Search Results - "RENICK, JOEL" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Development of Prodrug 4-Chloro-3-(5-methyl-3-{[4-(2-pyrrolidin-1-ylethoxy)phenyl]amino}-1,2,4-benzotriazin-7-yl)phenyl Benzoate (TG100801): A Topically Administered Therapeutic Candidate in Clinical Trials for the Treatment of Age-Related Macular Degeneration

Development of Prodrug 4-Chloro-3-(5-methyl-3-{[4-(2-pyrrolidin-1-ylethoxy)phenyl]amino}-1,2,4-benzotriazin-7-yl)phenyl Benzoate (TG100801): A Topically Administered Therapeutic Candidate in Clinical Trials for the Treatment of Age-Related Macular Degeneration

by Palanki, Moorthy S. S, Akiyama, Hideo, Campochiaro, Peter, Cao, Jianguo, Chow, Chun P, Dellamary, Luis, Doukas, John, Fine, Richard, Gritzen, Colleen, Hood, John D, Hu, Steven, Kachi, Shu, Kang, Xinshan, Klebansky, Boris, Kousba, Ahmed, Lohse, Dan, Mak, Chi Ching, Martin, Michael, McPherson, Andrew, Pathak, Ved P, Renick, Joel, Soll, Richard, Umeda, Naoyasu, Yee, Shiyin, Yokoi, Katsutoshi, Zeng, Binqi, Zhu, Hong, Noronha, Glenn
Published in Journal of medicinal chemistry (27.03.2008)

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Journal Article

Inhibitors of ABL and the ABL-T315I mutation

Inhibitors of ABL and the ABL-T315I mutation

by Noronha, Glenn, Cao, Jianguo, Chow, Chun P, Dneprovskaia, Elena, Fine, Richard M, Hood, John, Kang, Xinshan, Klebansky, Boris, Lohse, Dan, Mak, Chi Ching, McPherson, Andre, Palanki, Moorthy S S, Pathak, Ved P, Renick, Joel, Soll, Richard, Zeng, Binqi
Published in Current topics in medicinal chemistry (01.07.2008)

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Discovery and preliminary structure–activity relationship studies of novel benzotriazine based compounds as Src inhibitors

Discovery and preliminary structure–activity relationship studies of novel benzotriazine based compounds as Src inhibitors

by Noronha, Glenn, Barrett, Kathy, Cao, Jianguo, Dneprovskaia, Elena, Fine, Richard, Gong, Xianchang, Gritzen, Colleen, Hood, John, Kang, Xinshan, Klebansky, Boris, Li, G., Liao, W., Lohse, Dan, Mak, Chi Ching, McPherson, Andrew, Palanki, Moorthy S.S., Pathak, Ved P., Renick, Joel, Soll, Richard, Splittgerber, Ute, Wrasidlo, Wolfgang, Zeng, Binqi, Zhao, Ningning, Zhou, Y.
Published in Bioorganic & medicinal chemistry letters (01.11.2006)

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Metabolism and Pharmacokinetics of a Novel Src Kinase Inhibitor TG100435 ([7-(2,6-Dichloro-phenyl)-5-methyl-benzo[1,2,4]triazin-3-yl]-[4-(2-pyrrolidin-1-yl-ethoxy)-phenyl]-amine) and Its Active N-Oxide Metabolite TG100855 ([7-(2,6-Dichloro-phenyl)-5-methylbenzo[1,2,4]triazin-3-yl]-{4-[2-(1-oxy-pyrrolidin-1-yl)-ethoxy]-phenyl}-amine)

Metabolism and Pharmacokinetics of a Novel Src Kinase Inhibitor TG100435 ([7-(2,6-Dichloro-phenyl)-5-methyl-benzo[1,2,4]triazin-3-yl]-[4-(2-pyrrolidin-1-yl-ethoxy)-phenyl]-amine) and Its Active N-Oxide Metabolite TG100855 ([7-(2,6-Dichloro-phenyl)-5-methylbenzo[1,2,4]triazin-3-yl]-{4-[2-(1-oxy-pyrrolidin-1-yl)-ethoxy]-phenyl}-amine)

by Hu, Steven X, Soll, Richard, Yee, Shiyin, Lohse, Daniel L, Kousba, Ahmed, Zeng, Binqi, Yu, Xiyun, McPherson, Andrew, Renick, Joel, Cao, Jianguo, Tabak, Arek, Hood, John, Doukas, John, Noronha, Glenn, Martin, Michael
Published in Drug metabolism and disposition (01.06.2007)

