Rapid Discovery of a Novel Series of Abl Kinase Inhibitors by Application of an Integrated Microfluidic Synthesis and Screening Platform
Desai, Bimbisar, Dixon, Karen, Farrant, Elizabeth, Feng, Qixing, Gibson, Karl R, van Hoorn, Willem P, Mills, James, Morgan, Trevor, Parry, David M, Ramjee, Manoj K, Selway, Christopher N, Tarver, Gary J, Whitlock, Gavin, Wright, Adrian G
Published in Journal of medicinal chemistry (11.04.2013)
Published in Journal of medicinal chemistry (11.04.2013)
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The background, discovery and clinical development of BCR-ABL inhibitors
Lambert, Gemma K., Duhme-Klair, Anne-Kathrin, Morgan, Trevor, Ramjee, Manoj K.
Published in Drug discovery today (01.10.2013)
Published in Drug discovery today (01.10.2013)
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Design, Synthesis, and Testing of Potent, Selective Hepsin Inhibitors via Application of an Automated Closed-Loop Optimization Platform
Pant, Shishir M, Mukonoweshuro, Amanda, Desai, Bimbisar, Ramjee, Manoj K, Selway, Christopher N, Tarver, Gary J, Wright, Adrian G, Birchall, Kristian, Chapman, Timothy M, Tervonen, Topi A, Klefström, Juha
Published in Journal of medicinal chemistry (24.05.2018)
Published in Journal of medicinal chemistry (24.05.2018)
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Integrated Synthesis and Testing of Substituted Xanthine Based DPP4 Inhibitors: Application to Drug Discovery
Czechtizky, Werngard, Dedio, Jüergen, Desai, Bimbisar, Dixon, Karen, Farrant, Elizabeth, Feng, Qixing, Morgan, Trevor, Parry, David M, Ramjee, Manoj K, Selway, Christopher N, Schmidt, Thorsten, Tarver, Gary J, Wright, Adrian G
Published in ACS medicinal chemistry letters (08.08.2013)
Published in ACS medicinal chemistry letters (08.08.2013)
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Substrate mapping and inhibitor profiling of falcipain-2, falcipain-3 and berghepain-2: implications for peptidase anti-malarial drug discovery
Ramjee, Manoj K, Flinn, Nicholas S, Pemberton, Tracy P, Quibell, Martin, Wang, Yikang, Watts, John P
Published in Biochemical journal (01.10.2006)
Published in Biochemical journal (01.10.2006)
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The thrombogram: monitoring thrombin generation in platelet-rich plasma
Hemker, H C, Giesen, P L, Ramjee, M, Wagenvoord, R, Béguin, S
Published in Thrombosis and haemostasis (01.04.2000)
Published in Thrombosis and haemostasis (01.04.2000)
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Bicyclic peptidomimetic tetrahydrofuro[3,2- b]pyrrol-3-one and hexahydrofuro[3,2- b]pyridine-3-one based scaffolds: synthesis and cysteinyl proteinase inhibition
Quibell, Martin, Benn, Alex, Flinn, Nick, Monk, Tracy, Ramjee, Manoj, Wang, Yikang, Watts, John
Published in Bioorganic & medicinal chemistry (01.11.2004)
Published in Bioorganic & medicinal chemistry (01.11.2004)
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Novel Chemoselective Linkage Chemistry toward Controlled Loading of Ligands to Proteins through In Situ Real-Time Quantification of Conjugate Formation
Flinn, Nicholas S, Quibell, Martin, Turnell, William G, Monk, Tracy P, Ramjee, Manoj K
Published in Bioconjugate chemistry (01.09.2004)
Published in Bioconjugate chemistry (01.09.2004)
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Selective Phenylimidazole-Based Inhibitors of the Mycobacterium tuberculosis Proteasome
