Aminoguanidine Hydrazone Derivatives as Nonpeptide NPFF1 Receptor Antagonists Reverse Opioid Induced Hyperalgesia
Hammoud, Hassan, Elhabazi, Khadija, Quillet, Raphäelle, Bertin, Isabelle, Utard, Valérie, Laboureyras, Emilie, Bourguignon, Jean-Jacques, Bihel, Frédéric, Simonnet, Guy, Simonin, Frédéric, Schmitt, Martine
Published in ACS chemical neuroscience (21.11.2018)
Published in ACS chemical neuroscience (21.11.2018)
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Journal Article
Characterisation of NPFF-expressing neurons in the superficial dorsal horn of the mouse spinal cord
Quillet, Raphaëlle, Dickie, Allen C, Polgár, Erika, Gutierrez-Mecinas, Maria, Bell, Andrew M, Goffin, Luca, Watanabe, Masahiko, Todd, Andrew J
Published in Scientific reports (11.04.2023)
Published in Scientific reports (11.04.2023)
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Journal Article
Grpr expression defines a population of superficial dorsal horn vertical cells that have a role in both itch and pain
Polgár, Erika, Dickie, Allen C, Gutierrez-Mecinas, Maria, Bell, Andrew M, Boyle, Kieran A, Quillet, Raphaëlle, Ab Rashid, Elisha, Clark, Ross A, German, Morgan T, Watanabe, Masahiko, Riddell, John S, Todd, Andrew J
Published in Pain (Amsterdam) (01.01.2023)
Published in Pain (Amsterdam) (01.01.2023)
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Antibodies Against the Gastrin-releasing Peptide Precursor Pro-Gastrin-releasing Peptide Reveal Its Expression in the Mouse Spinal Dorsal Horn
Gutierrez-Mecinas, Maria, Kókai, Éva, Polgár, Erika, Quillet, Raphaëlle, Titterton, Heather F., Weir, Greg A., Watanabe, Masahiko, Todd, Andrew J.
Published in Neuroscience (01.02.2023)
Published in Neuroscience (01.02.2023)
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Journal Article
Characterisation of lamina I anterolateral system neurons that express Cre in a Phox2a-Cre mouse line
Alsulaiman, Wafa A. A., Quillet, Raphaelle, Bell, Andrew M., Dickie, Allen C., Polgár, Erika, Boyle, Kieran A., Watanabe, Masahiko, Roome, R. Brian, Kania, Artur, Todd, Andrew J., Gutierrez-Mecinas, Maria
Published in Scientific reports (09.09.2021)
Published in Scientific reports (09.09.2021)
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Journal Article
RF-amide neuropeptides and their receptors in Mammals: Pharmacological properties, drug development and main physiological functions
Quillet, Raphaëlle, Ayachi, Safia, Bihel, Frédéric, Elhabazi, Khadija, Ilien, Brigitte, Simonin, Frédéric
Published in Alimentary Pharmacology & Therapeutics (Suppl) (01.04.2016)
Published in Alimentary Pharmacology & Therapeutics (Suppl) (01.04.2016)
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Journal Article
Synaptic circuits involving gastrin-releasing peptide receptor-expressing neurons in the dorsal horn of the mouse spinal cord
Quillet, Raphaëlle, Gutierrez-Mecinas, Maria, Polgár, Erika, Dickie, Allen C, Boyle, Kieran A, Watanabe, Masahiko, Todd, Andrew J
Published in Frontiers in molecular neuroscience (07.12.2023)
Published in Frontiers in molecular neuroscience (07.12.2023)
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Journal Article
Neuropeptide FF increases M2 activation and self-renewal of adipose tissue macrophages
Waqas, Syed F Hassnain, Hoang, Anh Cuong, Lin, Ya-Tin, Ampem, Grace, Azegrouz, Hind, Balogh, Lajos, Thuróczy, Julianna, Chen, Jin-Chung, Gerling, Ivan C, Nam, Sorim, Lim, Jong-Seok, Martinez-Ibañez, Juncal, Real, José T, Paschke, Stephan, Quillet, Raphaëlle, Ayachi, Safia, Simonin, Frédéric, Schneider, E Marion, Brinkman, Jacqueline A, Lamming, Dudley W, Seroogy, Christine M, Röszer, Tamás
Published in The Journal of clinical investigation (01.09.2017)
Published in The Journal of clinical investigation (01.09.2017)
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Journal Article
Identification of an N‑acylated‑DArg-Leu-NH2 Dipeptide as a Highly Selective Neuropeptide FF1 Receptor Antagonist That Potently Prevents Opioid-Induced Hyperalgesia
Quillet, Raphaëlle, Schneider, Séverine, Utard, Valérie, Drieu la Rochelle, Armand, Elhabazi, Khadija, Henningsen, Jo Beldring, Gizzi, Patrick, Schmitt, Martine, Kugler, Valérie, Simonneaux, Valérie, Ilien, Brigitte, Simonin, Frédéric, Bihel, Frédéric
Published in Journal of medicinal chemistry (10.06.2021)
Published in Journal of medicinal chemistry (10.06.2021)
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Journal Article
A bifunctional-biased mu-opioid agonist-neuropeptide FF receptor antagonist as analgesic with improved acute and chronic side effects
Drieu la Rochelle, Armand, Guillemyn, Karel, Dumitrascuta, Maria, Martin, Charlotte, Utard, Valérie, Quillet, Raphaëlle, Schneider, Séverine, Daubeuf, François, Willemse, Tom, Mampuys, Pieter, Maes, Bert U W, Frossard, Nelly, Bihel, Frédéric, Spetea, Mariana, Simonin, Frédéric, Ballet, Steven