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Rapid identification of a novel phosphodiesterase 7B tracer for receptor occupancy studies using LC─MS/MS

Rapid identification of a novel phosphodiesterase 7B tracer for receptor occupancy studies using LC─MS/MS

by Chen, Jie, Gu, Guibao, Chen, Mi, Scott, Trevor, Heger, Lindsay, Zook, Douglas, Chung, DeMichael, Keenan, Terence, Renick, Joel, Santora, Vincent J., Vivian, Jeffrey, Stauber, Kathe, Breitenbucher, James Guy, Tabatabaei, Ali
Published in Neurochemistry international (01.07.2020)

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Design and Synthesis of Novel and Selective Glycine Transporter‑1 (GlyT1) Inhibitors with Memory Enhancing Properties

Design and Synthesis of Novel and Selective Glycine Transporter‑1 (GlyT1) Inhibitors with Memory Enhancing Properties

by Santora, Vincent J, Almos, Theresa A, Barido, Richard, Basinger, Jillian, Bellows, Chris L, Bookser, Brett C, Breitenbucher, J. Guy, Broadbent, Nicola J, Cabebe, Clifford, Chai, Chih-Kun, Chen, Mi, Chow, Stephine, Chung, De Michael, Crickard, Lindsay, Danks, Anne M, Freestone, Graeme C, Gitnick, Dany, Gupta, Varsha, Hoffmaster, Christine, Hudson, Andrew R, Kaplan, Alan P, Kennedy, Michael R, Lee, Dong, Limberis, James, Ly, Kiev, Mak, Chi Ching, Masatsugu, Brittany, Morse, Andrew C, Na, Jim, Neul, David, Nikpur, John, Peters, Marco, Petroski, Robert E, Renick, Joel, Sebring, Kristen, Sevidal, Samantha, Tabatabaei, Ali, Wen, Jenny, Yan, Yingzhuo, Yoder, Zachary W, Zook, Douglas
Published in Journal of medicinal chemistry (26.07.2018)

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Azetidine-based selective glycine transporter-1 (GlyT1) inhibitors with memory enhancing properties

Azetidine-based selective glycine transporter-1 (GlyT1) inhibitors with memory enhancing properties

by Hudson, Andrew R., Santora, Vincent J., Petroski, Robert E., Almos, Theresa A., Anderson, Gary, Barido, Richard, Basinger, Jillian, Bellows, Chris L., Bookser, Brett C., Broadbent, Nicola J., Cabebe, Clifford, Chai, Chih-Kun, Chen, Mi, Chow, Stephine, Chung, De Michael, Heger, Lindsay, Danks, Anne M., Freestone, Graeme C., Gitnick, Dany, Gupta, Varsha, Hoffmaster, Christine, Kaplan, Alan P., Kennedy, Michael R., Lee, Dong, Limberis, James, Ly, Kiev, Mak, Chi Ching, Masatsugu, Brittany, Morse, Andrew C., Na, Jim, Neul, David, Nikpur, John, Renick, Joel, Sebring, Kristen, Sevidal, Samantha, Tabatabaei, Ali, Wen, Jenny, Xia, Shouzhen, Yan, Yingzhuo, Yoder, Zachary W., Zook, Douglas, Peters, Marco, Breitenbucher, J. Guy
Published in Bioorganic & medicinal chemistry letters (15.07.2020)

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Discovery of [7-(2,6-dichlorophenyl)-5-methylbenzo [1,2,4]triazin-3-yl]-[4-(2-pyrrolidin-1-ylethoxy)phenyl]amine—a potent, orally active Src kinase inhibitor with anti-tumor activity in preclinical assays

Discovery of [7-(2,6-dichlorophenyl)-5-methylbenzo [1,2,4]triazin-3-yl]-[4-(2-pyrrolidin-1-ylethoxy)phenyl]amine—a potent, orally active Src kinase inhibitor with anti-tumor activity in preclinical assays

by Noronha, Glenn, Barrett, Kathy, Boccia, Antonio, Brodhag, Tessa, Cao, Jianguo, Chow, Chun P., Dneprovskaia, Elena, Doukas, John, Fine, Richard, Gong, Xianchang, Gritzen, Colleen, Gu, Hong, Hanna, Ehab, Hood, John D., Hu, Steven, Kang, Xinshan, Key, Jann, Klebansky, Boris, Kousba, Ahmed, Li, Ge, Lohse, Dan, Mak, Chi Ching, McPherson, Andrew, Palanki, Moorthy S.S., Pathak, Ved P., Renick, Joel, Shi, Feng, Soll, Richard, Splittgerber, Ute, Stoughton, Silva, Tang, Suhan, Yee, Shiyin, Zeng, Binqi, Zhao, Ningning, Zhu, Hong
Published in Bioorganic & medicinal chemistry letters (01.02.2007)

