Search Results - "RAFALSKI, Maria" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Matrix metalloproteinase–activated doxorubicin prodrugs inhibit HT1080 xenograft growth better than doxorubicin with less toxicity

Matrix metalloproteinase–activated doxorubicin prodrugs inhibit HT1080 xenograft growth better than doxorubicin with less toxicity

by Albright, Charles F, Graciani, Nilsa, Han, Wei, Yue, Eddy, Stein, Ross, Lai, Zhihong, Diamond, Melody, Dowling, Randine, Grimminger, Lisa, Zhang, Shu-Yun, Behrens, Davette, Musselman, Amy, Bruckner, Robert, Zhang, Mingzhu, Jiang, Xiang, Hu, Daniel, Higley, Anne, Dimeo, Susan, Rafalski, Maria, Mandlekar, Sandya, Car, Bruce, Yeleswaram, Swamy, Stern, Andrew, Copeland, Robert A, Combs, Andrew, Seitz, Steve P, Trainor, George L, Taub, Rebecca, Huang, Pearl, Oliff, Allen
Published in Molecular cancer therapeutics (01.05.2005)

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Journal Article

Solid supported [formula omitted] CN cross-coupling reactions

Solid supported [formula omitted] CN cross-coupling reactions

by Combs, Andrew P., Saubern, Simon, Rafalski, Maria, Lam, Patrick Y.S.
Published in Tetrahedron letters (01.02.1999)

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Journal Article

Solid supported aryl/heteroaryl C-N cross-coupling reactions

Solid supported aryl/heteroaryl C-N cross-coupling reactions

by Combs, AP, Saubern, S, Rafalski, M, Lam, PYS
Published in Tetrahedron letters (26.02.1999)

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Journal Article

In Vitro Intrinsic Clearance-Based Optimization of N 3-Phenylpyrazinones as Corticotropin-Releasing Factor-1 (CRF1) Receptor Antagonists

In Vitro Intrinsic Clearance-Based Optimization of N 3-Phenylpyrazinones as Corticotropin-Releasing Factor-1 (CRF1) Receptor Antagonists

by Hartz, Richard A, Ahuja, Vijay T, Rafalski, Maria, Schmitz, William D, Brenner, Allison B, Denhart, Derek J, Ditta, Jonathan L, Deskus, Jeffrey A, Yue, Eddy W, Arvanitis, Argyrios G, Lelas, Snjezana, Li, Yu-Wen, Molski, Thaddeus F, Wong, Harvey, Grace, James E, Lentz, Kimberley A, Li, Jianqing, Lodge, Nicholas J, Zaczek, Robert, Combs, Andrew P, Olson, Richard E, Mattson, Ronald J, Bronson, Joanne J, Macor, John E
Published in Journal of medicinal chemistry (23.07.2009)

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Synthesis, Structure−Activity Relationships, and In Vivo Evaluation of N 3-Phenylpyrazinones as Novel Corticotropin-Releasing Factor-1 (CRF1) Receptor Antagonists

Synthesis, Structure−Activity Relationships, and In Vivo Evaluation of N 3-Phenylpyrazinones as Novel Corticotropin-Releasing Factor-1 (CRF1) Receptor Antagonists

by Hartz, Richard A, Ahuja, Vijay T, Arvanitis, Argyrios G, Rafalski, Maria, Yue, Eddy W, Denhart, Derek J, Schmitz, William D, Ditta, Jonathan L, Deskus, Jeffrey A, Brenner, Allison B, Hobbs, Frank W, Payne, Joseph, Lelas, Snjezana, Li, Yu-Wen, Molski, Thaddeus F, Mattson, Gail K, Peng, Yong, Wong, Harvey, Grace, James E, Lentz, Kimberley A, Qian-Cutrone, Jingfang, Zhuo, Xiaoliang, Shu, Yue-Zhong, Lodge, Nicholas J, Zaczek, Robert, Combs, Andrew P, Olson, Richard E, Bronson, Joanne J, Mattson, Ronald J, Macor, John E
Published in Journal of medicinal chemistry (23.07.2009)

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Discovery of matrix metalloproteases selective and activated peptide–doxorubicin prodrugs as anti-tumor agents

