Synthesis and Pharmacological Characterization of 2‑(2,6-Dichlorophenyl)-1-((1S,3R)‑5-(3-hydroxy-3-methylbutyl)-3-(hydroxymethyl)-1-methyl-3,4-dihydroisoquinolin-2(1H)‑yl)ethan-1-one (LY3154207), a Potent, Subtype Selective, and Orally Available Positive Allosteric Modulator of the Human Dopamine D1 Receptor
Hao, Junliang, Beck, James P, Schaus, John M, Krushinski, Joseph H, Chen, Qi, Beadle, Christopher D, Vidal, Paloma, Reinhard, Matthew R, Dressman, Bruce A, Massey, Steven M, Boulet, Serge L, Cohen, Michael P, Watson, Brian M, Tupper, David, Gardinier, Kevin M, Myers, Jason, Johansson, Anette M, Richardson, Jeffery, Richards, Daniel S, Hembre, Erik J, Remick, David M, Coates, David A, Bhardwaj, Rajni M, Diseroad, Benjamin A, Bender, David, Stephenson, Greg, Wolfangel, Craig D, Diaz, Nuria, Getman, Brian G, Wang, Xu-shan, Heinz, Beverly A, Cramer, Jeff W, Zhou, Xin, Maren, Deanna L, Falcone, Julie F, Wright, Rebecca A, Mitchell, Stephen N, Carter, Guy, Yang, Charles R, Bruns, Robert F, Svensson, Kjell A
Published in Journal of medicinal chemistry (10.10.2019)
Published in Journal of medicinal chemistry (10.10.2019)
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Hao, Junliang, Beck, James, Zhou, Xin, Lackner, Gregory L, Johnston, Richard, Reinhard, Matt, Goldsmith, Paul, Hollinshead, Sean, Dehlinger, Veronique, Filla, Sandra A, Wang, Xu-shan, Richardson, Jeffery, Posada, Maria, Mohutsky, Mike, Schober, Doug, Katner, Jason S, Chen, Qi, Hu, Bingjie, Remick, David M, Coates, David A, Mathes, Brian M, Hawk, Mai K, Svensson, Kjell A, Hembre, Erik
Published in Journal of medicinal chemistry (10.03.2022)
Published in Journal of medicinal chemistry (10.03.2022)
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Synthesis, Crystallization, and Biological Evaluation of an Orally Active Prodrug of Gemcitabine
Bender, David M, Bao, Jingqi, Dantzig, Anne H, Diseroad, William D, Law, Kevin L, Magnus, Nicholas A, Peterson, Jeffrey A, Perkins, Everett J, Pu, Yangwei J, Reutzel-Edens, Susan M, Remick, David M, Starling, James J, Stephenson, Gregory A, Vaid, Radhe K, Zhang, Deyi, McCarthy, James R
Published in Journal of medicinal chemistry (26.11.2009)
Published in Journal of medicinal chemistry (26.11.2009)
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Isolation and Physical Property Optimization of an Amorphous Drug Substance Utilizing a High Surface Area Magnesium Aluminometasilicate (Neusilin(®) US2)
Allgeier, Matthew C, Piper, Jared L, Hinds, Jeremy, Yates, Matthew H, Kolodsick, Kevin J, Meury, Richard, Shaw, Bruce, Kulkarni, Mehuli R, Remick, David M
Published in Journal of pharmaceutical sciences (01.10.2016)
Published in Journal of pharmaceutical sciences (01.10.2016)
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Novel Method for the Determination of Piperazine in Pharmaceutical Drug Substances Using Hydrophilic Interaction Chromatography and Evaporative Light Scattering Detection
McClintic, Carlie, Remick, David M., Peterson, Jeffrey A., Risley, Donald S.
Published in Journal of liquid chromatography & related technologies (01.11.2003)
Published in Journal of liquid chromatography & related technologies (01.11.2003)
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Year of Publication 12.09.2024
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Year of Publication 12.09.2024
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Isolation and Physical Property Optimization of an Amorphous Drug Substance Utilizing a High Surface Area Magnesium Aluminometasilicate (Neusilin® US2)
Allgeier, Matthew C., Piper, Jared L., Hinds, Jeremy, Yates, Matthew H., Kolodsick, Kevin J., Meury, Richard, Shaw, Bruce, Kulkarni, Mehuli R., Remick, David M.
Published in Journal of pharmaceutical sciences (01.10.2016)
Published in Journal of pharmaceutical sciences (01.10.2016)
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CDK7을 억제하는데 유용한 화합물
REMICK DAVID MICHAEL, PATEL BHARVIN KUMAR RAMESCHANDRA, YADAV VIPIN, MONTERO CARLOS, COATES DAVID ANDREW
Year of Publication 17.06.2020
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Year of Publication 17.06.2020
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