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Journal Article

The design and preliminary structure–activity relationship studies of benzotriazines as potent inhibitors of Abl and Abl-T315I enzymes

The design and preliminary structure–activity relationship studies of benzotriazines as potent inhibitors of Abl and Abl-T315I enzymes

by Cao, Jianguo, Fine, Richard, Gritzen, Colleen, Hood, John, Kang, Xinshan, Klebansky, Boris, Lohse, Dan, Mak, Chi Ching, McPherson, Andrew, Noronha, Glenn, Palanki, Moorthy S.S., Pathak, Ved P., Renick, Joel, Soll, Richard, Zeng, Binqi, Zhu, Hong
Published in Bioorganic & medicinal chemistry letters (01.11.2007)

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Journal Article

Metabolism and pharmacokinetics of a novel Src kinase inhibitor TG100435 ([7-(2,6-dichloro-phenyl)-5-methyl-benzo[1,2,4]triazin-3-yl]-[4-(2-pyrrolidin-1 -yl-ethoxy)-phenyl]-amine) and its active N-oxide metabolite TG100855 ([7-(2,6-dichloro-phenyl)-5-methyl-benzo[1,2,4]triazin-3-yl]-{4-[2-(1 -oxy-pyrrolidin-1 -yl)-ethoxy]-phenyl}-amine)

Metabolism and pharmacokinetics of a novel Src kinase inhibitor TG100435 ([7-(2,6-dichloro-phenyl)-5-methyl-benzo[1,2,4]triazin-3-yl]-[4-(2-pyrrolidin-1 -yl-ethoxy)-phenyl]-amine) and its active N-oxide metabolite TG100855 ([7-(2,6-dichloro-phenyl)-5-methyl-benzo[1,2,4]triazin-3-yl]-{4-[2-(1 -oxy-pyrrolidin-1 -yl)-ethoxy]-phenyl}-amine)

by HU, Steven X, SOIL, Richard, TABAK, Arek, HOOD, John, DOUKAS, John, NORONHA, Glenn, MARTIN, Michael, SHIYIN YEE, LOHSE, Daniel L, KOUSBA, Ahmed, BINQI ZENG, XIYUN YU, MCPHERSON, Andrew, RENICK, Joel, CAO, Jianguo
Published in Drug metabolism and disposition (01.06.2007)

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Journal Article

JAK2 Inhibitors for the Treatment of Myeloprolifertive Disorders

JAK2 Inhibitors for the Treatment of Myeloprolifertive Disorders

by Hood, John, Cao, Jon, Hanna, Ehab, Lohse, Dan, Mak, Chi Ching, McPherson, Andrew, Noronha, Glenn, Renick, Joel, Zheng, Binqi, Zhu, Hong, Soll, Richard
Published in Blood (16.11.2006)

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Journal Article

BI-ARYL META-PYRIMIDINE INHIBITORS OF KINASES

BI-ARYL META-PYRIMIDINE INHIBITORS OF KINASES

by NORONHA GLENN, SOLL RICHARD M, MC PHERSON ANDREW, CAO JIANGUO, ZENG BINQI, RENICK JOEL, HOOD JOHN, MAK CHI CHING, LOHSE DANIEL, PATHAK VED
Year of Publication 10.09.2013

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Patent

Omega-carboxypyridyl substituted ureas as Raf kinase inhibitors: SAR of the amide substituent

Omega-carboxypyridyl substituted ureas as Raf kinase inhibitors: SAR of the amide substituent

by Khire, Uday R., Bankston, Donald, Barbosa, James, Brittelli, David R., Caringal, Yolanda, Carlson, Robert, Dumas, Jacques, Gane, Todd, Heald, Sarah L., Hibner, Barbara, Johnson, Jeffrey S., Katz, Michael E., Kennure, Nancy, Kingery-Wood, Jill, Lee, Wendy, Liu, Xiao-Gao, Lowinger, Timothy B., McAlexander, Ian, Monahan, Mary-Katherine, Natero, Reina, Renick, Joel, Riedl, Bernd, Rong, Hong, Sibley, Robert N., Smith, Roger A., Wolanin, Donald
Published in Bioorganic & medicinal chemistry letters (09.02.2004)