Discovery of matrix metalloproteases selective and activated peptide–doxorubicin prodrugs as anti-tumor agents

by Hu, Zilun, Jiang, Xiangjun, Albright, Charles F., Graciani, Nilsa, Yue, Eddy, Zhang, Mingzhu, Zhang, Shu-Yun, Bruckner, Robert, Diamond, Melody, Dowling, Randine, Rafalski, Maria, Yeleswaram, Swamy, Trainor, George L., Seitz, Steven P., Han, Wei
Published in Bioorganic & medicinal chemistry letters (01.02.2010)

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Journal Article

Synthesis and structure–activity relationships of pyrido[3,2-b]pyrazin-3(4H)-ones and pteridin-7(8H)-ones as corticotropin-releasing factor-1 receptor antagonists

Synthesis and structure–activity relationships of pyrido[3,2-b]pyrazin-3(4H)-ones and pteridin-7(8H)-ones as corticotropin-releasing factor-1 receptor antagonists

by Dzierba, Carolyn D., Sielecki, Thais M., Arvanitis, Argyrios G., Galka, Amy, Johnson, Tricia L., Takvorian, Amy G., Rafalski, Maria, Kasireddy-Polam, Padmaja, Vig, Shikha, Dasgupta, Bireshwar, Zhang, Ge, Molski, Thaddeus F., Wong, Harvey, Zaczek, Robert C., Lodge, Nicholas J., Combs, Andrew P., Gilligan, Paul J., Trainor, George L., Bronson, Joanne J., Macor, John E.
Published in Bioorganic & medicinal chemistry letters (01.08.2012)

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Journal Article

HETEROARYL SUBSTITUTED PYRROLO[2,3-b]PYRIDINE AND PYRROLO[2,3-b]PYRIMIDINE AS JANUS KINASE INHIBITORS

HETEROARYL SUBSTITUTED PYRROLO[2,3-b]PYRIDINE AND PYRROLO[2,3-b]PYRIMIDINE AS JANUS KINASE INHIBITORS

by JALLURI RAVI KUMAR, RAFALSKI MARIA, FALAHATPISHEH NIKOO, STORACE LOUIS, MADUSKUIE THOMAS P, SHEPARD STACEY, FRIDMAN JORDAN S, VADDI KRISHNA, WANG HAISHENG, RODGERS JAMES D, ARVANITIS ARGYRIOS G
Year of Publication 05.11.2015

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Patent

N-Arylation of Primary and Secondary Aliphatic Amines on Solid Supports

N-Arylation of Primary and Secondary Aliphatic Amines on Solid Supports

by Combs, Andrew P, Tadesse, Seifu, Rafalski, Maria, Haque, Tasir S, Lam, Patrick Y. S
Published in Journal of combinatorial chemistry (01.03.2002)

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Journal Article

FURO- AND THIENO-PYRIDINE CARBOXAMIDE COMPOUNDS USEFUL AS PIM KINASE INHIBITORS

FURO- AND THIENO-PYRIDINE CARBOXAMIDE COMPOUNDS USEFUL AS PIM KINASE INHIBITORS

by RAFALSKI MARIA, YE HAI FEN, BURNS DAVID M, MEI SONG, VECHORKIN OLEG, LI YUN LONG, FENG HAO, HUANG TAISHENG, ZHU WENYU, WANG ANLAI, XUE CHU BIAO, PAN JUN
Year of Publication 20.05.2016

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Patent

Corrections to In Vitro Intrinsic Clearance-Based Optimization of N 3-Phenylpyrazinones as Corticotropin-Releasing Factor-1 (CRF1) Receptor Antagonists

Corrections to In Vitro Intrinsic Clearance-Based Optimization of N 3-Phenylpyrazinones as Corticotropin-Releasing Factor-1 (CRF1) Receptor Antagonists

by Hartz, Richard A., Ahuja, Vijay T., Rafalski, Maria, Schmitz, William D., Brenner, Allison B., Denhart, Derek J., Ditta, Jonathan L., Deskus, Jeffrey A., Yue, Eddy W., Arvanitis, Argyrios G., Lelas, Snjezana, Li, Yu-Wen, Molski, Thaddeus F., Wong, Harvey, Grace, James E., Lentz, Kimberley A., Li, Jianqing, Lodge, Nicholas J., Zaczek, Robert, Combs, Andrew P., Olson, Richard E., Mattson, Ronald J., Bronson, Joanne J., Macor, John E.
Published in Journal of medicinal chemistry (24.09.2009)

