Covalent Trapping of Methyllycaconitine at the α4-α4 Interface of the α4β2 Nicotinic Acetylcholine Receptor
Absalom, Nathan L., Quek, Gracia, Lewis, Trevor M., Qudah, Taima, von Arenstorff, Ida, Ambrus, Joseph I., Harpsøe, Kasper, Karim, Nasiara, Balle, Thomas, Mcleod, Malcolm D., Chebib, Mary
Published in The Journal of biological chemistry (01.09.2013)
Published in The Journal of biological chemistry (01.09.2013)
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Revisiting autosomal dominant nocturnal frontal lobe epilepsy (ADNFLE) mutations in the nicotinic acetylcholine receptor reveal an increase in efficacy regardless of stochiometry
Indurthi, Dinesh C., Qudah, Taima, Liao, Vivian W., Ahring, Philip K., Lewis, Trevor M., Balle, Thomas, Chebib, Mary, Absalom, Nathan L.
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Published in Pharmacological research (01.01.2019)
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AE Succinimide, an Analogue of Methyllycaconitine, When Bound Generates a Nonconducting Conformation of the α4β2 Nicotinic Acetylcholine Receptor
Qudah, Taima, Quek, Gracia X, Indurthi, Dinesh, Karim, Nasiara, Halliday, Jill I, Absalom, Nathan, McLeod, Malcolm D, Chebib, Mary
Published in ACS chemical neuroscience (05.02.2020)
Published in ACS chemical neuroscience (05.02.2020)
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Covalent trapping of methyllycaconitine at the α4-α4 interface of the α4β2 nicotinic acetylcholine receptor: antagonist binding site and mode of receptor inhibition revealed
Absalom, Nathan L, Quek, Gracia, Lewis, Trevor M, Qudah, Taima, von Arenstorff, Ida, Ambrus, Joseph I, Harpsøe, Kasper, Karim, Nasiara, Balle, Thomas, McLeod, Malcolm D, Chebib, Mary
Published in The Journal of biological chemistry (13.09.2013)
Published in The Journal of biological chemistry (13.09.2013)
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An additional binding site for methyllycaconitine (MLA) and analogs occurs at the α4–α4 interface of the (α4)3(β2)2 nAChR
Chebib, Mary, Absalom, Nathan L., Quek, Gracia, Indurthi, Dinesh, Lewis, Trevor M., Qudah, Taima, von Arenstorff, Ida, Halliday, Jill I., Ambrus, Joseph I., Harpsøe, Kasper, Karim, Nasiara, Balle, Thomas, Mcleod, Malcolm D.
Published in Biochemical pharmacology (15.10.2013)
Published in Biochemical pharmacology (15.10.2013)
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