Comparison of the cancer gene targeting and biochemical selectivities of all targeted kinase inhibitors approved for clinical use
Uitdehaag, Joost C M, de Roos, Jeroen A D M, van Doornmalen, Antoon M, Prinsen, Martine B W, de Man, Jos, Tanizawa, Yoshinori, Kawase, Yusuke, Yoshino, Kohichiro, Buijsman, Rogier C, Zaman, Guido J R
Published in PloS one (20.03.2014)
Published in PloS one (20.03.2014)
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Selective Targeting of CTNBB1-, KRAS- or MYC-Driven Cell Growth by Combinations of Existing Drugs
Uitdehaag, Joost C M, de Roos, Jeroen A D M, van Doornmalen, Antoon M, Prinsen, Martine B W, Spijkers-Hagelstein, Jill A P, de Vetter, Judith R F, de Man, Jos, Buijsman, Rogier C, Zaman, Guido J R
Published in PloS one (27.05.2015)
Published in PloS one (27.05.2015)
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Rb and FZR1/Cdh1 determine CDK4/6-cyclin D requirement in C. elegans and human cancer cells
The, Inge, Ruijtenberg, Suzan, Bouchet, Benjamin P, Cristobal, Alba, Prinsen, Martine B W, van Mourik, Tim, Koreth, John, Xu, Huihong, Heck, Albert J R, Akhmanova, Anna, Cuppen, Edwin, Boxem, Mike, Muñoz, Javier, van den Heuvel, Sander
Published in Nature communications (06.01.2015)
Published in Nature communications (06.01.2015)
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TTK Inhibitors as a Targeted Therapy for CTNNB1 ( β -catenin) Mutant Cancers
Zaman, Guido J R, de Roos, Jeroen A D M, Libouban, Marion A A, Prinsen, Martine B W, de Man, Jos, Buijsman, Rogier C, Uitdehaag, Joost C M
Published in Molecular cancer therapeutics (01.11.2017)
Published in Molecular cancer therapeutics (01.11.2017)
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Targeting Indoleamine 2,3-Dioxygenase in Cancer Models Using the Novel Small Molecule Inhibitor NTRC 3883-0
Grobben, Yvonne, de Man, Jos, van Doornmalen, Antoon M, Muller, Michelle, Willemsen-Seegers, Nicole, Vu-Pham, Diep, Mulder, Winfried R, Prinsen, Martine B W, de Wit, Joeri, Sterrenburg, Jan Gerard, van Cauter, Freek, den Ouden, Judith E, van Altena, Anne M, Massuger, Leon F, Uitdehaag, Joost C M, Buijsman, Rogier C, Zaman, Guido J R
Published in Frontiers in immunology (28.01.2021)
Published in Frontiers in immunology (28.01.2021)
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Comparative kinase and cancer cell panel profiling of kinase inhibitors approved for clinical use from 2018 to 2020
Kooijman, Jeffrey J., van Riel, Wilhelmina E., Dylus, Jelle, Prinsen, Martine B. W., Grobben, Yvonne, de Bitter, Tessa J. J., van Doornmalen, Antoon M., Melis, Janneke J. T. M., Uitdehaag, Joost C. M., Narumi, Yugo, Kawase, Yusuke, de Roos, Jeroen A. D. M., Willemsen-Seegers, Nicole, Zaman, Guido J. R.
Published in Frontiers in oncology (14.09.2022)
Published in Frontiers in oncology (14.09.2022)
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Caenorhabditis elegans cyclin D/CDK4 and cyclin E/CDK2 induce distinct cell cycle re-entry programs in differentiated muscle cells
Korzelius, Jerome, The, Inge, Ruijtenberg, Suzan, Prinsen, Martine B W, Portegijs, Vincent, Middelkoop, Teije C, Groot Koerkamp, Marian J, Holstege, Frank C P, Boxem, Mike, van den Heuvel, Sander
Published in PLoS genetics (01.11.2011)
Published in PLoS genetics (01.11.2011)
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Compound Selectivity and Target Residence Time of Kinase Inhibitors Studied with Surface Plasmon Resonance
Willemsen-Seegers, Nicole, Uitdehaag, Joost C.M., Prinsen, Martine B.W., de Vetter, Judith R.F., de Man, Jos, Sawa, Masaaki, Kawase, Yusuke, Buijsman, Rogier C., Zaman, Guido J.R.