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Journal Article

In Vitro Intrinsic Clearance-Based Optimization of N3-Phenylpyrazinones as Corticotropin-Releasing Factor-1 (CRF1) Receptor Antagonists

In Vitro Intrinsic Clearance-Based Optimization of N3-Phenylpyrazinones as Corticotropin-Releasing Factor-1 (CRF1) Receptor Antagonists

by HARTZ, Richard A, AHUJA, Vijay T, LELAS, Snjezana, LI, Yu-Wen, MOLSKI, Thaddeus F, WONG, Harvey, GRACE, James E, LENTZ, Kimberley A, JIANQING LI, LODGE, Nicholas J, ZACZEK, Robert, COMBS, Andrew P, RAFALSKI, Maria, OLSON, Richard E, MATTSON, Ronald J, BRONSON, Joanne J, MACOR, John E, SCHMITZ, William D, BRENTER, Allison B, DENHART, Derek J, DITTA, Jonathan L, DESKUS, Jeffrey A, YUE, Eddy W, ARVANITIS, Argyrios G
Published in Journal of medicinal chemistry (23.07.2009)

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Journal Article

Synthesis, Structure—Activity Relationships, and In Vivo Evaluation of N3-Phenylpyrazinones as Novel Corticotropin-Releasing Factor-1 (CRF1) Receptor Antagonists

Synthesis, Structure—Activity Relationships, and In Vivo Evaluation of N3-Phenylpyrazinones as Novel Corticotropin-Releasing Factor-1 (CRF1) Receptor Antagonists

by HARTZ, Richard A, AHUJA, Vijay T, HOBBS, Frank W, PAYNE, Joseph, LELAS, Snjezana, LI, Yu-Wen, MOLSKI, Thaddeus F, MATTSON, Gail K, YONG PENG, WONG, Harvey, GRACE, James E, LENTZ, Kimberley A, ARVANITIS, Argyrios G, QIAN-CUTRONE, Jingfang, XIAOLIANG ZHUO, SHU, Yue-Zhong, LODGER, Nicholas J, ZACZEK, Robert, COMBS, Andrew P, OLSON, Richard E, BRONSON, Joanne J, MATTSON, Ronald J, MACOR, John E, RAFALSKI, Maria, YUE, Eddy W, DENHART, Derek J, SCHMITZ, William D, DITTA, Jonathan L, DESKUS, Jeffrey A, BRENNER, Allison B
Published in Journal of medicinal chemistry (23.07.2009)

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Journal Article

Dihydropyridopyrazinones and Dihydropteridinones as Corticotropin-Releasing Factor-1 Receptor Antagonists: Structure−Activity Relationships and Computational Modeling

Dihydropyridopyrazinones and Dihydropteridinones as Corticotropin-Releasing Factor-1 Receptor Antagonists: Structure−Activity Relationships and Computational Modeling

by Dzierba, Carolyn D, Tebben, Andrew J, Wilde, Richard G, Takvorian, Amy G, Rafalski, Maria, Kasireddy-Polam, Padmaja, Klaczkiewicz, John D, Pechulis, Anthony D, Davis, Amy L, Sweet, Mark P, Woo, Alex M, Yang, Zhicai, Ebeltoft, Sarah M, Molski, Thaddeus F, Zhang, Ge, Zaczek, Robert C, Trainor, George L, Combs, Andrew P, Gilligan, Paul J
Published in Journal of medicinal chemistry (03.05.2007)

