BACE-1 inhibitory activities of new substituted phenyl-piperazine coupled to various heterocycles: Chromene, coumarin and quinoline
Garino, Cédrik, Pietrancosta, Nicolas, Laras, Younes, Moret, Vincent, Rolland, Amandine, Quéléver, Gilles, Kraus, Jean-Louis
Published in Bioorganic & medicinal chemistry letters (01.04.2006)
Published in Bioorganic & medicinal chemistry letters (01.04.2006)
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Journal Article
New Antiviral Nucleoside Prodrugs Await Application
Anastasi, Carole, Quéléver, Gilles, Burlet, Stéphane, Garino, Cédrik, Souard, Florence, Kraus, Jean-Louis
Published in Current medicinal chemistry (01.09.2003)
Published in Current medicinal chemistry (01.09.2003)
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Journal Article
New 2-bromomethyl-8-substituted-benzo[ c]chromen-6-ones. Synthesis and biological properties
Garino, Cédrik, Bihel, Frédéric, Pietrancosta, Nicolas, Laras, Younes, Quéléver, Gilles, Woo, Irene, Klein, Peter, Bain, Jenny, Boucher, Jean-Luc, Kraus, Jean-Louis
Published in Bioorganic & medicinal chemistry letters (03.01.2005)
Published in Bioorganic & medicinal chemistry letters (03.01.2005)
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Journal Article
Novel cyclized Pifithrin-α p53 inactivators: synthesis and biological studies
Pietrancosta, Nicolas, Maina, Flavio, Dono, Rosanna, Moumen, Anice, Garino, Cédrik, Laras, Younes, Burlet, Stéphane, Quéléver, Gilles, Kraus, Jean-Louis
Published in Bioorganic & medicinal chemistry letters (15.03.2005)
Published in Bioorganic & medicinal chemistry letters (15.03.2005)
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Journal Article
Prospects for the Resistance to HIV Protease Inhibitors: Current Drug Design Approaches and Perspectives
Burlet, S., Pietrancosta, N., Laras, Y., Garino, C., Quelever, G., Kraus, J.-
Published in Current pharmaceutical design (01.09.2005)
Published in Current pharmaceutical design (01.09.2005)
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Journal Article
Synthesis of new 3-alkoxy-7-amino-4-chloro-isocoumarin derivatives as new β-amyloid peptide production inhibitors and their activities on various classes of protease
Bihel, Frédéric, Quéléver, Gilles, Lelouard, Hugues, Petit, Agnès, Alvès da Costa, Cristine, Pourquié, Olivier, Checler, Frédéric, Thellend, Annie, Pierre, Philippe, Kraus, Jean-Louis
Published in Bioorganic & medicinal chemistry (17.07.2003)
Published in Bioorganic & medicinal chemistry (17.07.2003)
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Journal Article
Substituted thiazolamide coupled to a redox delivery system: a new gamma-secretase inhibitor with enhanced pharmacokinetic profile
Laras, Y, Quelever, G, Garino, C, Pietrancosta, N, Sheha, M, Bihel, F, Wolfe, MS, Kraus, JL
Published in Organic & biomolecular chemistry (21.02.2005)
Published in Organic & biomolecular chemistry (21.02.2005)
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Journal Article
Synthesis of new 7-membered α-phenylthio cyclic oxamides: HIV inhibitors
Medou, M., Priem, G., Quélever, G., Camplo, M., Kraus, J.L.
Published in Tetrahedron letters (04.06.1998)
Published in Tetrahedron letters (04.06.1998)
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Journal Article
Design of potential new HIV protease inhibitors: enantioconvergent synthesis of new pyrrolidin-3-ol, and pyrrolidin-3-one peptide conjugates
Courcambeck, J, Bihel, F, De Michelis, C, Quelever, G, Kraus, JL
Published in Perkin 1 : an international journal of organic and bio-organic chemistry (01.01.2001)
Published in Perkin 1 : an international journal of organic and bio-organic chemistry (01.01.2001)
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Journal Article
Conformational sensibility of PEO-PAMAM hybrid molecules to cations adducted upon electrospray ionization - A mass spectrometry, ion mobility and molecular modeling study
Tintaru, A., Chendo, C., Wang, Qiang, Viel, S., Quelever, G., Peng, Ling, Posocco, P., Pricl, S., Charles, L.
Published in Analytica chimica acta (2014)
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Published in Analytica chimica acta (2014)
Journal Article
CS Coupling Using a Mixed-Ligand Pd Catalyst: A Highly Effective Strategy for Synthesizing Arylthio-Substituted Heterocycles
Cong, Mei, Fan, Yuting, Raimundo, Jean-Manuel, Xia, Yi, Liu, Yang, Quéléver, Gilles, Qu, Fanqi, Peng, Ling
Published in Chemistry : a European journal (16.12.2013)
Published in Chemistry : a European journal (16.12.2013)
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Journal Article
Synthesis of Poly(amino)ester Dendrimers via Active Cyanomethyl Ester Intermediates
Bouillon, Camille, Tintaru, Aura, Monnier, Valérie, Charles, Laurence, Quéléver, Gilles, Peng, Ling
Published in Journal of organic chemistry (17.12.2010)
Published in Journal of organic chemistry (17.12.2010)
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Journal Article
Naphthyl and Coumarinyl Biarylpiperazine Derivatives as Highly Potent Human β-Secretase Inhibitors. Design, Synthesis, and Enzymatic BACE-1 and Cell Assays
Garino, Cédrik, Tomita, Taisuke, Pietrancosta, Nicolas, Laras, Younes, Rosas, Roselyne, Herbette, Gaëtan, Maigret, Bernard, Quéléver, Gilles, Iwatsubo, Takeshi, Kraus, Jean-Louis
Published in Journal of medicinal chemistry (13.07.2006)
Published in Journal of medicinal chemistry (13.07.2006)
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