Discovery of PiragliatinFirst Glucokinase Activator Studied in Type 2 Diabetic Patients
Sarabu, Ramakanth, Bizzarro, Fred T, Corbett, Wendy L, Dvorozniak, Mark T, Geng, Wanping, Grippo, Joseph F, Haynes, Nancy-Ellen, Hutchings, Stanley, Garofalo, Lisa, Guertin, Kevin R, Hilliard, Darryl W, Kabat, Marek, Kester, Robert F, Ka, Wang, Liang, Zhenmin, Mahaney, Paige E, Marcus, Linda, Matschinsky, Franz M, Moore, David, Racha, Jagdish, Radinov, Roumen, Ren, Yi, Qi, Lida, Pignatello, Michael, Spence, Cheryl L, Steele, Thomas, Tengi, John, Grimsby, Joseph
Published in Journal of medicinal chemistry (23.08.2012)
Published in Journal of medicinal chemistry (23.08.2012)
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Journal Article
Allosteric Activators of Glucokinase: Potential Role in Diabetes Therapy
Grimsby, Joseph, Sarabu, Ramakanth, Corbett, Wendy L., Haynes, Nancy-Ellen, Bizzarro, Fred T., Coffey, John W., Guertin, Kevin R., Hilliard, Darryl W., Kester, Robert F., Mahaney, Paige E., Marcus, Linda, Qi, Lida, Spence, Cheryl L., Tengi, John, Magnuson, Mark A., Chu, Chang An, Dvorozniak, Mark T., Matschinsky, Franz M., Grippo, Joseph F.
Published in Science (American Association for the Advancement of Science) (18.07.2003)
Published in Science (American Association for the Advancement of Science) (18.07.2003)
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Journal Article
4-Substituted-7-N-alkyl-N-acetyl 2-aminobenzothiazole amides: Drug-like and non-xanthine based A2B adenosine receptor antagonists
Cheung, Adrian Wai-Hing, Brinkman, John, Firooznia, Fariborz, Flohr, Alexander, Grimsby, Joseph, Gubler, Mary Lou, Guertin, Kevin, Hamid, Rachid, Marcopulos, Nicholas, Norcross, Roger D., Qi, Lida, Ramsey, Gwendolyn, Tan, Jenny, Wen, Yang, Sarabu, Ramakanth
Published in Bioorganic & medicinal chemistry letters (15.07.2010)
Published in Bioorganic & medicinal chemistry letters (15.07.2010)
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Journal Article
Identification of a novel class of orally active pyrimido[5,4-3][1,2,4]triazine-5,7-diamine-based hypoglycemic agents with protein tyrosine phosphatase inhibitory activity
Guertin, Kevin R., Setti, Lina, Qi, Lida, Dunsdon, Rachel M., Dymock, Brian W., Jones, Philip S., Overton, Hilary, Taylor, Mathew, Williams, Glyn, Sergi, Joseph A., Wang, Karen, Peng, Ying, Renzetti, Marcia, Boyce, Rogely, Falcioni, Fiorenza, Garippa, Ralph, Olivier, Andrée R.
