Catalysis by Amberlite IR-120 resin: a rapid and green method for the synthesis of phenols from arylboronic acids under metal, ligand, and base-free conditions
Mulakayala, Naveen, Ismail, Kumar, Kottur Mohan, Rapolu, Rajesh Kumar, Kandagatla, Bhaskar, Rao, Pallavi, Oruganti, Srinivas, Pal, Manojit
Published in Tetrahedron letters (07.11.2012)
Published in Tetrahedron letters (07.11.2012)
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Journal Article
InCl3-catalysed synthesis of 2-aryl quinazolin-4(3H)-ones and 5-aryl pyrazolo[4,3-d]pyrimidin-7(6H)-ones and their evaluation as potential anticancer agents
Mulakayala, Naveen, Kandagatla, Bhaskar, Ismail, Rapolu, Rajesh Kumar, Rao, Pallavi, Mulakayala, Chaitanya, Kumar, Chitta Suresh, Iqbal, Javed, Oruganti, Srinivas
Published in Bioorganic & medicinal chemistry letters (01.08.2012)
Published in Bioorganic & medicinal chemistry letters (01.08.2012)
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Journal Article
Novel method for the synthesis of Sulfonamide Urea’s from p-toluene sulfonyl isocyanate using Amberlite IRA-400 Cl resin: Application towards the synthesis of Gliclazide
Sadineni, Ravi Kumar, Rapolu, Rajesh Kumar, Raju, V.V.N.K.V. Prasada, Navuluri, Srinivasu, Malladi, Sireesha, Mulakayala, Naveen
Published in Results in Chemistry (01.01.2021)
Published in Results in Chemistry (01.01.2021)
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Journal Article
Novel method for the synthesis of lenvatinib using 4-nitrophenyl cyclopropylcarbamate and their pharmaceutical salts
Sadineni, Ravi Kumar, Rapolu, Rajesh Kumar, Raju, V. V. N. K. V. Prasada, Srinivasu, N., Malladi, Sireesha, Mulakayala, Naveen
Published in Chemical papers (01.04.2021)
Published in Chemical papers (01.04.2021)
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Journal Article
A diastereoselective synthesis of boceprevir's gem-dimethyl bicyclic [3.1.0] proline intermediate from an insecticide ingredient cis-cypermethric acid
Kallam, Srinivasa Reddy, Eda, Vishnuvardhan Reddy, Sen, Saikat, Datrika, Rajender, Rapolu, Rajesh Kumar, Khobare, Sandip, Gajare, Vikas, Banda, Malavika, Khan, Rashid Abdul Rehman, Singh, Manpreet, Lloyd, Michael, Kandagatla, Bhaskar, Janagili, Moses Babu, Tadikonda, Veerabhadra Pratap, Vidavalur, Siddaiah, Iqbal, Javed, Fox, Martin E., Dahanukar, Vilas H., Oruganti, Srinivas
Published in Tetrahedron (27.07.2017)
Published in Tetrahedron (27.07.2017)
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Journal Article
A morpholine-free process amenable convergent synthesis of apixaban: a potent factor Xa inhibitor
Nevuluri, Narasimha Rao, Rapolu, Rajesh Kumar, Iqbal, Javed, Kandagatla, Bhaskar, Sen, Saikat, Dahanukar, Vilas H., Oruganti, Srinivas
Published in Monatshefte für Chemie (01.08.2017)
Published in Monatshefte für Chemie (01.08.2017)
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Journal Article
Silica sulfuric acid: a reusable solid catalyst for the synthesis of N-substituted amides via the Ritter reaction
Rapolu, Rajesh Kumar, NabaMukul, Buragohain, Bommineni, Srinath Reddy, Potham, Rajender, Mulakayala, Naveen, Oruganti, Srinivas
Published in RSC advances (01.01.2013)
Published in RSC advances (01.01.2013)
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Journal Article
Silica sulfuric acid: a reusable solid catalyst for the synthesis of N-substituted amides viathe Ritter reaction
Rapolu, Rajesh Kumar, NabaMukul, Buragohain, Bommineni, Srinath Reddy, Potham, Rajender, Mulakayala, Naveen, Oruganti, Srinivas
Published in RSC advances (01.03.2013)