Published in Pain (Amsterdam) (01.09.2018)
Published in Pain (Amsterdam) (01.09.2018)
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Journal Article
RF313, an orally bioavailable neuropeptide FF receptor antagonist, opposes effects of RF-amide-related peptide-3 and opioid-induced hyperalgesia in rodents
Elhabazi, Khadija, Humbert, Jean-Paul, Bertin, Isabelle, Quillet, Raphaelle, Utard, Valérie, Schneider, Séverine, Schmitt, Martine, Bourguignon, Jean-Jacques, Laboureyras, Emilie, Ben Boujema, Meric, Simonnet, Guy, Ancel, Caroline, Simonneaux, Valérie, Beltramo, Massimiliano, Bucher, Bernard, Sorg, Tania, Meziane, Hamid, Schneider, Elodie, Petit-Demoulière, Benoit, Ilien, Brigitte, Bihel, Frédéric, Simonin, Frédéric
Published in Neuropharmacology (15.05.2017)
Published in Neuropharmacology (15.05.2017)
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Journal Article
Neuropeptide FF increases M2 activation and self-renewal of adipose tissue macrophages
Waqas, Syed F Hassnain, Hoang, Anh Cuong, Lin, Ya-Tin, Ampem, Grace, Azegrouz, Hind, Balogh, Lajos, Thuróczy, Julianna, Chen, Jin-Chung, Gerling, Ivan C, Nam, Sorim, Lim, Jong-Seok, Martinez-Ibañez, Juncal, Real, José T, Paschke, Stephan, Quillet, Raphaëlle, Ayachi, Safia, Simonin, Frédéric, Schneider, E Marion, Brinkman, Jacqueline A, Lamming, Dudley W, Seroogy, Christine M, Röszer, Tamás
Published in The Journal of clinical investigation (01.09.2017)
Published in The Journal of clinical investigation (01.09.2017)
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Journal Article
Characterization of anti-GASP motif antibodies that inhibit the interaction between GPRASP1 and G protein-coupled receptors
Zeder-Lutz, Gabrielle, Bornert, Olivier, Fellmann-Clauss, Rosine, Knittel-Obrecht, Adeline, Tranchant, Thibaud, Bouteben, Sarah, Kaeffer, Juliette, Quillet, Raphaëlle, Villa, Pascal, Wagner, Renaud, Lecat, Sandra, Simonin, Frédéric
Published in Analytical biochemistry (15.03.2023)
Published in Analytical biochemistry (15.03.2023)
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Journal Article
Identification of an N-acylated-(D)Arg-Leu-NH2 Dipeptide as a Highly Selective Neuropeptide FF1 Receptor Antagonist That Potently Prevents Opioid-Induced Hyperalgesia
Quillet, Raphaelle, Schneider, Severine, Utard, Valerie, la Rochelle, Armand Drieu, Elhabazi, Khadija, Henningsen, Jo Beldring, Gizzi, Patrick, Schmitt, Martine, Kugler, Valerie, Simonneaux, Valerie, Ilien, Brigitte, Simonin, Frederic, Bihel, Frederic
Published in Journal of medicinal chemistry (10.06.2021)
Published in Journal of medicinal chemistry (10.06.2021)
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Journal Article
Deep sequencing of Phox2a nuclei reveals five classes of anterolateral system neurons
Bell, Andrew M, Utting, Charlotte, Dickie, Allen C, Kucharczyk, Mateusz W, Quillet, Raphaëlle, Gutierrez-Mecinas, Maria, Razlan, Aimi N B, Cooper, Andrew H, Lan, Yuxuan, Hachisuka, Junichi, Weir, Greg A, Bannister, Kirsty, Watanabe, Masahiko, Kania, Artur, Hoon, Mark A, Macaulay, Iain C, Denk, Franziska, Todd, Andrew J
Published in Proceedings of the National Academy of Sciences - PNAS (04.06.2024)
Published in Proceedings of the National Academy of Sciences - PNAS (04.06.2024)
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Journal Article
Identification of an N -acylated- D Arg-Leu-NH 2 Dipeptide as a Highly Selective Neuropeptide FF1 Receptor Antagonist That Potently Prevents Opioid-Induced Hyperalgesia
Quillet, Raphaëlle, Schneider, Séverine, Utard, Valérie, Drieu la Rochelle, Armand, Elhabazi, Khadija, Henningsen, Jo Beldring, Gizzi, Patrick, Schmitt, Martine, Kugler, Valérie, Simonneaux, Valérie, Ilien, Brigitte, Simonin, Frédéric, Bihel, Frédéric
Published in Journal of medicinal chemistry (10.06.2021)
Published in Journal of medicinal chemistry (10.06.2021)
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Journal Article
Neuropeptide FF increases M2 activation and self-renewal of adipose tissue macrophages
Waqas, Syed F. Hassnain, Hoang, Anh Cuong, Lin, Ya-Tin, Ampem, Grace, Azegrouz, Hind, Balogh, Lajos, Thuroczy, Julianna, Chen, Jin-Chung, Gerling, Ivan C, Nam, Sorim, Lim, Jong-Seok, Martinez-Ibanez, Juncal, Real, Jose T, Paschke, Stephan, Quillet, Raphaelle, Ayachi, Safia, Simonin, Frederic, Schneider, E. Marion, Brinkman, Jacqueline A, Lamming, Dudley W, Seroogy, Christine M, Roszer, Tamas
Published in The Journal of clinical investigation (01.07.2017)
Published in The Journal of clinical investigation (01.07.2017)
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