Selective ortho-Bromination of Substituted Benzaldoximes Using Pd-Catalyzed C–H Activation: Application to the Synthesis of Substituted 2-Bromobenzaldehydes
Dubost, Emmanuelle, Fossey, Christine, Cailly, Thomas, Rault, Sylvain, Fabis, Frederic
Published in Journal of organic chemistry (05.08.2011)
Published in Journal of organic chemistry (05.08.2011)
Get full text
Journal Article
Discovery of Bis-Imidazoline Derivatives as New CXCR4 Ligands
Zhou, Zhicheng, Staropoli, Isabelle, Brelot, Anne, Suzanne, Peggy, Lesnard, Aurélien, Fontaine, Fanny, Perato, Serge, Rault, Sylvain, Helynck, Olivier, Arenzana-Seisdedos, Fernando, Sopkova-de Oliveira Santos, Jana, Lagane, Bernard, Munier-Lehmann, Hélène, Colin, Philippe
Published in Molecules (Basel, Switzerland) (24.01.2023)
Published in Molecules (Basel, Switzerland) (24.01.2023)
Get full text
Journal Article
Synthesis and Structure–Affinity Relationships of Selective High-Affinity 5‑HT4 Receptor Antagonists: Application to the Design of New Potential Single Photon Emission Computed Tomography Tracers
Dubost, Emmanuelle, Dumas, Noé, Fossey, Christine, Magnelli, Rosa, Butt-Gueulle, Sabrina, Ballandonne, Céline, Caignard, Daniel H, Dulin, Fabienne, Sopkova de-Oliveira Santos, Jana, Millet, Philippe, Charnay, Yves, Rault, Sylvain, Cailly, Thomas, Fabis, Frederic
Published in Journal of medicinal chemistry (26.11.2012)
Published in Journal of medicinal chemistry (26.11.2012)
Get full text
Journal Article
Two-Step Synthesis of Substituted 3-Aminoindazoles from 2-Bromobenzonitriles
Lefebvre, Valerie, Cailly, Thomas, Fabis, Frederic, Rault, Sylvain
Published in Journal of organic chemistry (16.04.2010)
Published in Journal of organic chemistry (16.04.2010)
Get full text
Journal Article
(6-bromo-1,4-dimethyl-9H-carbazol-3-yl-methylene)-hydrazine (carbhydraz) acts as a GPER agonist in breast cancer cells
Sinicropi, Maria Stefania, Lappano, Rosamaria, Caruso, Anna, Santolla, Maria Francesca, Pisano, Assunta, Rosano, Camillo, Capasso, Anna, Panno, Antonella, Lancelot, Jean Charles, Rault, Sylvain, Saturnino, Carmela, Maggiolini, Marcello
Published in Current topics in medicinal chemistry (01.01.2015)
Published in Current topics in medicinal chemistry (01.01.2015)
Get more information
Journal Article
Use of allostery to identify inhibitors of calmodulin-induced activation of Bacillus anthracis edema factor
Laine, Elodie, Goncalves, Christophe, Karst, Johanna C., Lesnard, Aurélien, Rault, Sylvain, Tang, Wei-Jen, Malliavin, Thérèse E., Ladant, Daniel, Blondel, Arnaud, Kuriyan, John
Published in Proceedings of the National Academy of Sciences - PNAS (22.06.2010)
Published in Proceedings of the National Academy of Sciences - PNAS (22.06.2010)
Get full text
Journal Article
Sonogashira cross-coupling reaction in 4-chloro-2-trichloromethylquinazoline series is possible despite a side dimerization reaction
Kieffer, Charline, Verhaeghe, Pierre, Primas, Nicolas, Castera-Ducros, Caroline, Gellis, Armand, Rosas, Roselyne, Rault, Sylvain, Rathelot, Pascal, Vanelle, Patrice
Published in Tetrahedron (08.04.2013)
Published in Tetrahedron (08.04.2013)
Get full text
Journal Article
Synthesis and in vitro antiplasmodial evaluation of 4-anilino-2-trichloromethylquinazolines
VERHAEGHE, Pierre, AZAS, Nadine, VANELLE, Patrice, HUTTER, Sébastien, CASTERA-DUCROS, Caroline, LAGET, Michèle, DUMETRE, Aurélien, GASQUET, Monique, REBOUL, Jean-Pierre, RAULT, Sylvain, RATHELOT, Pascal
Published in Bioorganic & medicinal chemistry (01.07.2009)
Published in Bioorganic & medicinal chemistry (01.07.2009)
Get full text
Journal Article
Intramolecular cyclisation of β-aryl-β-amino acids in the design of novel heterocyclic systems with therapeutic interest: an unfailing source of diversity
Rochais, Christophe, Rault, Sylvain, Dallemagne, Patrick
Published in Current medicinal chemistry (01.12.2010)
Published in Current medicinal chemistry (01.12.2010)
Get more information
Journal Article
A general synthesis of halo-oligopyridines. The Garlanding concept
Voisin-Chiret, Anne Sophie, Bouillon, Alexandre, Burzicki, Grégory, Célant, Melanie, Legay, Rémi, El-Kashef, Hussein, Rault, Sylvain
Published in Tetrahedron (01.01.2009)
Published in Tetrahedron (01.01.2009)
Get full text
Journal Article
Tripentones: a promising series of potent anti-cancer agents
Rochais, Christophe, Dallemagne, Patrick, Rault, Sylvain
Published in Anti-cancer agents in medicinal chemistry (01.05.2009)
Published in Anti-cancer agents in medicinal chemistry (01.05.2009)
Get more information
Journal Article
One-pot synthesis of new aza- and diaza-aminophenanthrenes
Rochais, Christophe, Yougnia, Rodrigue, Cailly, Thomas, Sopková-de Oliveira Santos, Jana, Rault, Sylvain, Dallemagne, Patrick
Published in Tetrahedron (12.08.2011)
Published in Tetrahedron (12.08.2011)
Get full text
Journal Article
Review of 5-HT4R ligands: state of art and clinical applications
Bureau, Ronan, Boulouard, Michel, Dauphin, François, Lezoualc'h, Frank, Rault, Sylvain
Published in Current topics in medicinal chemistry (01.04.2010)
Published in Current topics in medicinal chemistry (01.04.2010)
Get more information
Journal Article
Synthesis of novel halopyridinylboronic acids and esters. Part 4: Halopyridin-2-yl-boronic acids and esters are stable, crystalline partners for classical Suzuki cross-coupling
Bouillon, Alexandre, Lancelot, Jean-Charles, Sopkova de Oliveira Santos, Jana, Collot, Valérie, Bovy, Philipppe R, Rault, Sylvain
Published in Tetrahedron (08.12.2003)
Published in Tetrahedron (08.12.2003)
Get full text
Journal Article
A new synthetic route to original sulfonamide derivatives in 2-trichloromethylquinazoline series: a structure-activity relationship study of antiplasmodial activity
Primas, Nicolas, Verhaeghe, Pierre, Cohen, Anita, Kieffer, Charline, Dumètre, Aurélien, Hutter, Sébastien, Rault, Sylvain, Rathelot, Pascal, Azas, Nadine, Vanelle, Patrice
Published in Molecules (Basel, Switzerland) (05.07.2012)
Published in Molecules (Basel, Switzerland) (05.07.2012)
Get full text
Journal Article