An alignment-independent three-dimensional quantitative structure-activity relationship study on ron receptor tyrosine kinase inhibitors
Zarei, Omid, Raeppel, Stéphane L, Hamzeh-Mivehroud, Maryam
Published in Journal of bioinformatics and computational biology (01.06.2022)
Published in Journal of bioinformatics and computational biology (01.06.2022)
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Journal Article
When RON MET TAM in Mesothelioma: All Druggable for One, and One Drug for All?
Baird, Anne-Marie, Easty, David, Jarzabek, Monika, Shiels, Liam, Soltermann, Alex, Klebe, Sonja, Raeppel, Stéphane, MacDonagh, Lauren, Wu, Chengguang, Griggs, Kim, Kirschner, Michaela B, Stanfill, Bryan, Nonaka, Daisuke, Goparaju, Chandra M, Murer, Bruno, Fennell, Dean A, O'Donnell, Dearbhaile M, Barr, Martin P, Mutti, Luciano, Reid, Glen, Finn, Stephen, Cuffe, Sinead, Pass, Harvey I, Opitz, Isabelle, Byrne, Annette T, O'Byrne, Kenneth J, Gray, Steven G
Published in Frontiers in endocrinology (Lausanne) (26.02.2019)
Published in Frontiers in endocrinology (Lausanne) (26.02.2019)
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N-(4-(6,7-Disubstituted-quinolin-4-yloxy)-3-fluorophenyl)-2-oxo-3-phenylimidazolidine-1-carboxamides: A novel series of dual c-Met/VEGFR2 receptor tyrosine kinase inhibitors
Mannion, Michael, Raeppel, Stéphane, Claridge, Stephen, Zhou, Nancy, Saavedra, Oscar, Isakovic, Ljubomir, Zhan, Lijie, Gaudette, Frédéric, Raeppel, Franck, Déziel, Robert, Beaulieu, Normand, Nguyen, Hannah, Chute, Ian, Beaulieu, Carole, Dupont, Isabelle, Robert, Marie-France, Lefebvre, Sylvain, Dubay, Marja, Rahil, Jubrail, Wang, James, Ste-Croix, Hélène, Robert Macleod, A., Besterman, Jeffrey M., Vaisburg, Arkadii
Published in Bioorganic & medicinal chemistry letters (01.12.2009)
Published in Bioorganic & medicinal chemistry letters (01.12.2009)
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N-(3-fluoro-4-(2-arylthieno[3,2- b]pyridin-7-yloxy)phenyl)-2-oxo-3-phenylimidazolidine-1-carboxamides: A novel series of dual c-Met/VEGFR2 receptor tyrosine kinase inhibitors
Raeppel, Stéphane, Claridge, Stephen, Saavedra, Oscar, Gaudette, Frédéric, Zhan, Lijie, Mannion, Michael, Zhou, Nancy, Raeppel, Franck, Granger, Marie-Claude, Isakovic, Ljubomir, Déziel, Robert, Nguyen, Hannah, Beaulieu, Normand, Beaulieu, Carole, Dupont, Isabelle, Robert, Marie-France, Lefebvre, Sylvain, Dubay, Marja, Rahil, Jubrail, Wang, James, Ste-Croix, Hélène, Robert Macleod, A., Besterman, Jeffrey, Vaisburg, Arkadii
Published in Bioorganic & medicinal chemistry letters (01.03.2009)
Published in Bioorganic & medicinal chemistry letters (01.03.2009)
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Journal Article
Identification of potent and selective VEGFR receptor tyrosine kinase inhibitors having new amide isostere headgroups
Gaudette, Frédéric, Raeppel, Stéphane, Nguyen, Hannah, Beaulieu, Normand, Beaulieu, Carole, Dupont, Isabelle, Macleod, A. Robert, Besterman, Jeffrey M., Vaisburg, Arkadii
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
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Journal Article
Identification of a novel series of potent RON receptor tyrosine kinase inhibitors
