UPLC-based assay to assess the hydrophobicity of Antibody-Drug Conjugate (ADC) payloads
Pysz, Ilona, Jackson, Paul J.M., Barlow, David J., Rahman, Khondaker Miraz, Thurston, David E.
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (01.06.2020)
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (01.06.2020)
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Journal Article
Abstract 211: A new class of sequence-selective DNA cross-linking ADC payloads with increased in vivo tolerability
Procopiou, George, Auer, Jennifer, Mascio, Daniella di, Fox, Keith R., Andriollo, Paolo, Pysz, Ilona, Cascio, Francesco, Veillard, Nicolas, Rahman, K. Miraz, Jackson, Paul J., Thurston, David E.
Published in Cancer research (Chicago, Ill.) (01.07.2019)
Published in Cancer research (Chicago, Ill.) (01.07.2019)
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Journal Article
Use of pyrrolobenzodiazepines and related covalent-binding DNA-interactive molecules as ADC payloads: Is mechanism related to systemic toxicity?
Jackson, Paul J.M., Kay, Syafiq, Pysz, Ilona, Thurston, David E.
Published in Drug discovery today. Technologies (01.12.2018)
Published in Drug discovery today. Technologies (01.12.2018)
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Journal Article
Abstract 736: Pyridinobenzodiazepines (PDDs): A new class of sequence-selective DNA mono-alkylating ADC payloads with low hydrophobicity
Veillard, Nicolas, Andriollo, Paolo, Mantaj, Julia, Fox, Keith R., Rahman, K Miraz, Procopiou, George, Cascio, Francesco, Corcoran, David B., Pysz, Ilona, Cooper, Patricia A., Shnyder, Steven D., Ju, Yawen, Tan, Edwin, Schopperle, William M., Jackson, Paul J., Thurston, David E.
Published in Cancer research (Chicago, Ill.) (01.07.2018)
Published in Cancer research (Chicago, Ill.) (01.07.2018)
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Journal Article
Abstract 1749: A new class of DNA sequence-selective G-A cross-linking antibody-drug conjugate (ADC) payloads
Procopiou, George, Jackson, Paul J., di Mascio, Daniella M., Auer, Jennifer L., Andriollo, Paolo, Pysz, Ilona, Rahman, Khondaker M., Fox, Keith R., Thurston, David E.
Published in Cancer research (Chicago, Ill.) (15.06.2022)
Published in Cancer research (Chicago, Ill.) (15.06.2022)
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