Biochemical Evaluation of the Inhibition Properties of Favipiravir and 2'-C-Methyl-Cytidine Triphosphates against Human and Mouse Norovirus RNA Polymerases
Jin, Zhinan, Tucker, Kathryn, Lin, Xiaoyan, Kao, C Cheng, Shaw, Ken, Tan, Hua, Symons, Julian, Behera, Ishani, Rajwanshi, Vivek K, Dyatkina, Natalia, Wang, Guangyi, Beigelman, Leo, Deval, Jerome
Published in Antimicrobial agents and chemotherapy (01.12.2015)
Published in Antimicrobial agents and chemotherapy (01.12.2015)
Get full text
Journal Article
Structure-activity relationship analysis of mitochondrial toxicity caused by antiviral ribonucleoside analogs
Jin, Zhinan, Kinkade, April, Behera, Ishani, Chaudhuri, Shuvam, Tucker, Kathryn, Dyatkina, Natalia, Rajwanshi, Vivek K., Wang, Guangyi, Jekle, Andreas, Smith, David B., Beigelman, Leo, Symons, Julian A., Deval, Jerome
Published in Antiviral research (01.07.2017)
Published in Antiviral research (01.07.2017)
Get full text
Journal Article
Tumor Regression upon Intratumoral and Subcutaneous Dosing of the STING Agonist ALG-031048 in Mouse Efficacy Models
Jekle, Andreas, Thatikonda, Santosh Kumar, Jaisinghani, Ruchika, Ren, Suping, Kinkade, April, Stevens, Sarah K, Stoycheva, Antitsa, Rajwanshi, Vivek K, Williams, Caroline, Deval, Jerome, Mukherjee, Sucheta, Zhang, Qingling, Chanda, Sushmita, Smith, David B, Blatt, Lawrence M, Symons, Julian A, Gonzalvez, Francois, Beigelman, Leonid
Published in International journal of molecular sciences (01.11.2023)
Published in International journal of molecular sciences (01.11.2023)
Get full text
Journal Article
Distinct Effects of T-705 (Favipiravir) and Ribavirin on Influenza Virus Replication and Viral RNA Synthesis
Vanderlinden, Evelien, Vrancken, Bram, Van Houdt, Jeroen, Rajwanshi, Vivek K, Gillemot, Sarah, Andrei, Graciela, Lemey, Philippe, Naesens, Lieve
Published in Antimicrobial agents and chemotherapy (01.11.2016)
Published in Antimicrobial agents and chemotherapy (01.11.2016)
Get full text
Journal Article
Synthesis and Anti-Influenza Activity of Pyridine, Pyridazine, and Pyrimidine C‑Nucleosides as Favipiravir (T-705) Analogues
Wang, Guangyi, Wan, Jinqiao, Hu, Yujian, Wu, Xiangyang, Prhavc, Marija, Dyatkina, Natalia, Rajwanshi, Vivek K, Smith, David B, Jekle, Andreas, Kinkade, April, Symons, Julian A, Jin, Zhinan, Deval, Jerome, Zhang, Qingling, Tam, Yuen, Chanda, Sushmita, Blatt, Lawrence, Beigelman, Leonid
Published in Journal of medicinal chemistry (26.05.2016)
Published in Journal of medicinal chemistry (26.05.2016)
Get full text
Journal Article
Synthesis and Anti-HCV Activity of Sugar-Modified Guanosine Analogues: Discovery of AL-611 as an HCV NS5B Polymerase Inhibitor for the Treatment of Chronic Hepatitis C
Wang, Guangyi, Dyatkina, Natalia, Prhavc, Marija, Williams, Caroline, Serebryany, Vladimir, Hu, Yujian, Huang, Yongfei, Wu, Xiangyang, Chen, Tongqian, Huang, Wensheng, Rajwanshi, Vivek K, Deval, Jerome, Fung, Amy, Jin, Zhinan, Stoycheva, Antitsa, Shaw, Kenneth, Gupta, Kusum, Tam, Yuen, Jekle, Andreas, Smith, David B, Beigelman, Leonid
Published in Journal of medicinal chemistry (24.09.2020)
Published in Journal of medicinal chemistry (24.09.2020)
Get full text
Journal Article
LNA (Locked Nucleic Acids): Synthesis of the adenine, cytosine, guanine, 5-methylcytosine, thymine and uracil bicyclonucleoside monomers, oligomerisation, and unprecedented nucleic acid recognition
Koshkin, Alexei A., Singh, Sanjay K., Nielsen, Poul, Rajwanshi, Vivek K., Kumar, Ravindra, Meldgaard, Michael, Olsen, Carl Erik, Wengel, Jesper
Published in Tetrahedron (01.04.1998)