Raeppel, Stéphane, Gaudette, Frédéric, Mannion, Michael, Claridge, Stephen, Saavedra, Oscar, Isakovic, Ljubomir, Déziel, Robert, Beaulieu, Normand, Beaulieu, Carole, Dupont, Isabelle, Nguyen, Hannah, Wang, James, Macleod, A. Robert, Maroun, Christiane, Besterman, Jeffrey M., Vaisburg, Arkadii
Published in Bioorganic & medicinal chemistry letters (01.05.2010)
Published in Bioorganic & medicinal chemistry letters (01.05.2010)
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Journal Article
Design and synthesis of 4-[( s-triazin-2-ylamino)methyl]- N-(2-aminophenyl)-benzamides and their analogues as a novel class of histone deacetylase inhibitors
Paquin, Isabelle, Raeppel, Stéphane, Leit, Silvana, Gaudette, Frédéric, Zhou, Nancy, Moradei, Oscar, Saavedra, Oscar, Bernstein, Naomy, Raeppel, Franck, Bouchain, Giliane, Fréchette, Sylvie, Woo, Soon H., Vaisburg, Arkadii, Fournel, Marielle, Kalita, Ann, Robert, Marie-France, Lu, Aihua, Trachy-Bourget, Marie-Claude, Yan, Pu Theresa, Liu, Jianhong, Rahil, Jubrail, MacLeod, A. Robert, Besterman, Jeffrey M., Li, Zuomei, Delorme, Daniel
Published in Bioorganic & medicinal chemistry (01.02.2008)
Published in Bioorganic & medicinal chemistry (01.02.2008)
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Journal Article
Identification of a Novel Series of Potent TrkA Receptor Tyrosine Kinase Inhibitors
Raeppel, Stéphane L., Gaudette, Frédéric, Nguyen, Hannah, Beaulieu, Normand, Wang, James, Maroun, Christiane, Besterman, Jeffrey M., Vaisburg, Arkadii
Published in International Journal of Medicinal Chemistry (Online) (01.01.2012)
Published in International Journal of Medicinal Chemistry (Online) (01.01.2012)
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Journal Article
SAR and biological evaluation of analogues of a small molecule histone deacetylase inhibitor N-(2-aminophenyl)-4-((4-(pyridin-3-yl)pyrimidin-2-ylamino)methyl)benzamide ( MGCD0103)
Raeppel, Stéphane, Zhou, Nancy, Gaudette, Frédéric, Leit, Silvana, Paquin, Isabelle, Larouche, Guillaume, Moradei, Oscar, Fréchette, Sylvie, Isakovic, Ljubomir, Delorme, Daniel, Fournel, Marielle, Kalita, Ann, Lu, Aihua, Trachy-Bourget, Marie-Claude, Yan, Pu Theresa, Liu, Jianhong, Rahil, Jubrail, Wang, James, Besterman, Jeffrey M., Murakami, Koji, Li, Zuomei, Vaisburg, Arkadii
Published in Bioorganic & medicinal chemistry letters (01.02.2009)
Published in Bioorganic & medicinal chemistry letters (01.02.2009)
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Journal Article
Substituted N-(2-aminophenyl)-benzamides, ( E)- N-(2-aminophenyl)-acrylamides and their analogues: Novel classes of histone deacetylase inhibitors
Moradei, Oscar, Leit, Silvana, Zhou, Nancy, Fréchette, Sylvie, Paquin, Isabelle, Raeppel, Stéphane, Gaudette, Frédéric, Bouchain, Giliane, Woo, Soon H., Vaisburg, Arkadii, Fournel, Marielle, Kalita, Ann, Lu, Aihua, Trachy-Bourget, Marie-Claude, Yan, Pu T., Liu, Jianhong, Li, Zuomei, Rahil, Jubrail, MacLeod, A. Robert, Besterman, Jeffrey M., Delorme, Daniel
Published in Bioorganic & medicinal chemistry letters (01.08.2006)
Published in Bioorganic & medicinal chemistry letters (01.08.2006)
