Efficacy in diet-induced obese mice of the hepatotropic, peripheral cannabinoid 1 receptor inverse agonist TM38837
Cooper, Martin E, Nørregaard, Pia K, Högberg, Thomas, Andersson, Gunnar, Receveur, Jean-Marie, Linget, Jean-Michel, Elling, Christian E
Published in British journal of pharmacology (01.10.2024)
Published in British journal of pharmacology (01.10.2024)
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Journal Article
Optimizing and characterizing 4-methyl substituted pyrazol-3-carboxamides leading to the peripheral cannabinoid 1 receptor inverse agonist TM38837
Högberg, Thomas, Receveur, Jean-Marie, Murray, Anthony, Linget, Jean-Michel, Nørregaard, Pia K., Little, Paul B., Cooper, Martin
Published in Bioorganic & medicinal chemistry letters (15.01.2024)
Published in Bioorganic & medicinal chemistry letters (15.01.2024)
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Journal Article
Effects of MCH and a MCH1-receptor antagonist on (palatable) food and water intake
Morens, Céline, Nørregaard, Pia, Receveur, Jean-Marie, van Dijk, Gertjan, Scheurink, Anton J.W.
Published in Brain research (16.11.2005)
Published in Brain research (16.11.2005)
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Impurity Dimethylcarbamoyl-OBt Detected in an API Induced by the Degradation of HBTU in DMF
Yang, Yi, Hansen, Lena, Sjögren, Jörgen Kjellgren, León, Ileana Rodríguez, Receveur, Jean-Marie, Badalassi, Fabrizio
Published in Organic process research & development (20.08.2021)
Published in Organic process research & development (20.08.2021)
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Journal Article
Conversion of 4-cyanomethyl-pyrazole-3-carboxamides into CB1 antagonists with lowered propensity to pass the blood–brain-barrier
Receveur, Jean-Marie, Murray, Anthony, Linget, Jean-Michel, Nørregaard, Pia K., Cooper, Martin, Bjurling, Emelie, Nielsen, Peter Aadal, Högberg, Thomas
Published in Bioorganic & medicinal chemistry letters (15.01.2010)
Published in Bioorganic & medicinal chemistry letters (15.01.2010)
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Journal Article
Exploring SAR features in diverse library of 4-cyanomethyl-pyrazole-3-carboxamides suitable for further elaborations as CB1 antagonists
Cooper, Martin, Receveur, Jean-Marie, Bjurling, Emelie, Nørregaard, Pia K., Nielsen, Peter Aadal, Sköld, Niklas, Högberg, Thomas
Published in Bioorganic & medicinal chemistry letters (2010)
Published in Bioorganic & medicinal chemistry letters (2010)
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Journal Article
Novel selective thiazoleacetic acids as CRTH2 antagonists developed from in silico derived hits. Part 1
Rist, Øystein, Grimstrup, Marie, Receveur, Jean-Marie, Frimurer, Thomas M., Ulven, Trond, Kostenis, Evi, Högberg, Thomas
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
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Journal Article
6-Acylamino-2-aminoquinolines as Potent Melanin-Concentrating Hormone 1 Receptor Antagonists. Identification, Structure−Activity Relationship, and Investigation of Binding Mode
Ulven, Trond, Frimurer, Thomas M, Receveur, Jean-Marie, Little, Paul Brian, Rist, Øystein, Nørregaard, Pia K, Högberg, Thomas
Published in Journal of medicinal chemistry (08.09.2005)
Published in Journal of medicinal chemistry (08.09.2005)
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Exploration of SAR features by modifications of thiazoleacetic acids as CRTH2 antagonists
Grimstrup, Marie, Receveur, Jean-Marie, Rist, Øystein, Frimurer, Thomas M., Nielsen, Peter Aadal, Mathiesen, Jesper M., Högberg, Thomas
Published in Bioorganic & medicinal chemistry letters (01.03.2010)
Published in Bioorganic & medicinal chemistry letters (01.03.2010)
