Discovery of SCH 900271, a Potent Nicotinic Acid Receptor Agonist for the Treatment of Dyslipidemia
Palani, Anandan, Rao, Ashwin U, Chen, Xiao, Huang, Xianhai, Su, Jing, Tang, Haiqun, Huang, Ying, Qin, Jun, Xiao, Dong, Degrado, Sylvia, Sofolarides, Michael, Zhu, Xiaohong, Liu, Zhidan, McKittrick, Brian, Zhou, Wei, Aslanian, Robert, Greenlee, William J, Senior, Mary, Cheewatrakoolpong, Boonlert, Zhang, Hongtao, Farley, Constance, Cook, John, Kurowski, Stan, Li, Qiu, van Heek, Margaret, Wang, Gangfeng, Hsieh, Yunsheng, Li, Fangbiao, Greenfeder, Scott, Chintala, Madhu
Published in ACS medicinal chemistry letters (12.01.2012)
Published in ACS medicinal chemistry letters (12.01.2012)
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Journal Article
Facile synthesis of tetracyclic azepine and oxazocine derivatives and their potential as MAPKAP-K2 (MK2) inhibitors
Rao, Ashwin U., Xiao, Dong, Huang, Xianhai, Zhou, Wei, Fossetta, James, Lundell, Dan, Tian, Fang, Trivedi, Prashant, Aslanian, Robert, Palani, Anandan
Published in Bioorganic & medicinal chemistry letters (15.01.2012)
Published in Bioorganic & medicinal chemistry letters (15.01.2012)
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Journal Article
Synthesis and structure-activity relationships of 2-(1,4'-bipiperidin-1'-yl) thiazolopyridine as H3 receptor antagonists
RAO, Ashwin U, PALANI, Anandan, LACHOWICZ, Jean, XIAO CHEN, YING HUANG, ASLANIAN, Robert G, WEST, Robert E, WILLIAMS, Shirley M, WU, Ren-Long, HWA, Joyce, SONDEY, Christopher
Published in Bioorganic & medicinal chemistry letters (01.11.2009)
Published in Bioorganic & medicinal chemistry letters (01.11.2009)
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Journal Article
SAR studies of C2 ethers of 2H-pyrano[2,3-d]pyrimidine-2,4,7(1H,3H)-triones as nicotinic acid receptor (NAR) agonist
Huang, Xianhai, Su, Jing, Rao, Ashwin U., Tang, Haiqun, Zhou, Wei, Zhu, Xiaohong, Chen, Xiao, Liu, Zhidan, Huang, Ying, Degrado, Sylvia, Xiao, Dong, Qin, Jun, Aslanian, Robert, McKittrick, Brian A., Greenfeder, Scott, Heek, Margaret van, Chintala, Madhu, Palani, Anandan
Published in Bioorganic & medicinal chemistry letters (15.01.2012)
Published in Bioorganic & medicinal chemistry letters (15.01.2012)
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Journal Article
Discovery of a Potent Thiadiazole Class of Histamine H3 Receptor Antagonist for the Treatment of Diabetes
Rao, Ashwin U, Shao, Ning, Aslanian, Robert G, Chan, Tin-Yau, Degrado, Sylvia J, Wang, Li, McKittrick, Brian, Senior, Mary, West, Robert E, Williams, Shirley M, Wu, Ren-Long, Hwa, Joyce, Patel, Bhuneshwari, Zheng, Shuqin, Sondey, Christopher, Palani, Anandan
Published in ACS medicinal chemistry letters (08.03.2012)
Published in ACS medicinal chemistry letters (08.03.2012)
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Journal Article
Synthesis and structure–activity relationships of 2-(1,4′-bipiperidin-1′-yl)thiazolopyridine as H 3 receptor antagonists
Rao, Ashwin U., Palani, Anandan, Chen, Xiao, Huang, Ying, Aslanian, Robert G., West, Robert E., Williams, Shirley M., Wu, Ren-Long, Hwa, Joyce, Sondey, Christopher, Lachowicz, Jean
Published in Bioorganic & medicinal chemistry letters (01.11.2009)
Published in Bioorganic & medicinal chemistry letters (01.11.2009)
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Journal Article
Discovery of a Potent Thiadiazole Class of Histamine H-3 Receptor Antagonist for the Treatment of Diabetes
Rao, Ashwin U., Shao, Ning, Aslanian, Robert G., Chan, Tin-Yau, Degrado, Sylvia J., Wang, Li, McKittrick, Brian, Senior, Mary, West, Robert E., Williams, Shirley M., Wu, Ren-Long, Hwa, Joyce, Patel, Bhuneshwari, Zheng, Shuqin, Sondey, Christopher, Palani, Anandan
Published in ACS medicinal chemistry letters (08.03.2012)
Published in ACS medicinal chemistry letters (08.03.2012)
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Journal Article
Synthesis and structure-activity relationships of 2-(1,4'-bipiperidin-1'-yl)thiazolopyridine as H sub(3) receptor antagonists
Rao, Ashwin U, Palani, Anandan, Chen, Xiao, Huang, Ying, Aslanian, Robert G, West, Robert E, Williams, Shirley M, Wu, Ren-Long, Sondey, Christopher, Lachowicz, Jean
Published in Bioorganic & medicinal chemistry letters (01.11.2009)
Published in Bioorganic & medicinal chemistry letters (01.11.2009)
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Journal Article
FUSED PYRAZOLE UREA ANALOGS AS GLUCOSYLCERAMIDE SYNTHASE INHIBITORS
LOUGHRAN, H. Marie, RAO, Ashwin, U, TONG, Ling, LIANG, Tao, SCHIRRIPA, Kathy, M, FRALEY, Mark, E, ROECKER, Anthony, J
Year of Publication 09.10.2024