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Journal Article
4-(Heteroarylaminomethyl)- N-(2-aminophenyl)-benzamides and their analogs as a novel class of histone deacetylase inhibitors
Fréchette, Sylvie, Leit, Silvana, Woo, Soon Hyung, Lapointe, Guillaume, Jeannotte, Guillaume, Moradei, Oscar, Paquin, Isabelle, Bouchain, Giliane, Raeppel, Stéphane, Gaudette, Frédéric, Zhou, Nancy, Vaisburg, Arkadii, Fournel, Marielle, Yan, Pu Theresa, Trachy-Bourget, Marie-Claude, Kalita, Ann, Robert, Marie-France, Lu, Aihua, Rahil, Jubrail, Robert MacLeod, A., Besterman, Jeffrey M., Li, Zuomei, Delorme, Daniel
Published in Bioorganic & medicinal chemistry (15.02.2008)
Published in Bioorganic & medicinal chemistry (15.02.2008)
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Journal Article
P3.03-021 When RON MET TAM in Mesothelioma: All Druggable for One, and One Drug for All?: Topic: Mesothelioma Transitional
Baird, Anne-Marie, Easty, David, Jarzabek, Monika, Shiels, Liam, Soltermann, Alex, Raeppel, Stéphane, Mcdonagh, Lauren, Wu, Chengguang, Goparju, Chandra, Stanfill, Bryan, Barr, Martin, Nonaka, Daisuke, Murer, Bruno, Fennell, Dean, O’Donnell, Dearbhaile, Mutti, Luciano, Finn, Stephen, Cuffe, Sinead, Pass, Harvey, Schmitt-Opitz, Isabelle, Byrne, Annette, O’Byrne, Kenneth, Gray, Steven
Published in Journal of thoracic oncology (01.01.2017)
Published in Journal of thoracic oncology (01.01.2017)
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Journal Article
P3.03-021 When RON MET TAM in Mesothelioma: All Druggable for One, and One Drug for All?
Baird, Anne-Marie, Easty, David, Jarzabek, Monika, Shiels, Liam, Soltermann, Alex, Raeppel, Stéphane, Mcdonagh, Lauren, Wu, Chengguang, Goparju, Chandra, Stanfill, Bryan, Barr, Martin, Nonaka, Daisuke, Murer, Bruno, Fennell, Dean, O’Donnell, Dearbhaile, Mutti, Luciano, Finn, Stephen, Cuffe, Sinead, Pass, Harvey, Schmitt-Opitz, Isabelle, Byrne, Annette, O’Byrne, Kenneth, Gray, Steven
Published in Journal of thoracic oncology (01.01.2017)
Published in Journal of thoracic oncology (01.01.2017)
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Journal Article
Lewis acid-catalyzed Mannich type reactions with potassium organotrifluoroborates
Tremblay-Morin, Jean-Philipe, Raeppel, Stéphane, Gaudette, Frédéric
Published in Tetrahedron letters (19.04.2004)
Published in Tetrahedron letters (19.04.2004)
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Journal Article
A potential signaling axis between RON kinase receptor and hypoxia‐inducible factor‐1 alpha in pancreatic cancer
Kato, Akihisa, Ng, Serina, Thangasamy, Amalraj, Han, Haiyong, Zhou, Wendi, Raeppel, Stephane, Fallon, Michael, Guha, Sushovan, Ammanamanchi, Sudhakar
Published in Molecular carcinogenesis (01.11.2021)
Published in Molecular carcinogenesis (01.11.2021)
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Journal Article
Cover Image, Volume 60, Issue 11
Kato, Akihisa, Ng, Serina, Thangasamy, Amalraj, Han, Haiyong, Zhou, Wendi, Raeppel, Stephane, Fallon, Michael, Guha, Sushovan, Ammanamanchi, Sudhakar
Published in Molecular carcinogenesis (01.11.2021)
Published in Molecular carcinogenesis (01.11.2021)
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