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Journal Article
Novel selective thiazoleacetic acids as CRTH2 antagonists developed from in silico derived hits. Part 2
Grimstrup, Marie, Rist, Øystein, Receveur, Jean-Marie, Frimurer, Thomas M., Ulven, Trond, Mathiesen, Jesper M., Kostenis, Evi, Högberg, Thomas
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
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Journal Article
Novel Selective Orally Active CRTH2 Antagonists for Allergic Inflammation Developed from in Silico Derived Hits
Ulven, Trond, Receveur, Jean-Marie, Grimstrup, Marie, Rist, Øystein, Frimurer, Thomas M, Gerlach, Lars-Ole, Mathiesen, Jesper Mosolff, Kostenis, Evi, Uller, Lena, Högberg, Thomas
Published in Journal of medicinal chemistry (16.11.2006)
Published in Journal of medicinal chemistry (16.11.2006)
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Discovery of novel, orally available benzimidazoles as melanin concentrating hormone receptor 1 (MCHR1) antagonists
Sasmal, Pradip K., Sasmal, Sanjita, Rao, P. Tirumala, Venkatesham, B., Roshaiah, M., Abbineni, Chandrasekhar, Khanna, Ish, Jadhav, Vikram P., Suresh, J., Talwar, Rashmi, Muzeeb, Syed, Receveur, Jean-Marie, Frimurer, Thomas M., Rist, Øystein, Elster, Lisbeth, Högberg, Thomas
Published in Bioorganic & medicinal chemistry letters (15.09.2010)
Published in Bioorganic & medicinal chemistry letters (15.09.2010)
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Journal Article
4-Acylamino- and 4-ureidobenzamides as melanin-concentrating hormone (MCH) receptor 1 antagonists
RECEVEUR, Jean-Marie, BJURLING, Emelie, ULVEN, Trond, LITTLE, Paul Brian, NØRREGAARD, Pia K, HÖGBERG, Thomas
Published in Bioorganic & medicinal chemistry letters (18.10.2004)
Published in Bioorganic & medicinal chemistry letters (18.10.2004)
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Journal Article
6-Acylamino-2-amino-4-methylquinolines as potent melanin-concentrating hormone 1 receptor antagonists: Structure–activity exploration of eastern and western parts
Ulven, Trond, Little, Paul Brian, Receveur, Jean-Marie, Frimurer, Thomas M., Rist, Øystein, Nørregaard, Pia K., Högberg, Thomas
Published in Bioorganic & medicinal chemistry letters (15.02.2006)
Published in Bioorganic & medicinal chemistry letters (15.02.2006)
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Journal Article
An in vitro investigation into conformational aspects of gabapentin
Bryans, Justin S., Horwell, David C., Ratcliffe, Giles S., Receveur, Jean-Marie, Rubin, J.Ronald
Published in Bioorganic & medicinal chemistry (01.05.1999)
Published in Bioorganic & medicinal chemistry (01.05.1999)
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Journal Article
CANNABINOID RECEPTOR MODULATORS
NIELSEN PETER AADAL, ALMHOLT DORTHE, MURRAY ANTHONY, NOERREGAARD PIA KARINA, BJURLING EMELIE, HOEGBERG THOMAS, RECEVEUR JEAN MARIE, LINGET JEAN MICHEL
Year of Publication 18.08.2010
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Year of Publication 18.08.2010
Patent
BICYCLIC AMINO ACIDS AS PHARMACEUTICAL AGENTS
OSBORNE SIMON, RECEVEUR JEAN MARIE, BRYANS JUSTIN STEPHEN, BLAKEMORE DAVID CLIVE
Year of Publication 13.02.2006
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Year of Publication 13.02.2006
Patent
ChemInform Abstract: Conversion of 4-Cyanomethyl-pyrazole-3-carboxamides into CB1 Antagonists with Lowered Propensity to Pass the Blood-Brain-Barrier
Receveur, Jean-Marie, Murray, Anthony, Linget, Jean-Michel, Noerregaard, Pia K., Cooper, Martin, Bjurling, Emelie, Nielsen, Peter Aadal, Hoegberg, Thomas
Published in ChemInform (08.06.2010)
Published in ChemInform (08.06.2010)
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