A patent review of transient receptor potential vanilloid type 1 modulators (2014-present)
Gao, Mengkang, Wang, Yusui, Liu, Lanqi, Qiao, Zhenrui, Yan, Lin
Published in Expert opinion on therapeutic patents (01.02.2021)
Published in Expert opinion on therapeutic patents (01.02.2021)
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Journal Article
Discovery of (S)–N-(3-isopropylphenyl)-2-(5-phenylthiazol-2-yl)pyrrolidine-1-carboxamide as potent and brain-penetrant TRPV1 antagonist
Qiao, Yue, Zhang, Yang, Qiao, Zhenrui, He, Wenya, Chen, Yingda, Song, Depu, Wang, Guohao, Guo, Ning, Shao, Lulian, Tian, Zhiyong, Wang, Qiang, Yan, Lin, Qian, Hai
Published in European journal of medicinal chemistry (05.04.2022)
Published in European journal of medicinal chemistry (05.04.2022)
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Journal Article
Novel dual-target FAAH and TRPV1 ligands as potential pharmacotherapeutics for pain management
Qiao, Zhenrui, Liu, Shuyu, zhai, Weibin, Jiang, Lei, Ma, Yunmeng, Zhang, Zhikang, Wang, Bingxin, Shao, Jingwen, Qian, Hai, Zhao, Fenqin, Yan, Lin
Published in European journal of medicinal chemistry (05.03.2024)
Published in European journal of medicinal chemistry (05.03.2024)
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Journal Article
Study on chemical modification and analgesic activity of N-(4-tert-butylphenyl)-4-(3-chloropyridin-2-yl) piperazine-1-carboxamide
Nie, Cunbin, Li, Qifei, Qiao, Yue, Hu, Jing, Gao, Mengkang, Wang, Yusui, Qiao, Zhenrui, Wang, Qiang, Yan, Lin, Qian, Hai
Published in European journal of medicinal chemistry (15.05.2020)
Published in European journal of medicinal chemistry (15.05.2020)
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Journal Article
Novel piperazine urea derivatives as highly potent transient receptor potential vanilloid 1 (TRPV1) antagonists
Hu, Jing, Gao, Mengkang, Zhang, Yang, Wang, Yusui, Qiao, Zhenrui, Zhang, Weiya, Wang, Qiang, Yan, Lin, Qian, Hai
Published in Bioorganic chemistry (01.10.2021)
Published in Bioorganic chemistry (01.10.2021)
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Journal Article
Novel TRPV1 antagonism/FAAH inhibition double-target drug, and preparation method and application thereof
GAO MENGKANG, CHEN YINGDA, SONG DEPU, QIAO ZHENRUI, WANG GUOHAO, YAN LIN, WANG YUSUI
Year of Publication 10.08.2021
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Year of Publication 10.08.2021
Patent
A wear -resisting tee bend that is used for high temperature high pressure condition to use
CAO PEIKUAN, BAI JIZHAO, QIAO ZHENRUI, LIU YANG, YANG SHAOFEI, DU FANGHONG, ZHANG NAN
Year of Publication 19.04.2017
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Year of Publication 19.04.2017
Patent