Published in Bioorganic & medicinal chemistry letters (01.09.2003)
Published in Bioorganic & medicinal chemistry letters (01.09.2003)
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Journal Article
Structure-activity relationship of linear peptide Bu-His-DPhe-Arg-Trp-Gly-NH2 at the human melanocortin-1 and -4 receptors: Arginine substitution
CHEUNG, Adrian Wai-Hing, DANHO, Waleed, SWISTOK, Joseph, QI, Lida, KURYLKO, Grazyna, FRANCO, Lucia, YAGALOFF, Keith, LI CHEN
Published in Bioorganic & medicinal chemistry letters (02.09.2002)
Published in Bioorganic & medicinal chemistry letters (02.09.2002)
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Journal Article
Discovery of 1-amino-4-phenylcyclohexane-1-carboxylic acid and its influence on agonist selectivity between human melanocortin-4 and -1 receptors in linear pentapeptides
Chu, Xin-Jie, Bartkovitz, David, Danho, Waleed, Swistok, Joseph, Cheung, Adrian Wai-Hing, Kurylko, Grazyna, Rowan, Karen, Yeon, Mitch, Franco, Lucia, Qi, Lida, Chen, Li, Yagaloff, Keith
Published in Bioorganic & medicinal chemistry letters (15.11.2005)
Published in Bioorganic & medicinal chemistry letters (15.11.2005)
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Journal Article
Structure-activity relationship of linear peptide Bu-His-DPhe-Arg-Trp-Gly-NH2 at the human melanocortin-1 and -4 receptors: Histidine substitution
CHEUNG, Adrian Wai-Hing, DANHO, Waleed, YAGALOFF, Keith, SWISTOK, Joseph, LIDA QI, KURYLKO, Grazyna, ROWAN, Karen, YEON, Mitch, FRANCO, Lucia, CHU, Xin-Jie, LI CHEN
Published in Bioorganic & medicinal chemistry letters (06.01.2003)
Published in Bioorganic & medicinal chemistry letters (06.01.2003)
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Journal Article
Preparation of human Melanocortin-4 receptor agonist libraries : Linear peptides X-Y-DPhe7-Arg8-Trp(or 2-Nal)9-Z-NH2
CHEUNG, Adrian Wai-Hing, LIDA QI, GORE, Vijay, CHU, Xin-Jie, BARTKOVITZ, David, KURYLKO, Grazyna, SWISTOK, Joseph, DANHO, Waleed, LI CHEN, YAGALOFF, Keith
Published in Bioorganic & medicinal chemistry letters (15.12.2005)
Published in Bioorganic & medicinal chemistry letters (15.12.2005)
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Journal Article
Discovery, Structure−Activity Relationships, Pharmacokinetics, and Efficacy of Glucokinase Activator (2R)-3-Cyclopentyl-2-(4-methanesulfonylphenyl)-N-thiazol-2-yl-propionamide (RO0281675)
Haynes, Nancy-Ellen, Corbett, Wendy L, Bizzarro, Fred T, Guertin, Kevin R, Hilliard, Darryl W, Holland, George W, Kester, Robert F, Mahaney, Paige E, Qi, Lida, Spence, Cheryl L, Tengi, John, Dvorozniak, Mark T, Railkar, Aruna, Matschinsky, Franz M, Grippo, Joseph F, Grimsby, Joseph, Sarabu, Ramakanth
Published in Journal of medicinal chemistry (13.05.2010)
Published in Journal of medicinal chemistry (13.05.2010)
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Journal Article
Discovery of camphor-derived pyrazolones as 11β-hydroxysteroid dehydrogenase type 1 inhibitors
Gillespie, Paul, Pietranico-Cole, Sherrie, Myers, Michael, Bilotta, Joseph A., Conde-Knape, Karin, Fotouhi, Nader, Goodnow, Robert A., Guertin, Kevin R., Hamilton, Matthew M., Haynes, Nancy-Ellen, Liu, Baolian, Qi, Lida, Ren, Yonglin, Scott, Nathan R., So, Sung-Sau, Spence, Cheryl, Taub, Rebecca, Thakkar, Kshitij, Tilley, Jefferson W., Zwingelstein, Catherine
Published in Bioorganic & medicinal chemistry letters (15.06.2014)
Published in Bioorganic & medicinal chemistry letters (15.06.2014)
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Journal Article
Structure-activity relationship of cyclic peptide Penta-c[Asp-His6-DPhe7-Arg8-Trp9-Lys]-NH2 at the human melanocortin-1 and -4 receptors: His6 substitution
WAI-HING CHEUNG, Adrian, DANHO, Waleed, YAGALOFF, Keith, SWISTOK, Joseph, QI, Lida, KURYLKO, Grazyna, ROWAN, Karen, YEON, Mitch, FRANCO, Lucia, CHU, Xin-Jie, LI CHEN
Published in Bioorganic & medicinal chemistry letters (01.04.2003)
Published in Bioorganic & medicinal chemistry letters (01.04.2003)
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Journal Article
