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Published in Proceedings of the National Academy of Sciences - PNAS (14.08.2018)
Published in Proceedings of the National Academy of Sciences - PNAS (14.08.2018)
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Selective Janus Kinase 2 (JAK2) Pseudokinase Ligands with a Diaminotriazole Core
Liosi, Maria-Elena, Krimmer, Stefan G, Newton, Ana S, Dawson, Thomas K, Puleo, David E, Cutrona, Kara J, Suzuki, Yoshihisa, Schlessinger, Joseph, Jorgensen, William L
Published in Journal of medicinal chemistry (28.05.2020)
Published in Journal of medicinal chemistry (28.05.2020)
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Indoloxytriazines as binding molecules for the JAK2 JH2 pseudokinase domain and its V617F variant
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Published in Tetrahedron letters (03.08.2021)
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Regulated induced proximity targeting chimeras—RIPTACs—A heterobifunctional small molecule strategy for cancer selective therapies
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Published in Cell chemical biology (15.08.2024)
Published in Cell chemical biology (15.08.2024)
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Structure-Based Evaluation of Non-nucleoside Inhibitors with Improved Potency and Solubility That Target HIV Reverse Transcriptase Variants
Frey, Kathleen M, Puleo, David E, Spasov, Krasimir A, Bollini, Mariella, Jorgensen, William L, Anderson, Karen S
Published in Journal of medicinal chemistry (26.03.2015)
Published in Journal of medicinal chemistry (26.03.2015)
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Identification and Characterization of JAK2 Pseudokinase Domain Small Molecule Binders
Puleo, David E, Kucera, Kaury, Hammarén, Henrik M, Ungureanu, Daniela, Newton, Ana S, Silvennoinen, Olli, Jorgensen, William L, Schlessinger, Joseph
Published in ACS medicinal chemistry letters (08.06.2017)
Published in ACS medicinal chemistry letters (08.06.2017)
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JAK2 JH2 Fluorescence Polarization Assay and Crystal Structures for Complexes with Three Small Molecules
Newton, Ana S, Deiana, Luca, Puleo, David E, Cisneros, José A, Cutrona, Kara J, Schlessinger, Joseph, Jorgensen, William L
Published in ACS medicinal chemistry letters (08.06.2017)
Published in ACS medicinal chemistry letters (08.06.2017)
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Patenting the microbiome: trends, challenges and insights
Sabatelli, Anthony D, Vincent, Nicholas G, Puleo, David E
Published in Pharmaceutical patent analyst (01.11.2017)
Published in Pharmaceutical patent analyst (01.11.2017)
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Regulated Induced Proximity Targeting Chimeras (RIPTACs): a Novel Heterobifunctional Small Molecule Therapeutic Strategy for Killing Cancer Cells Selectively
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Published in bioRxiv (02.01.2023)
Published in bioRxiv (02.01.2023)
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Year of Publication 13.04.2023
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HETEROBIFUNCTIONAL COMPOUNDS AND METHODS OF TREATING DISEASE
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Year of Publication 14.03.2024
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Year of Publication 14.03.2024
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Year of Publication 14.03.2024
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Year of Publication 14.03.2024
Patent
HETEROBIFUNCTIONAL COMPOUNDS AND METHODS OF TREATING DISEASE
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Year of Publication 14.03.2024
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GERRITZ, Samuel W, KAYSER-BRICKER, Katherine J, PULEO, David E, EASTMAN, Kyle J, CHEN, Jinshan M, CREWS, Craig
Year of Publication 17.11.2021
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Year of Publication 17.11.2021
Patent