Published in RSC advances (01.03.2013)
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Journal Article
PROCESS FOR THE PREPARATION OF INDOLINE COMPOUND
RAPOLU, Rajesh Kumar, VETUKURI, Prasada Raju VNKV, CHIGURUPATI, Krishna Prasad, BHUPATHI, Rajasekhar
Year of Publication 07.06.2018
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Year of Publication 07.06.2018
Patent
CRYSTALLINE ERTUGLIFLOZIN PROCESS
RAPOLU, Rajesh Kumar, VNKV VETUKURI, Prasada Raju, CHIGURUPATI, Krishna Prasad, GILLA, Goverdhan, BHUPATHI, Rajasekhar
Year of Publication 29.03.2018
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Year of Publication 29.03.2018
Patent
NOVEL POLYMORPHIC FORMS OF ((1S,2S,3S,4R,5S))-2,3,4-(TRIS-BENZYLOXY)-5-(4-CHLORO-3-(4-ETHOXY-BENZYL)PHENYL)-6,8-DIOXA-BICYCLO[3.2.1]OCT-1-YL-METHANOL
RAPOLU, Rajesh Kumar, VETUKURI, Prasada Raju Vnkv, CHIGURUPATI, Krishna Prasad, GILLA, Goverdhan, BHUPATHI, Rajashekar
Year of Publication 18.01.2018
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Year of Publication 18.01.2018
Patent
AN IMPROVED PROCESS FOR THE PREPARATION OF HCV INHIBITOR
RAPOLU RAJESH KUMAR, GILLA GOVERDHAN, CHIGURUPATI KRISHNA PRASAD, VETUKURI PRASAD RAJU VNKV
Year of Publication 11.01.2018
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Year of Publication 11.01.2018
Patent
TEMOZOLOMIDE PROCESS
CHATURVEDI, Akshay Kant, RAPOLU, Rajesh Kumar, NARAYANA, Rama Krishna Reddy, VETUKURI, Prasada Raju VNKV, CHIGURUPATI, Krishna Prasad
Year of Publication 05.07.2018
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Year of Publication 05.07.2018
Patent
AN IMPROVED PROCESS FOR THE PREPARATION OF HCV INHIBITOR
GILLA, GOVERDHAN, RAPOLU, RAJESH KUMAR, CHIGURUPATI, KRISHNA PRASAD, VETUKURI, PRASADA RAJU VNKV
Year of Publication 30.06.2016
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Year of Publication 30.06.2016
Patent
ChemInform Abstract: Catalysis by Amberlite IR-120 Resin: A Rapid and Green Method for the Synthesis of Phenols from Arylboronic Acids under Metal, Ligand, and Base-Free Conditions
Mulakayala, Naveen, Ismail, Ismail, Kumar, Kottur Mohan, Rapolu, Rajesh Kumar, Kandagatla, Bhaskar, Rao, Pallavi, Oruganti, Srinivas, Pal, Manojit
Published in ChemInform (05.02.2013)
Published in ChemInform (05.02.2013)
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Journal Article
PREPARATION OF TICAGRELOR
DAHANUKAR, VILAS, RAPOLU, RAJESH KUMAR, ELATI, RAVI RAM CHANDRASEKHAR, ORUGANTI, SRINIVAS, KURELLA, SREENIVASULU
Year of Publication 07.01.2016
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Year of Publication 07.01.2016
Patent
ChemInform Abstract: InCl3-Catalyzed Synthesis of 2-Aryl Quinazolin-4(3H)-ones and 5-Aryl Pyrazolo[4,3-d]pyrimidin-7(6H)-ones and Their Evaluation as Potential Anticancer Agents
Mulakayala, Naveen, Kandagatla, Bhaskar, Ismail, Ismail, Rapolu, Rajesh Kumar, Rao, Pallavi, Mulakayala, Chaitanya, Kumar, Chitta Suresh, Iqbal, Javed, Oruganti, Srinivas
Published in ChemInform (18.12.2012)
Published in ChemInform (18.12.2012)
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Journal Article
ChemInform Abstract: InCl 3 ‐Catalyzed Synthesis of 2‐Aryl Quinazolin‐4(3H)‐ones and 5‐Aryl Pyrazolo[4,3‐d]pyrimidin‐7(6H)‐ones and Their Evaluation as Potential Anticancer Agents
Mulakayala, Naveen, Kandagatla, Bhaskar, Ismail, Ismail, Rapolu, Rajesh Kumar, Rao, Pallavi, Mulakayala, Chaitanya, Kumar, Chitta Suresh, Iqbal, Javed, Oruganti, Srinivas
Published in ChemInform (18.12.2012)
Published in ChemInform (18.12.2012)
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Journal Article