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Journal Article

Development of novel benzotriazines for drug discovery

Development of novel benzotriazines for drug discovery

by Palanki, Moorthy Ss, Cao, Jianguo, Chow, Chun P, Dneprovskaia, Elena, Mak, Chi Ching, McPherson, Andrew, Pathak, Ved P, Renick, Joel, Soll, Richard, Zeng, Binqi, Noronha, Glenn
Published in Expert opinion on drug discovery (01.01.2009)

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Journal Article

ω-CARBOXYARYL SUBSTITUTED DIPHENYL UREAS AS RAF KINASE INHIBITORS

ω-CARBOXYARYL SUBSTITUTED DIPHENYL UREAS AS RAF KINASE INHIBITORS

by KHIRE UDAY, MONAHAN MARY KATHERINE, RIEDL BERND, SMITH ROGER A, WOOD JILL E, RENICK JOEL, LOWINGER TIMOTHY B, DUMAS JACQUES, SIBLEY ROBERT N, SCOTT WILLIAM J, NATERO REINA
Year of Publication 10.06.2011

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Patent

p38 Kinase inhibitors for the treatment of arthritis and osteoporosis: thienyl, furyl, and pyrrolyl ureas

p38 Kinase inhibitors for the treatment of arthritis and osteoporosis: thienyl, furyl, and pyrrolyl ureas

by Redman, Anikó M, Johnson, Jeffrey S, Dally, Robert, Swartz, Steve, Wild, Hanno, Paulsen, Holger, Caringal, Yolanda, Gunn, David, Renick, Joel, Osterhout, Martin, Kingery-Wood, Jill, Smith, Roger A, Lee, Wendy, Dumas, Jacques, Wilhelm, Scott M, Housley, Timothy J, Bhargava, Ajay, Ranges, Gerald E, Shrikhande, Alka, Young, Deborah, Bombara, Michael, Scott, William J
Published in Bioorganic & medicinal chemistry letters (08.01.2001)

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SPINNING VESSEL SYSTEMS AND METHODS FOR MIXING, SUSPENDING PARTICULATES, ALIQUOTING, WASHING MAGNETIC BEADS, AND CONCENTRATING ANALYTES

SPINNING VESSEL SYSTEMS AND METHODS FOR MIXING, SUSPENDING PARTICULATES, ALIQUOTING, WASHING MAGNETIC BEADS, AND CONCENTRATING ANALYTES

by RENICK, Joel, I, HICKMAN, Christopher, P.W, MYERS, Kristi, K, ANGELO, Christopher, A, LOI, Alan, J, CHAVEZ, John, E, KNUTH, Natalie, A, CLEVELAND, Patrick, H
Year of Publication 12.07.2023

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Patent

Spinning vessel systems and methods for mixing, suspending particulates, aliquoting, washing magnetic beads, and concentrating analytes

Spinning vessel systems and methods for mixing, suspending particulates, aliquoting, washing magnetic beads, and concentrating analytes

by Cleveland, Patrick H, Myers, Kristi K, Loi, Alan J, Knuth, Natalie A, Angelo, Christopher A, Renick, Joel I, Chavez, John E, Hickman, Christopher P. W
Year of Publication 11.04.2023

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Patent

SPINNING VESSEL SYSTEMS AND METHODS FOR MIXING, SUSPENDING PARTICULATES, ALIQUOTING, WASHING MAGNETIC BEADS, AND CONCENTRATING ANALYTES

SPINNING VESSEL SYSTEMS AND METHODS FOR MIXING, SUSPENDING PARTICULATES, ALIQUOTING, WASHING MAGNETIC BEADS, AND CONCENTRATING ANALYTES

by RENICK, Joel, I, HICKMAN, Christopher, P.W, MYERS, Kristi, K, ANGELO, Christopher, A, LOI, Alan, J, CHAVEZ, John, E, KNUTH, Natalie, A, CLEVELAND, Patrick, H
Year of Publication 31.08.2022

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Patent

SPINNING VESSEL SYSTEMS AND METHODS FOR MIXING, SUSPENDING PARTICULATES, ALIQUOTING, WASHING MAGNETIC BEADS, AND CONCENTRATING ANALYTES

SPINNING VESSEL SYSTEMS AND METHODS FOR MIXING, SUSPENDING PARTICULATES, ALIQUOTING, WASHING MAGNETIC BEADS, AND CONCENTRATING ANALYTES

by KNUTH, Natalie, RENICK, Joel, MYERS, Kristi, LOI, Alan, HICKMAN, Christopher, CLEVELAND, Patrick, CHAVEZ, John, ANGELO, Christopher
Year of Publication 04.06.2020

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