Zhan, Wenhu, Hsu, Hao-Chi, Morgan, Trevor, Ouellette, Tierra, Burns-Huang, Kristin, Hara, Ryoma, Wright, Adrian G, Imaeda, Toshihiro, Okamoto, Rei, Sato, Kenjiro, Michino, Mayako, Ramjee, Manoj, Aso, Kazuyoshi, Meinke, Peter T, Foley, Michael, Nathan, Carl F, Li, Huilin, Lin, Gang
Published in Journal of medicinal chemistry (24.10.2019)
Published in Journal of medicinal chemistry (24.10.2019)
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Crystal structure of aspartate decarboxylase at 2.2 A resolution provides evidence for an ester in protein self-processing
Albert, A, Dhanaraj, V, Genschel, U, Khan, G, Ramjee, M K, Pulido, R, Sibanda, B L, von Delft, F, Witty, M, Blundell, T L, Smith, A G, Abell, C
Published in Nature structural biology (01.04.1998)
Published in Nature structural biology (01.04.1998)
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The design and synthesis of inhibitors of the cysteinyl protease, Der p I
Billson, Jeremy, Clark, Jonathan, Conway, Simon P., Hart, Terance, Johnson, Tony, Langston, Steven P., Ramjee, Manoj, Quibell, Martin, Scott, Richard K.
Published in Bioorganic & medicinal chemistry letters (05.05.1998)
Published in Bioorganic & medicinal chemistry letters (05.05.1998)
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Spectrophotometric detection of a modified flavin mononucleotide (FMN) intermediate formed during the catalytic cycle of chorismate synthase
Ramjee, Manoj N, Coggins, John R, Hawkes, Timothy R, Lowe, David J, Thorneley, Roger N. F
Published in Journal of the American Chemical Society (01.10.1991)
Published in Journal of the American Chemical Society (01.10.1991)
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Reaction of (6R)-6-fluoroEPSP with recombinant Escherichia coli chorismate synthase generates a stable flavin mononucleotide semiquinone radical
Ramjee, Manoj N, Balasubramanian, Shankar, Abell, Chris, Coggins, John R, Davies, Gareth M, Hawkes, Timothy R, Lowe, David J, Thorneley, Roger N. F
Published in Journal of the American Chemical Society (01.04.1992)
Published in Journal of the American Chemical Society (01.04.1992)
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Escherichia coli Chorismate Synthase Catalyzes the Conversion of (6S)-6-Fluoro-5-enolpyruvylshikimate-3-phosphate to 6-Fluorochorismate
Bornemann, Stephen, Ramjee, Manoj K., Balasubramanian, Shankar, Abell, Chris, Coggins, John R., Lowe, David J., Thorneley, Roger N.F.
Published in The Journal of biological chemistry (29.09.1995)
Published in The Journal of biological chemistry (29.09.1995)
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Corrigendum to “Functionalised 2,3-dimethyl-3-aminotetrahydrofuran-4-one and N-(3-oxo-hexahydrocyclopenta[ b]furan-3 a-yl)acylamide based scaffolds: synthesis and cysteinyl proteinase inhibition” [Bioorg. Med. Chem. 12 (2004) 2903–2925]
Watts, John, Benn, Alex, Flinn, Nick, Monk, Tracy, Ramjee, Manoj, Ray, Peter, Wang, Yikang, Quibell, Martin
Published in Bioorganic & medicinal chemistry (01.09.2005)
Published in Bioorganic & medicinal chemistry (01.09.2005)
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Functionalised 2,3-dimethyl-3-aminotetrahydrofuran-4-one and N-(3-oxo-hexahydrocyclopenta[ b]furan-3 a-yl)acylamide based scaffolds: synthesis and cysteinyl proteinase inhibition
Watts, John, Benn, Alex, Flinn, Nick, Monk, Tracy, Ramjee, Manoj, Ray, Peter, Wang, Yikang, Quibell, Martin
Published in Bioorganic & medicinal chemistry (01.06.2004)
Published in Bioorganic & medicinal chemistry (01.06.2004)
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