Optimization of 3-(1H-Indazol-3-ylmethyl)-1,5-benzodiazepines as Potent, Orally Active CCK-A Agonists
Henke, Brad R, Aquino, Christopher J, Birkemo, Larry S, Croom, Dallas K, Dougherty, Robert W, Ervin, Gregory N, Grizzle, Mary K, Hirst, Gavin C, James, Michael K, Johnson, Michael F, Queen, Kennedy L, Sherrill, Ronald G, Sugg, Elizabeth E, Suh, Edward M, Szewczyk, Jerzy W, Unwalla, Rayomand J, Yingling, Jeff, Willson, Timothy M
Published in Journal of medicinal chemistry (15.08.1997)
Published in Journal of medicinal chemistry (15.08.1997)
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Discovery of 1,5-Benzodiazepines with Peripheral Cholecystokinin (CCK-A) Receptor Agonist Activity. 1. Optimization of the Agonist “Trigger”
Aquino, Christopher J, Armour, Duncan R, Berman, Judd M, Birkemo, Larry S, Carr, Robin A. E, Croom, Dallas K, Dezube, Milana, Dougherty, Robert W, Ervin, Gregory N, Grizzle, Mary K, Head, Julie E, Hirst, Gavin C, James, Michael K, Johnson, Michael F, Miller, Laurence J, Queen, Kennedy L, Rimele, Thomas J, Smith, David N, Sugg, Elizabeth E
Published in Journal of medicinal chemistry (19.01.1996)
Published in Journal of medicinal chemistry (19.01.1996)
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1,4-Benzodiazepine Peripheral Cholecystokinin (CCK-A) Receptor Agonists
Sherrill, Ronald G, Berman, Judd M, Birkemo, Lawrence, Croom, Dallas K, Dezube, Milana, Ervin, Gregory N, Grizzle, Mary K, James, Michael K, Johnson, Michael F, Queen, Kennedy L, Rimele, Thomas J, Vanmiddlesworth, Frank, Sugg, Elizabeth E
Published in Bioorganic & medicinal chemistry letters (07.05.2001)
Published in Bioorganic & medicinal chemistry letters (07.05.2001)
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3-(1H-Indazol-3-ylmethyl)-1,5-benzodiazepines: CCK-A Agonists That Demonstrate Oral Activity as Satiety Agents
Henke, Brad R, Willson, Timothy M, Sugg, Elizabeth E, Croom, Dallas K, Dougherty, Robert W, Queen, Kennedy L, Birkemo, Larry S, Ervin, Gregory N, Grizzle, Mary K, Johnson, Michael F, James, Michael K
Published in Journal of medicinal chemistry (05.07.1996)
Published in Journal of medicinal chemistry (05.07.1996)
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3-[2-(N-Phenylacetamide)]-1,5-benzodiazepines: Orally Active, Binding Selective CCK-A Agonists
Willson, Timothy M, Henke, Brad R, Momtahen, Tanya M, Myers, Peter L, Sugg, Elizabeth E, Unwalla, Rayomand J, Croom, Dallas K, Dougherty, Robert W, Grizzle, Mary K, Johnson, Michael F, Queen, Kennedy L, Rimele, Thomas J, Yingling, Jeffrey D, James, Michael K
Published in Journal of medicinal chemistry (19.07.1996)
Published in Journal of medicinal chemistry (19.07.1996)
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The Acute Extracellular Flux (XF) Assay to Assess Compound Effects on Mitochondrial Function
Wang, Ruolan, Novick, Steven J., Mangum, James B., Queen, Kennedy, Ferrick, David A., Rogers, George W., Stimmel, Julie B.
Published in Journal of biomolecular screening (01.03.2015)
Published in Journal of biomolecular screening (01.03.2015)
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CCK-A Receptor Selective Antagonists Derived from the CCK-A Receptor Selective Tetrapeptide Agonist Boc-Trp-Lys(Tac)-Asp-MePhe-NH2 (A-71623)
Sugg, Elizabeth E, Kimery, Millard J, Ding, Jian Mei, Kenakin, Deborah C, Miller, Laurence J, Queen, Kennedy L, Rimele, Thomas J
Published in Journal of medicinal chemistry (01.01.1995)
Published in Journal of medicinal chemistry (01.01.1995)
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Structure activity relationships of a series of buspirone analogs at alpha-1 adrenoceptors: further evidence that rat aorta alpha-1 adrenoceptors are of the alpha-1D-subtype
D L Saussy, Jr, A S Goetz, K L Queen, H K King, M W Lutz, T J Rimele
Published in The Journal of pharmacology and experimental therapeutics (01.07.1996)
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Published in The Journal of pharmacology and experimental therapeutics (01.07.1996)
Journal Article
Discovery of 1,5-Benzodiazepines with Peripheral Cholecystokinin (CCK-A) Receptor Agonist Activity (II): Optimization of the C3 Amino Substituent
Hirst, Gavin C., Aquino, Christopher, Birkemo, Lawrence, Croom, Dallas K., Dezube, Milana, Dougherty, Robert W., Ervin, Gregory N., Grizzle, Mary K., Henke, Brad, James, Michael K., Johnson, Michael F., Momtahen, Tanya, Queen, Kennedy L., Sherrill, Ronald G., Szewczyk, Jerzy, Willson, Timothy M., Sugg, Elizabeth E.
Published in Journal of medicinal chemistry (20.12.1996)
Published in Journal of medicinal chemistry (20.12.1996)
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Conversion of acyclic nonpeptide CCK antagonists into CCK agonists
Hirst, Gavin C., Queen, Kennedy L., Sugg, Elizabeth F., Willson, Timothy M.
Published in Bioorganic & medicinal chemistry letters (04.03.1997)
Published in Bioorganic & medicinal chemistry letters (04.03.1997)
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Journal Article
Modification of Receptor Selectivity and Functional Activity in Cholecystokinin Peptoid Ligands
Dezube, Milana, Sugg, Elizabeth E, Birkemo, Larry S, Croom, Dallas K, Dougherty, Robert W, Ervin, Gregory N, Grizzle, Mary K, James, Michael K, Johnson, Michael F
Published in Journal of medicinal chemistry (01.08.1995)
Published in Journal of medicinal chemistry (01.08.1995)
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A mathematical model for analysis of pharmacologically induced changes in the kinetics of cardiac muscle
Lutz, Michael W., Morgan, Paul H., Kenakin, Terry P., Goetz, Aaron, Queen, Kennedy, Irving, Paul, Rose, Dudley, Gill, James M., Rimele, Tom
Published in Journal of pharmacological and toxicological methods (01.11.1996)
Published in Journal of pharmacological and toxicological methods (01.11.1996)
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Do catecholamines contribute to the effects of neonatal hypoxia on development of brain and heart? Influence of concurrent alpha-adrenergic blockade on ornithine decarboxylase activity
Slotkin, T A, Orband-Miller, L, Queen, K L
Published in International journal of developmental neuroscience (1987)
Published in International journal of developmental neuroscience (1987)
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