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Journal Article

HETEROARYL SUBSTITUTED PYRROLO[2,3-B]PYRIDINES AND PYRROLO[2,3-B]PYRIMIDINES AS JANUS KINASE INHIBITORS

HETEROARYL SUBSTITUTED PYRROLO[2,3-B]PYRIDINES AND PYRROLO[2,3-B]PYRIMIDINES AS JANUS KINASE INHIBITORS

by ALVANITIS ARGYRIOS G, JALLURI RAVI KUMAR, RAFALSKI MARIA, FALAHATPISHEH NIKOO, STORACE LOUIS, MADUSKUIE THOMAS P, SHEPARD STACEY, FRIDMAN JORDAN S, VADDI KRISHNA, WANG HAISHENG, RODGERS JAMES D
Year of Publication 22.12.2011

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Patent

Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors

Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors

by Arvanitis, Argyrios G, Rafalski, Maria, Maduskuie, Thomas P, Storace, Louis, Wang, Haisheng, Vaddi, Krishna, Jalluri, Ravi Kumar, Shepard, Stacey, Fridman, Jordan S, Rogers, James D, Falahatpisheh, Nikoo
Year of Publication 01.08.2024

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Patent

HETEROARYL SUBSTITUTED PYRROLO[2,3-B]PYRIDINES AND PYRROLO[2,3-B]PYRIMIDINES AS JANUS KINASE INHIBITORS

HETEROARYL SUBSTITUTED PYRROLO[2,3-B]PYRIDINES AND PYRROLO[2,3-B]PYRIMIDINES AS JANUS KINASE INHIBITORS

by Arvanitis, Argyrios G, Rafalski, Maria, Maduskuie, Thomas P, Storace, Louis, Wang, Haisheng, Vaddi, Krishna, Jalluri, Ravi Kumar, Shepard, Stacey, Fridman, Jordan S, Rogers, James D, Falahatpisheh, Nikoo
Year of Publication 11.07.2024

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Patent

Synthesis, Structure−Activity Relationships, and in Vivo Properties of 3,4-Dihydro-1H-pyrido[2,3-b]pyrazin-2-ones as Corticotropin-Releasing Factor-1 Receptor Antagonists

Synthesis, Structure−Activity Relationships, and in Vivo Properties of 3,4-Dihydro-1H-pyrido[2,3-b]pyrazin-2-ones as Corticotropin-Releasing Factor-1 Receptor Antagonists

by Dzierba, Carolyn D, Takvorian, Amy G, Rafalski, Maria, Kasireddy-Polam, Padmaja, Wong, Harvey, Molski, Thaddeus F, Zhang, Ge, Li, Yu-Wen, Lelas, Snjezana, Peng, Yong, McElroy, John F, Zaczek, Robert C, Taub, Rebecca A, Combs, Andrew P, Gilligan, Paul J, Trainor, George L
Published in Journal of medicinal chemistry (04.11.2004)

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PYRROLO[2,3-D]PYRIMIDINE DERIVATIVE AS JANUS KINASE INHIBITOR

PYRROLO[2,3-D]PYRIMIDINE DERIVATIVE AS JANUS KINASE INHIBITOR

by JALLURI, Ravi Kuma, VADDI, Krishna, MADUSKUIE, Thomas P, WANG, Haisheng, FALAHATPISHEH, Nikoo, STORACE, Louis, FRIDMAN, Jordon S, RODGERS, James D, SHEPARD, Stacey, RAFALSKI, Maria, ARVANITIS, Argyrios G
Year of Publication 22.11.2023

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Patent

Synthesis, Structure−Activity Relationships, and in Vivo Properties of 3,4-Dihydro-1 H -pyrido[2,3- b ]pyrazin-2-ones as Corticotropin-Releasing Factor-1 Receptor Antagonists

Synthesis, Structure−Activity Relationships, and in Vivo Properties of 3,4-Dihydro-1 H -pyrido[2,3- b ]pyrazin-2-ones as Corticotropin-Releasing Factor-1 Receptor Antagonists

by Dzierba, Carolyn D., Takvorian, Amy G., Rafalski, Maria, Kasireddy-Polam, Padmaja, Wong, Harvey, Molski, Thaddeus F., Zhang, Ge, Li, Yu-Wen, Lelas, Snjezana, Peng, Yong, McElroy, John F., Zaczek, Robert C., Taub, Rebecca A., Combs, Andrew P., Gilligan, Paul J., Trainor, George L.
Published in Journal of medicinal chemistry (01.11.2004)

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