4-Substituted-7-N-alkyl-N-acetyl 2-aminobenzothiazole amides: Drug-like and non-xanthine based A sub(2B) adenosine receptor antagonists
Cheung, Adrian Wai-Hing, Brinkman, John, Firooznia, Fariborz, Flohr, Alexander, Grimsby, Joseph, Gubler, Mary Lou, Guertin, Kevin, Hamid, Rachid, Marcopulos, Nicholas, Norcross, Roger D, Qi, Lida, Ramsey, Gwendolyn, Tan, Jenny, Wen, Yang, Sarabu, Ramakanth
Published in Bioorganic & medicinal chemistry letters (15.07.2010)
Published in Bioorganic & medicinal chemistry letters (15.07.2010)
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Journal Article
Preparation of human Melanocortin-4 receptor agonist libraries: Linear peptides X-Y-DPhe 7-Arg 8-Trp(or 2-Nal) 9-Z-NH 2
Cheung, Adrian Wai-Hing, Qi, Lida, Gore, Vijay, Chu, Xin-Jie, Bartkovitz, David, Kurylko, Grazyna, Swistok, Joseph, Danho, Waleed, Chen, Li, Yagaloff, Keith
Published in Bioorganic & medicinal chemistry letters (2005)
Published in Bioorganic & medicinal chemistry letters (2005)
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Journal Article
Structure-activity relationship of linear peptide Bu-His-DPhe-Arg-Trp-Gly-NH(2) at the human melanocortin-1 and -4 receptors: arginine substitution
Cheung, Adrian Wai-Hing, Danho, Waleed, Swistok, Joseph, Qi, Lida, Kurylko, Grazyna, Franco, Lucia, Yagaloff, Keith, Chen, Li
Published in Bioorganic & medicinal chemistry letters (02.09.2002)
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Published in Bioorganic & medicinal chemistry letters (02.09.2002)
Journal Article
Structure-activity relationship of cyclic peptide penta-c[Asp-His(6)-DPhe(7)-Arg(8)-Trp(9)-Lys]-NH(2) at the human melanocortin-1 and -4 receptors: His(6) substitution
Cheung, Adrian Wai-Hing, Danho, Waleed, Swistok, Joseph, Qi, Lida, Kurylko, Grazyna, Rowan, Karen, Yeon, Mitch, Franco, Lucia, Chu, Xin-Jie, Chen, Li, Yagaloff, Keith
Published in Bioorganic & medicinal chemistry letters (07.04.2003)
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Published in Bioorganic & medicinal chemistry letters (07.04.2003)
Journal Article
Structure-activity relationship of linear peptide Bu-His-DPhe-Arg-Trp-Gly-NH(2) at the human melanocortin-1 and -4 receptors: histidine substitution
Cheung, Adrian Wai-Hing, Danho, Waleed, Swistok, Joseph, Qi, Lida, Kurylko, Grazyna, Rowan, Karen, Yeon, Mitch, Franco, Lucia, Chu, Xin-Jie, Chen, Li, Yagaloff, Keith
Published in Bioorganic & medicinal chemistry letters (06.01.2003)
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Published in Bioorganic & medicinal chemistry letters (06.01.2003)
Journal Article
Structure–Activity relationship of linear peptide Bu-His-DPhe-Arg-Trp-Gly-NH 2 at the human melanocortin-1 and -4 receptors: histidine substitution
Cheung, Adrian Wai-Hing, Danho, Waleed, Swistok, Joseph, Qi, Lida, Kurylko, Grazyna, Rowan, Karen, Yeon, Mitch, Franco, Lucia, Chu, Xin-Jie, Chen, Li, Yagaloff, Keith
Published in Bioorganic & medicinal chemistry letters (2003)
Published in Bioorganic & medicinal chemistry letters (2003)
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Journal Article
Structure–activity relationship of cyclic peptide penta-c[Asp-His 6-DPhe 7-Arg 8-Trp 9-Lys]-NH 2 at the human melanocortin-1 and -4 receptors: His 6 substitution
Cheung, Adrian Wai-Hing, Danho, Waleed, Swistok, Joseph, Qi, Lida, Kurylko, Grazyna, Rowan, Karen, Yeon, Mitch, Franco, Lucia, Chu, Xin-Jie, Chen, Li, Yagaloff, Keith
Published in Bioorganic & medicinal chemistry letters (2003)
Published in Bioorganic & medicinal chemistry letters (2003)
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Journal Article
Structure–Activity relationship of linear peptide Bu-His-DPhe-Arg-Trp-Gly-NH 2 at the human melanocortin-1 and -4 receptors: arginine substitution
Cheung, Adrian Wai-Hing, Danho, Waleed, Swistok, Joseph, Qi, Lida, Kurylko, Grazyna, Franco, Lucia, Yagaloff, Keith, Chen, Li
Published in Bioorganic & medicinal chemistry letters (2002)
Published in Bioorganic & medicinal chemistry letters (2002)
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Journal Article