A new wave of innovations within the DNA damage response
Li, Qi, Qian, Wenyuan, Zhang, Yang, Hu, Lihong, Chen, Shuhui, Xia, Yuanfeng
Published in Signal transduction and targeted therapy (08.09.2023)
Published in Signal transduction and targeted therapy (08.09.2023)
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Journal Article
Discovery of dihydroquinoxalinone acetamides containing bicyclic amines as potent Bradykinin B1 receptor antagonists
Chen, Jian Jeffrey, Qian, Wenyuan, Biswas, Kaustav, Viswanadhan, Vellarkad N., Askew, Benny C., Hitchcock, Stephen, Hungate, Randall W., Arik, Leyla, Johnson, Eileen
Published in Bioorganic & medicinal chemistry (15.08.2008)
Published in Bioorganic & medicinal chemistry (15.08.2008)
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Journal Article
Total Synthesis and Structural Elucidation of Azaspiracid-1. Construction of Key Building Blocks for Originally Proposed Structure
Nicolaou, K. C, Pihko, Petri M, Bernal, Federico, Frederick, Michael O, Qian, Wenyuan, Uesaka, Noriaki, Diedrichs, Nicole, Hinrichs, Jürgen, Koftis, Theocharis V, Loizidou, Eriketi, Petrovic, Goran, Rodriquez, Manuela, Sarlah, David, Zou, Ning
Published in Journal of the American Chemical Society (22.02.2006)
Published in Journal of the American Chemical Society (22.02.2006)
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Journal Article
Discovery of dehydro-oxopiperazine acetamides as novel bradykinin B1 receptor antagonists with enhanced in vitro potency
Qian, Wenyuan, Chen, Jian Jeffrey, Human, Jason, Aya, Toshihiro, Zhu, Jiawang, Biswas, Kaustav, Peterkin, Tanya, Hungate, Randall W., Arik, Leyla, Johnson, Eileen, Kumar, Gondi, Joseph, Smriti, Jona, Janan, Guo, Hong-Xun, Wu, Zufan
Published in Bioorganic & medicinal chemistry letters (15.01.2012)
Published in Bioorganic & medicinal chemistry letters (15.01.2012)
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Journal Article
Synthesis of Stable Derivatives of C62: The First Nonclassical Fullerene Incorporating a Four-Membered Ring
Qian, Wenyuan, Chuang, Shih-Ching, Amador, Roberto B, Jarrosson, Thibaut, Sander, Michael, Pieniazek, Susan, Khan, Saeed I, Rubin, Yves
Published in Journal of the American Chemical Society (26.02.2003)
Published in Journal of the American Chemical Society (26.02.2003)
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Journal Article
Total Synthesis of the Proposed Azaspiracid-1 Structure, Part 1: Construction of the Enantiomerically Pure C1-C20, C21-C27, and C28-C40 Fragments
Nicolaou, K. C., Li, Yiwei, Uesaka, Noriaki, Koftis, Theocharis V., Vyskocil, Stepan, Ling, Taotao, Govindasamy, Mugesh, Qian, Wenyuan, Bernal, Federico, Chen, David Y.-K.
Published in Angewandte Chemie (International ed.) (11.08.2003)
Published in Angewandte Chemie (International ed.) (11.08.2003)
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Journal Article
3-Oxo-2-piperazinyl acetamides as potent bradykinin B1 receptor antagonists for the treatment of pain and inflammation
Chen, Jian Jeffrey, Nguyen, Thomas, D’Amico, Derin C., Qian, Wenyuan, Human, Jason, Aya, Toshihiro, Biswas, Kaustav, Fotsch, Christopher, Han, Nianhe, Liu, Qingyian, Nishimura, Nobuko, Peterkin, Tanya A.N., Yang, Kevin, Zhu, Jiawang, Riahi, Babak Bobby, Hungate, Randall W., Andersen, Neil G., Colyer, John T., Faul, Margaret M., Kamassah, Augustus, Wang, Judy, Jona, Janan, Kumar, Gondi, Johnson, Eileen, Askew, Benny C.
Published in Bioorganic & medicinal chemistry letters (01.06.2011)
Published in Bioorganic & medicinal chemistry letters (01.06.2011)
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Journal Article
Aryl sulfones as novel Bradykinin B1 receptor antagonists for treatment of chronic pain
Biswas, Kaustav, Aya, Toshihiro, Qian, Wenyuan, Peterkin, Tanya A.N., Chen, Jian Jeffrey, Human, Jason, Hungate, Randall W., Kumar, Gondi, Arik, Leyla, Lester-Zeiner, Dianna, Biddlecome, Gloria, Manning, Barton H., Sun, Hong, Dong, Hong, Huang, Ming, Loeloff, Richard, Johnson, Eileen J., Askew, Benny C.
Published in Bioorganic & medicinal chemistry (01.09.2008)
Published in Bioorganic & medicinal chemistry (01.09.2008)
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Journal Article
Aryl sulfonamides containing tetralin allylic amines as potent and selective bradykinin B1 receptor antagonists
Liu, Qingyian, Qian, Wenyuan, Li, Aiwen, Biswas, Kaustav, Chen, Jian Jeffrey, Fotsch, Christopher, Han, Nianhe, Yuan, Chester, Arik, Leyla, Biddlecome, Gloria, Johnson, Eileen, Kumar, Gondi, Lester-Zeiner, Dianna, Ng, Gordon Y., Hungate, Randall W., Askew, Benny C.
Published in Bioorganic & medicinal chemistry letters (01.08.2010)
Published in Bioorganic & medicinal chemistry letters (01.08.2010)
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Journal Article
One-Pot Synthesis of 3‑Triazolyl-2-iminochromenes via a Catalytic Three Component Cascade Reaction
Qian, Wenyuan, Amegadzie, Albert, Winternheimer, David, Allen, Jennifer
Published in Organic letters (21.06.2013)
Published in Organic letters (21.06.2013)
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Journal Article
Identification of TUL01101: A Novel Potent and Selective JAK1 Inhibitor for the Treatment of Rheumatoid Arthritis
Zhou, Shuhao, Mao, Weiwei, Su, Yuan, Zheng, Xuejian, Qian, Wenyuan, Shen, Meiyue, Shan, Ningli, Li, Yaoshuang, Wang, Degang, Wu, Shouting, Sun, Tiemin, Mu, Liwei
Published in Journal of medicinal chemistry (22.12.2022)
Published in Journal of medicinal chemistry (22.12.2022)
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Journal Article
Synthesis and evaluation of hydrazinyl-containing pyrrolo[2,3-d]pyrimidine series as potent, selective and oral JAK1 inhibitors for the treatment of rheumatoid arthritis
Mao, Weiwei, Wu, Hao, Guo, Qiang, Zheng, Xuejian, Wei, Changqing, Liao, Yonggang, Shen, Liang, Mi, Jingyu, Li, Jian, Chen, Shuhui, Qian, Wenyuan
Published in Bioorganic & medicinal chemistry letters (15.10.2022)
Published in Bioorganic & medicinal chemistry letters (15.10.2022)
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Journal Article