Published in Tetrahedron (01.04.1998)
Get full text
Journal Article
Synthesis and Biological Evaluation of 6-(Alkyn-1-yl)furo[2,3-d]pyrimidin-2(3H)-one Base and Nucleoside Derivatives
Robins, Morris J, Miranda, Karl, Rajwanshi, Vivek K, Peterson, Matt A, Andrei, Graciela, Snoeck, Robert, De Clercq, Erik, Balzarini, Jan
Published in Journal of medicinal chemistry (12.01.2006)
Published in Journal of medicinal chemistry (12.01.2006)
Get full text
Journal Article
Structural Studies of LNA:RNA Duplexes by NMR: Conformations and Implications for RNase H Activity
Bondensgaard, Kent, Petersen, Michael, Singh, Sanjay K., Rajwanshi, Vivek K., Kumar, Ravindra, Wengel, Jesper, Jacobsen, Jens Peter
Published in Chemistry : a European journal (04.08.2000)
Published in Chemistry : a European journal (04.08.2000)
Get full text
Journal Article
Synthesis of AZT 5‘-Triphosphate Mimics and Their Inhibitory Effects on HIV-1 Reverse Transcriptase
Wang, Guangyi, Boyle, Nicholas, Chen, Fu, Rajappan, Vasanthakumar, Fagan, Patrick, Brooks, Jennifer L, Hurd, Tiffany, Leeds, Janet M, Rajwanshi, Vivek K, Jin, Yi, Prhavc, Marija, Bruice, Thomas W, Cook, P. Dan
Published in Journal of medicinal chemistry (30.12.2004)
Published in Journal of medicinal chemistry (30.12.2004)
Get full text
Journal Article
Synthesis and Antiviral Evaluation of 6-(Alkyl-heteroaryl)furo[2,3-d]pyrimidin-2(3H)-one Nucleosides and Analogues with Ethynyl, Ethenyl, and Ethyl Spacers at C6 of the Furopyrimidine Core
Robins, Morris J, Nowak, Ireneusz, Rajwanshi, Vivek K, Miranda, Karl, Cannon, John F, Peterson, Matt A, Andrei, Graciela, Snoeck, Robert, De Clercq, Erik, Balzarini, Jan
Published in Journal of medicinal chemistry (09.08.2007)
Published in Journal of medicinal chemistry (09.08.2007)
Get full text
Journal Article
The conformations of locked nucleic acids (LNA)
Petersen, Michael, Nielsen, Christina B., Nielsen, Katrine E., Jensen, Gitte A., Bondensgaard, Kent, Singh, Sanjay K., Rajwanshi, Vivek K., Koshkin, Alexei A., Dahl, Britta M., Wengel, Jesper, Jacobsen, Jens Peter
Published in Journal of molecular recognition (01.01.2000)
Published in Journal of molecular recognition (01.01.2000)
Get full text
Journal Article
Synthesis of 2‘,3‘-Dideoxynucleoside 5‘-α-P-Borano-β,γ-(difluoromethylene)triphosphates and Their Inhibition of HIV-1 Reverse Transcriptase
Boyle, Nicholas A, Rajwanshi, Vivek K, Prhavc, Marija, Wang, Guangyi, Fagan, Patrick, Chen, Fu, Ewing, Gregory J, Brooks, Jennifer L, Hurd, Tiffany, Leeds, Janet M, Bruice, Thomas W, Cook, P. Dan
Published in Journal of medicinal chemistry (07.04.2005)
Published in Journal of medicinal chemistry (07.04.2005)
Get full text
Journal Article
Polyphenols and alkaloids from piper species
Parmar, Virinder S, Jain, Subhash C, Gupta, Sangita, Talwar, Sangeeta, Rajwanshi, Vivek K, Kumar, Rajesh, Azim, Abul, Malhotra, Sanjay, Kumar, Naresh, Jain, Rajni, Sharma, Nawal K, Tyagi, Om D, Lawrie, Stephen J, Errington, William, Howarth, Oliwer W, Olsen, Carl E, Wengel, Sanjay K.Singh¶andJesper
Published in Phytochemistry (Oxford) (01.10.1998)
Published in Phytochemistry (Oxford) (01.10.1998)
Get full text
Journal Article
Synthesis of 5 '-triphosphate mimics (P3Ms) of 3 '-azido-3 ',5 '-dideoxythymidine and 3 ',5 '-dideoxy-5 '-difluoromethylenethymidine as HIV-1 reverse transcriptase inhibitors
Rajwanshi, VK, Prhavc, M, Fagan, P, Brooks, JL, Hurd, T, Cook, PD, Wang, GY
Published in Nucleosides, nucleotides & nucleic acids (01.01.2005)
Published in Nucleosides, nucleotides & nucleic acids (01.01.2005)
Get full text
Journal Article