Published in Journal of molecular biology (17.02.2017)
Published in Journal of molecular biology (17.02.2017)
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Target Residence Time-Guided Optimization on TTK Kinase Results in Inhibitors with Potent Anti-Proliferative Activity
Uitdehaag, Joost C.M., de Man, Jos, Willemsen-Seegers, Nicole, Prinsen, Martine B.W., Libouban, Marion A.A., Sterrenburg, Jan Gerard, de Wit, Joeri J.P., de Vetter, Judith R.F., de Roos, Jeroen A.D.M., Buijsman, Rogier C., Zaman, Guido J.R.
Published in Journal of molecular biology (07.07.2017)
Published in Journal of molecular biology (07.07.2017)
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Combined Cellular and Biochemical Profiling to Identify Predictive Drug Response Biomarkers for Kinase Inhibitors Approved for Clinical Use between 2013 and 2017
Uitdehaag, Joost C M, Kooijman, Jeffrey J, de Roos, Jeroen A D M, Prinsen, Martine B W, Dylus, Jelle, Willemsen-Seegers, Nicole, Kawase, Yusuke, Sawa, Masaaki, de Man, Jos, van Gerwen, Suzanne J C, Buijsman, Rogier C, Zaman, Guido J R
Published in Molecular cancer therapeutics (01.02.2019)
Published in Molecular cancer therapeutics (01.02.2019)
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Cell Panel Profiling Reveals Conserved Therapeutic Clusters and Differentiates the Mechanism of Action of Different PI3K/mTOR, Aurora Kinase and EZH2 Inhibitors
Uitdehaag, Joost C M, de Roos, Jeroen A D M, Prinsen, Martine B W, Willemsen-Seegers, Nicole, de Vetter, Judith R F, Dylus, Jelle, van Doornmalen, Antoon M, Kooijman, Jeffrey, Sawa, Masaaki, van Gerwen, Suzanne J C, de Man, Jos, Buijsman, Rogier C, Zaman, Guido J R
Published in Molecular cancer therapeutics (01.12.2016)
Published in Molecular cancer therapeutics (01.12.2016)
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Journal Article
Selective Targeting of CTNNB1-, KRAS- or MYC-Driven Cell Growth by Combinations of Existing Drugs
Uitdehaag, Joost C. M., de Roos, Jeroen A. D. M., van Doornmalen, Antoon M., Prinsen, Martine B. W., Spijkers-Hagelstein, Jill A. P., de Vetter, Judith R. F., de Man, Jos, Buijsman, Rogier C., Zaman, Guido J. R.
Published in PloS one (01.05.2015)
Published in PloS one (01.05.2015)
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Abstract 2646: The unique binding mode of NTRC 0066-0, a novel inhibitor of the spindle assembly checkpoint kinase TTK (Mps1), leads to long target residence time and potent antitumor activity
de Man, Jos, Uitdehaag, Joost C.M., Willemsen-Seegers, Nicole, Sterrenburg, Jan Gerard, de Wit, Joeri J.P., de Roos, Jeroen A.D.M., Prinsen, Martine B.W., Buijsman, Rogier C., Zaman, Guido J.R.
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Published in Cancer research (Chicago, Ill.) (15.07.2016)
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Caenorhabditis elegans Cyclin D/CDK4 and Cyclin E/CDK2 Induce Distinct Cell Cycle Re-Entry Programs in Differentiated Muscle Cells: e1002362
Korzelius, Jerome, The, Inge, Ruijtenberg, Suzan, Prinsen, Martine BW, Portegijs, Vincent, Middelkoop, Teije C, Koerkamp, Marian JGroot, Holstege, Frank CP, Boxem, Mike, Heuvel, Sander vanden
Published in PLoS genetics (01.11.2011)
Published in PLoS genetics (01.11.2011)
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Comparison of the Cancer Gene Targeting and Biochemical Selectivities of All Targeted Kinase Inhibitors Approved for Clinical Use: e92146
Uitdehaag, Joost CM, de Roos, D M, van Doornmalen, Antoon M, Prinsen, Martine BW, de Man, Jos, Tanizawa, Yoshinori, Kawase, Yusuke, Yoshino, Kohichiro, Buijsman, Rogier C, Zaman, Guido JR
Published in PloS one (01.03.2014)
Published in PloS one (01.03.2014)
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