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Published in Life (Basel, Switzerland) (01.10.2023)
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BV-2 Microglial Cells Respond to Rotenone Toxic Insult by Modifying Pregnenolone, 5α-Dihydroprogesterone and Pregnanolone Levels
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Published in Cells (Basel, Switzerland) (13.09.2020)
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Modulation of NMDA receptor activity by CR4056, an imidazoline-2 receptor ligand with analgesic properties
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Synthesis and Anticonvulsant Activity of Novel and Potent 6,7-Methylenedioxyphthalazin-1(2H)-ones
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Published in Journal of medicinal chemistry (27.07.2000)
Published in Journal of medicinal chemistry (27.07.2000)
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Novel Potent AMPA/Kainate Receptor Antagonists: Synthesis and Anticonvulsant Activity of a Series of 2-[(4-Alkylsemicarbazono)-(4-amino- phenyl)methyl]-4,5-methylenedioxyphenylacetic Acid Alkyl Esters
Micale, Nicola, Zappalà, Maria, Grasso, Silvana, Puja, Giulia, De Sarro, Giovambattista, Ferreri, Guido, De Sarro, Angela, Toma, Lucio, De Micheli, Carlo
Published in Journal of medicinal chemistry (26.09.2002)
Published in Journal of medicinal chemistry (26.09.2002)
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Novel Dithiolane-Based Ligands Combining Sigma and NMDA Receptor Interactions as Potential Neuroprotective Agents
Franchini, Silvia, Linciano, Pasquale, Puja, Giulia, Tait, Annalisa, Borsari, Chiara, Denora, Nunzio, Iacobazzi, Rosa Maria, Brasili, Livio, Sorbi, Claudia
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Published in ACS medicinal chemistry letters (14.05.2020)
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BV-2 Microglial Cells Respond to Rotenone Toxic Insult by Modifying Pregnenolone, 5[alpha]-Dihydroprogesterone and Pregnanolone Levels
Avallone, Rossella, Lucchi, Chiara, Puja, Giulia, Codeluppi, Alessandro, Filaferro, Monica, Vitale, Giovanni, Rustichelli, Cecilia, Biagini, Giuseppe
Published in Cells (Basel, Switzerland) (01.09.2020)
Published in Cells (Basel, Switzerland) (01.09.2020)
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An unexpected reversal in the pharmacological stereoselectivity of benzothiadiazine AMPA positive allosteric modulatorsThe authors declare no competing interests.We dedicate this work to Professor Carlo Parenti on the occasion of his retirement, who, with his great experience and dedication to organic synthesis, has given important contributions to scientific research
Battisti, Umberto M, Citti, Cinzia, Rastelli, Giulio, Pinzi, Luca, Puja, Giulia, Ravazzini, Federica, Ciccarella, Giuseppe, Braghiroli, Daniela, Cannazza, Giuseppe
Year of Publication 07.12.2016
Year of Publication 07.12.2016
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7‑Chloro-5-(furan-3-yl)-3-methyl‑4H‑benzo[e][1,2,4]thiadiazine 1,1-Dioxide as Positive Allosteric Modulator of α‑Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Receptor. The End of the Unsaturated-Inactive Paradigm?
Citti, Cinzia, Battisti, Umberto M, Cannazza, Giuseppe, Jozwiak, Krzysztof, Stasiak, Natalia, Puja, Giulia, Ravazzini, Federica, Ciccarella, Giuseppe, Braghiroli, Daniela, Parenti, Carlo, Troisi, Luigino, Zoli, Michele
Published in ACS chemical neuroscience (17.02.2016)
Published in ACS chemical neuroscience (17.02.2016)
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Journal Article
An unexpected reversal in the pharmacological stereoselectivity of benzothiadiazine AMPA positive allosteric modulators
Battisti, Umberto M., Citti, Cinzia, Rastelli, Giulio, Pinzi, Luca, Puja, Giulia, Ravazzini, Federica, Ciccarella, Giuseppe, Braghiroli, Daniela, Cannazza, Giuseppe
Published in MedChemComm (01.01.2016)
Published in MedChemComm (01.01.2016)
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7-Chloro-5-(furan-3-yl)-3-methyl-4 H -benzo[ e ][1,2,4]thiadiazine 1,1-Dioxide as Positive Allosteric Modulator of α-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Receptor. The End of the Unsaturated-Inactive Paradigm?
Citti, Cinzia, Battisti, Umberto M., Cannazza, Giuseppe, Jozwiak, Krzysztof, Stasiak, Natalia, Puja, Giulia, Ravazzini, Federica, Ciccarella, Giuseppe, Braghiroli, Daniela, Parenti, Carlo, Troisi, Luigino, Zoli, Michele
Published in ACS chemical neuroscience (17.02.2016)
Published in ACS chemical neuroscience (17.02.2016)
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Derivatives of 1,2,4-benzothiadiazine dioxide, their preparation and use as allosteric modulators of the AMPA receptor
BATTISTI, UMBERTO, CANNAZZA, GIUSEPPE, PARENTI, CARLO, CARROZZO, MARINA MARIA, BRAGHIROLI, DANIELA, JOZWIAK, KRZYSZTOF, PUJA, GIULIA, TROISI, LUIGINO
Year of Publication 30.05.2012
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Year of Publication 30.05.2012
Patent
DERIVATI DI 1,2,4-BENZOTIADIAZIN 1,1-DIOSSIDO, LORO PREPARAZIONE E LORO IMPIEGO COME MODULATORI ALLOSTERICI DEL RECETTORE AMPA
CANNAZZA GIUSEPPE, BRAGHIROLI DANIELA, JOZWIAK KRZYSZTOF, CARROZZO MARINA MARIA, PUJA GIULIA, BATTISTI UMBERTO, PARENTI CARLO, TROISI LUIGINO
Year of Publication 27.09.2013
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Year of Publication 27.09.2013
Patent
DERIVATI DI 1,2,4-BENZOTIADIAZIN 1,1-DIOSSIDO, LORO PREPARAZIONE E LORO IMPIEGO COME MODULATORI ALLOSTERICI DEL RECETTORE AMPA
CANNAZZA GIUSEPPE, BRAGHIROLI DANIELA, JOZWIAK KRZYSZTOF, CARROZZO MARINA MARIA, PUJA GIULIA, BATTISTI UMBERTO, PARENTI CARLO, TROISI LUIGINO
Year of Publication 30.05.2012
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Year of Publication 30.05.2012
Patent