIERRY, STAMM SIMON, HILPERT KURT
Year of Publication 17.08.2015
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Year of Publication 17.08.2015
Patent
HETEROCYCLIC AMIDE DERIVATIVES AS P2X7 RECEPTOR ANTAGONISTS
RENNEBERG DORTE, HUBLER FRANCIS, KIMMERLIN THIERRY, STAMM SIMON, HILPERT KURT
Year of Publication 23.09.2014
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Year of Publication 23.09.2014
Patent
Antisense properties of tricyclo-DNA
Renneberg, Dorte, Bouliong, Emilie, Reber, Ulrich, Schümperli, Daniel, Leumann, Christian J.
Published in Nucleic acids research (01.07.2002)
Published in Nucleic acids research (01.07.2002)
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