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Year of Publication 09.10.2024
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CYCLIC PEPTIDES FOR INHIBITING TNF RECEPTOR 1 ACTIVITY
Zultanski, Susan L, Mapelli, Claudio, Kekec, Ahmet, Boyer, Nicolas C, Biswas, Kaustav, Frost, John R, Chau, Ryan, Sindhikara, Daniel J, Ding, Fa-Xiang, Siu, Tony, Pasquini, Nicolo Maria, Haidle, Andrew M, Rao, Ashwin U, Gambini, Luca, Wan, Murray, Lee, Hu-Jung Julie, Jewell, James P, Zhu, Yuping, Wuo, Michael, Tozzi, Roberta, Cash, Brandon D, Garrigou, Michael B, Lin, Songnian, Proietti, Giordano, Orvieto, Federica, Abate, Luigi
Year of Publication 29.08.2024
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Year of Publication 29.08.2024
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CYCLIC PEPTIDES FOR INHIBITING TNF RECEPTOR 1 ACTIVITY
HAIDLE, Andrew M, ZHU, Yuping, WUO, Michael, ZULTANSKI, Susan L, FROST, John R, JEWELL, James P, DING, Fa-Xiang, GARRIGOU, Michael B, LIN, Songnian, ORVIETO, Federica, GAMBINI, Luca, SIU, Tony, LEE, Hu-Jung Julie, BOYER, Nicolas C, BISWAS, Kaustav, TOZZI, Roberta, KEKEC, Ahmet, ABATE, Luigi, RAO, Ashwin U, PASQUINI, Nicolo Maria, CHAU, Ryan, CASH, Brandon D, SINDHIKARA, Daniel J, MAPELLI, Claudio, PROIETTI, Giordano, WAN, Murray
Year of Publication 08.08.2024
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Year of Publication 08.08.2024
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SUBSTITUTED ISOQUINOLINES AS CRTH2 RECEPTOR MODULATORS
HUANG, Xianhai, RAO, Ashwin, U, PALANI, Anandan, ZHOU, Wei, ZHANG, Hongjun
Year of Publication 15.01.2020
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Year of Publication 15.01.2020
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FACTOR XIIA INHIBITORS
HICKS, Jacqueline, D, SO, Sung-Sau, MCCRACKEN, Amy Bittner, DAHLGREN, Markus, K, WHITEHEAD, Brent, R, TAYLOR, Jerry, A, BHAT, Sathesh, P, LOMBARDO, Matthew, KATIPALLY, Revathi Reddy, GABLE, Jonathan, E, RAO, Ashwin, U, MCKITTRICK, Brian Alexander, LAN, Ping, SUN, Zhongxiang, ORTH, Peter, WU, Zhicai, DEBENHAM, John, S, CHU, Hong Dong
Year of Publication 23.08.2023
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Year of Publication 23.08.2023
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Factor XIIa inhibitors
Taylor, Jerry A, Orth, Peter, Debenham, John S, Dahlgren, Markus K, McKittrick, Brian Alexander, Chu, Hong Dong, Wu, Zhicai, So, Sung-Sau, Sun, Zhongxiang, Whitehead, Brent R, Gable, Jonathan E, Lombardo, Matthew, Hicks, Jacqueline D, Lan, Ping, Bhat, Sathesh P, Bittner McCracken, Amy, Katipally, Revathi Reddy, Rao, Ashwin U
Year of Publication 29.12.2020
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Year of Publication 29.12.2020
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PIPERIDINE DERIVATIVES AS NK1 ANTAGONISTS
HUANG, Xianhai, PALIWAL, Sunil, PALANI, Anandan, RAO, Ashwin U, XIAO, Dong, SHAH, Sapna S, SHIH, Neng-Yang, WANG, Cheng, WROBLESKI, Michelle Laci, TSUI, Hon-Chung
Year of Publication 20.12.2018
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Year of Publication 20.12.2018
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NK 1 ANTAGONISTS
HUANG, Xianhai, PALIWAL, Sunil, PALANI, Anandan, RAO, Ashwin U, XIAO, Dong, SHAH, Sapna S, SHIH, Neng-Yang, WANG, Cheng, WROBLESKI, Michelle Laci, TSUI, Hon-Chung
Year of Publication 02.08.2018
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Year of Publication 02.08.2018
Patent
FACTOR XIIa INHIBITORS
HICKS, Jacqueline, D, SO, Sung-Sau, MCCRACKEN, Amy Bittner, DAHLGREN, Markus, K, WHITEHEAD, Brent, R, TAYLOR, Jerry, A, BHAT, Sathesh, P, LOMBARDO, Matthew, KATIPALLY, Revathi Reddy, GABLE, Jonathan, E, RAO, Ashwin, U, MCKITTRICK, Brian Alexander, LAN, Ping, SUN, Zhongxiang, ORTH, Peter, WU, Zhicai, DEBENHAM, John, S, CHU, Hong Dong
Year of Publication 13.05.2020
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Year of Publication 13.05.2020
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NK1 antagonists
Wrobleski, Michelle Laci, Huang, Xianhai, Paliwal, Sunil, Palani, Anandan, Tsui, Hon-Chung, Shih, Neng-Yang, Wang, Cheng, Shah, Sapna S, Rao, Ashwin U, Xiao, Dong
Year of Publication 15.05.2018
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Year of Publication 15.05.2018
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SUBSTITUTED ISOQUINOLINES AS CRTH2 RECEPTOR MODULATORS
RAO, ASHWIN, U, ZHANG, HONGJUN, ZHOU, WEI, HUANG, XIANHAI, PALANI, ANANDAN
Year of Publication 20.04.2016
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Year of Publication 20.04.2016
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