Novel Derivatives of Eugenol as a New Class of PPARγ Agonists in Treating Inflammation: Design, Synthesis, SAR Analysis and In Vitro Anti-Inflammatory Activity
Anjum, Noor Fathima, Shanmugarajan, Dhivya, Prashantha Kumar, B R, Faizan, Syed, Durai, Priya, Raju, Ruby Mariam, Javid, Saleem, Purohit, Madhusudan N
Published in Molecules (Basel, Switzerland) (05.05.2023)
Published in Molecules (Basel, Switzerland) (05.05.2023)
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Synthesis, characterization, and anti-cancer potential of novel p53-mediated Mdm2 and Pirh2 modulators: an integrated In silico and In vitro approach
Niazi, Sarfaraj, Kavana, C P, Aishwarya, H K, Dharmashekar, Chandan, Jain, Anisha, Wani, Tanveer A, Shivamallu, Chandan, Purohit, Madhusudan N, Kollur, Shiva Prasad
Published in Frontiers in chemistry (16.07.2024)
Published in Frontiers in chemistry (16.07.2024)
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Discovery of Novel Myristic Acid Derivatives as N-Myristoyltransferase Inhibitors: Design, Synthesis, Analysis, Computational Studies and Antifungal Activity
Javid, Saleem, Ather, Hissana, Hani, Umme, Siddiqua, Ayesha, Asif Ansari, Shaik Mohammad, Shanmugarajan, Dhivya, Yogish Kumar, Honnavalli, Arivuselvam, Rajaguru, Purohit, Madhusudan N, Kumar, B R Prashantha
Published in Antibiotics (Basel) (01.07.2023)
Published in Antibiotics (Basel) (01.07.2023)
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Synthesis and in vitro cytotoxicity studies of certain novel heterocycles derived from bis 1, 2, 4-triazoles and their DNA damage studies
Purohit, Madhusudan N, Mangannavar, Chandrashekhar Venkaraddi, Yergeri, Mayur C
Published in Medicinal chemistry (Shp-sariqah, United Arab Emirates) (01.12.2013)
Published in Medicinal chemistry (Shp-sariqah, United Arab Emirates) (01.12.2013)
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Journal Article
Rational design, synthesis, analysis and antifungal activity of novel myristic acid derivatives as N-myristoyltransferase inhibitors
Javid, Saleem, Shanmugarajan, Dhivya, Kumar, H. Yogish, Arivuselvam, Rajaguru, Anjum, Noor Fathima, Purohit, Madhusudan N, Susil, Aishwarya, Harindranath, Haritha, Nilugal, Kiran C., Nagojappa, Narendra Babu Shivanagere, Kumar, B.R. Prashantha
Published in Journal of molecular structure (05.05.2024)
Published in Journal of molecular structure (05.05.2024)
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Design, synthesis and 3D-QSAR studies of new diphenylamine containing 1,2,4-triazoles as potential antitubercular agents
Mohan Krishna, K., Inturi, Bharathkumar, Pujar, Gurubasavaraj V., Purohit, Madhusudan N., Vijaykumar, G.S.
Published in European journal of medicinal chemistry (12.09.2014)
Published in European journal of medicinal chemistry (12.09.2014)
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Journal Article
Novel derivatives of eugenol as potent anti-inflammatory agents via PPARγ agonism: rational design, synthesis, analysis, PPARγ protein binding assay and computational studies
Anjum, Noor Fathima, Shanmugarajan, Dhivya, Shivaraju, Vasanth Kumar, Faizan, Syed, Naishima, Namburu Lalitha, Prashantha Kumar, B. R., Javid, Saleem, Purohit, Madhusudan N.
Published in RSC advances (01.06.2022)
Published in RSC advances (01.06.2022)
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In-Vitro Cytotoxicity and Cell Cycle Analysis of Two Novel bis-1,2, 4-triazole derivatives: 1,4-bis[5-(5-mercapto-1,3,4-oxadiazol-2-yl-methyl)-thio-4-(p-tolyl)-1,2,4-triazol-3-yl]-butane (MNP-14) and 1,4-bis[5-(carbethoxy-methyl)-thio-4-(p-ethoxy phenyl)-1,2,4-triazol-3-yl]-butane (MNP-16)
Purohit, Madhusudan N., Panjamurthy, Kuppusamy, Elango, Santhini, Hebbar, Karteek, Mayur, Yergeri C., Raghavan, Sathees C.
Published in Nucleosides, nucleotides & nucleic acids (01.11.2011)
Published in Nucleosides, nucleotides & nucleic acids (01.11.2011)
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Journal Article
Novel derivatives of eugenol as potent anti-inflammatory agents PPARγ agonism: rational design, synthesis, analysis, PPARγ protein binding assay and computational studies
Anjum, Noor Fathima, Shanmugarajan, Dhivya, Shivaraju, Vasanth Kumar, Faizan, Syed, Naishima, Namburu Lalitha, Prashantha Kumar, B. R, Javid, Saleem, Purohit, Madhusudan N
Published in RSC advances (07.06.2022)
Published in RSC advances (07.06.2022)
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Journal Article
Semisynthetic Derivatives of Eugenol and their Biological Properties: A Fleeting Look at the Promising Molecules
Anjum, Noor Fathima, Purohit, Madhusudan N., Yogish Kumar, H., Ramya, K., Javid, Saleem, Salahuddin, M.D., Prashantha Kumar, B.R.
Published in Journal of biologically active products from nature (02.09.2020)
Published in Journal of biologically active products from nature (02.09.2020)
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Journal Article
Semisynthesis of Myristic Acid Derivatives and their Biological Activities: A Critical Insight
Javid, Saleem, Purohit, Madhusudan N., Yogish Kumar, H., Ramya, K., Mithuna, Noor Fathima Anjum, Salahuddin, M.D., Prashantha Kumar, B.R.
Published in Journal of biologically active products from nature (01.11.2020)
Published in Journal of biologically active products from nature (01.11.2020)
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Journal Article
Design, synthesis and 3D-QSAR studies of new diphenylamine containing 1,2,4-triazoles as potential antitubercular agents
Mohan Krishna, K., Inturi, Bharathkumar, Pujar, Gurubasavaraj V., Purohit, Madhusudan N., Vijaykumar, G.S.
Published in European journal of medicinal chemistry (01.09.2014)
Published in European journal of medicinal chemistry (01.09.2014)
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Journal Article