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Published in Nature (London) (03.05.2012)
Published in Nature (London) (03.05.2012)
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Maiso, Patricia, Liu, Yi, Morgan, Brittany, Azab, Abdel Kareem, Ren, Pingda, Martin, Michel B., Zhang, Yong, Liu, Yang, Sacco, Antonio, Ngo, Hai, Azab, Feda, Quang, Phong, Rodig, Scott J., Lin, Charles P., Roccaro, Aldo M., Rommel, Christian, Ghobrial, Irene M.
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Catalytic Asymmetric Benzylic C−H Activation by Means of Carbenoid-Induced C−H Insertions
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Published in Journal of organic chemistry (14.06.2002)
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Discovery of pyrimidine benzimidazoles as Src-family selective Lck inhibitors. Part II
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Selective Inhibition of Oncogenic KRAS Output with Small Molecules Targeting the Inactive State
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Menin inhibitor MI-3454 induces remission in MLL1-rearranged and NPM1-mutated models of leukemia
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Synthesis of 2β-Acyl-3β-(substituted naphthyl)-8-azabicyclo[3.2.1]octanes and Their Binding Affinities at Dopamine and Serotonin Transport Sites
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Published in Journal of medicinal chemistry (10.05.2001)
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Solid Form Selection and Process Development of KO-947 Drug Substances
Mei, Bo, Zhu, Linrong, Guo, Yushen, Wu, Tao, Ren, Pingda, Deng, Xiaohu
Published in Organic process research & development (16.07.2021)
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Development of a Recycling Process for an Industrial-Scale Production of Tipifarnib
Deng, Xiaohu, Ren, Pingda, Mai, Wanping, Fu, Thomas, Zhang, Hang, Cai, Xianfeng, Wang, Lu
Published in Organic process research & development (16.07.2021)
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From Lab Formulation Development to CTM Manufacturing of KO-947 Injectable Drug Products: a Case Study and Lessons Learned
Deng, Xiaohu, Ren, Pingda, Mai, Wanping, Wang, Yi, Zhang, Yuanyang, Wu, Hongbing, Xie, Yinwei, Chen, Huazhen
Published in AAPS PharmSciTech (01.07.2021)
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Selective Metalation of Functionalized Quinazolines to Enable Discovery and Advancement of Covalent KRAS Inhibitors
Allison, Brett D., Deng, Xiaohu, Li, Lian-Sheng, Liang, Jimmy, Mani, Neelakandha S., Ren, Pingda, Sales, Zachary S.
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PI3 Kinase δ Is a Key Regulator of Synoviocyte Function in Rheumatoid Arthritis
Bartok, Beatrix, Boyle, David L, Liu, Yi, Ren, Pingda, Ball, Scott T, Bugbee, William D, Rommel, Christian, Firestein, Gary S
Published in The American journal of pathology (01.05.2012)
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Hindered Biaryl Bond Construction and Subsequent Diastereomeric Crystallization to Produce an Atropisomeric Covalent KRASG12C Inhibitor ARS-2102
Yang, Xiaogen, Li, Zhiwen, Xu, Wenwen, Zhu, Guanming, Feng, Xiantong, Zhang, Jun, Zhao, Hongbin, Chen, Yuyin, Kong, Jianshe, Mai, Wanping, Li, Lian-Sheng, Pippel, Daniel J., Ren, Pingda, Deng, Xiaohu
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The p110δ structure: mechanisms for selectivity and potency of new PI(3)K inhibitors
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Published in Nature chemical biology (01.02.2010)
Published in Nature chemical biology (01.02.2010)
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