Search Results - "Primofiore, G" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

[1,2,4]Triazino[4,3-a]benzimidazole Acetic Acid Derivatives: A New Class of Selective Aldose Reductase Inhibitors

[1,2,4]Triazino[4,3-a]benzimidazole Acetic Acid Derivatives: A New Class of Selective Aldose Reductase Inhibitors

by Da Settimo, Federico, Primofiore, Giampaolo, Da Settimo, Antonio, La Motta, Concettina, Taliani, Sabrina, Simorini, Francesca, Novellino, Ettore, Greco, Giovanni, Lavecchia, Antonio, Boldrini, Enrico
Published in Journal of medicinal chemistry (06.12.2001)

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3-Aryl[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-ones: A New Class of Selective A1 Adenosine Receptor Antagonists

3-Aryl[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-ones: A New Class of Selective A1 Adenosine Receptor Antagonists

by Da Settimo, Federico, Primofiore, Giampaolo, Taliani, Sabrina, Marini, Anna Maria, La Motta, Concettina, Novellino, Ettore, Greco, Giovanni, Lavecchia, Antonio, Trincavelli, Letizia, Martini, Claudia
Published in Journal of medicinal chemistry (01.02.2001)

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Novel N-(Arylalkyl)indol-3-ylglyoxylylamides Targeted as Ligands of the Benzodiazepine Receptor: Synthesis, Biological Evaluation, and Molecular Modeling Analysis of the Structure−Activity Relationships

Novel N-(Arylalkyl)indol-3-ylglyoxylylamides Targeted as Ligands of the Benzodiazepine Receptor: Synthesis, Biological Evaluation, and Molecular Modeling Analysis of the Structure−Activity Relationships

by Primofiore, Giampaolo, Settimo, Federico Da, Taliani, Sabrina, Marini, Anna Maria, Novellino, Ettore, Greco, Giovanni, Lavecchia, Antonio, Besnard, François, Trincavelli, Letizia, Costa, Barbara, Martini, Claudia
Published in Journal of medicinal chemistry (05.07.2001)

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Synthesis and antiproliferative evaluation of new aryl substituted pyrido[3 ',2 ': 5,6]thiopyrano[4,3-c]pyrazoles

Synthesis and antiproliferative evaluation of new aryl substituted pyrido[3 ',2 ': 5,6]thiopyrano[4,3-c]pyrazoles

by Primofiore, G, Marini, AM, Salerno, S, Da Settimo, F, Bertini, D, Dalla Via, L
Published in Journal of heterocyclic chemistry (01.11.2005)

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Synthesis of pyrimido[1,2-alpha]benzimidazol-4(10H)-one derivatives and evaluation of their interactions with DNA

Synthesis of pyrimido[1,2-alpha]benzimidazol-4(10H)-one derivatives and evaluation of their interactions with DNA

by Da Settimo, A, Primofiore, G, Da Settimo, F, Marini, AM, Taliani, S, Salerno, S, Via, LD
Published in Journal of heterocyclic chemistry (01.11.2003)

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Synthesis of pyrrolo[3,4- c]pyridine derivatives possessing an acid group and their in vitro and in vivo evaluation as aldose reductase inhibitors

Synthesis of pyrrolo[3,4- c]pyridine derivatives possessing an acid group and their in vitro and in vivo evaluation as aldose reductase inhibitors

by Da Settimo, A, Primofiore, G, Da Settimo, F, Simorini, F, La Motta, C, Martinelli, A, Boldrini, E
Published in European journal of medicinal chemistry (1996)

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Facile synthesis of 3-substituted [1,2,4]triazino[3,4-f]purine-4,6,8-trione derivatives

Facile synthesis of 3-substituted [1,2,4]triazino[3,4-f]purine-4,6,8-trione derivatives

by Da Settimo, F, Marini, AM, Pardi, G, Primofiore, G, Salerno, S, Simorini, F
Published in Journal of heterocyclic chemistry (01.05.2001)

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Isosteric replacement of the indole nucleus by benzothiophene and benzofuran in a series of indolylglyoxylylamine derivatives with partial agonist activity at the benzodiazepine receptor

Isosteric replacement of the indole nucleus by benzothiophene and benzofuran in a series of indolylglyoxylylamine derivatives with partial agonist activity at the benzodiazepine receptor

by Da Settimo, F, Lucacchini, A, Marini, AM, Martini, C, Primofiore, G, Senatore, G, Taliani, S
Published in European journal of medicinal chemistry (1996)

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Indole derivatives as probes to study the benzodiazepine binding site in GABA receptor complex

Indole derivatives as probes to study the benzodiazepine binding site in GABA receptor complex

by Da Settimo, A, Primofiore, G, Da Settimo, F, Novellino, E, Greco, G, Martini, C, Senatore, G, Lucacehini, A
Published in Advances in experimental medicine and biology (1996)

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Benzisothiazole-1,1-dioxide alkanoic acid derivatives as inhibitors of rat lens aldose reductase

Benzisothiazole-1,1-dioxide alkanoic acid derivatives as inhibitors of rat lens aldose reductase

by Primofiore, G, Da Settimo, F, La Motta, C, Simorini, F, Minutolo, A, Boldrini, E
Published in Farmaco (Società chimica italiana : 1989) (01.10.1997)

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N,N-Dialkyl-2-phenylindol-3-ylglyoxylamides. A New Class of Potent and Selective Ligands at the Peripheral Benzodiazepine Receptor

N,N-Dialkyl-2-phenylindol-3-ylglyoxylamides. A New Class of Potent and Selective Ligands at the Peripheral Benzodiazepine Receptor

by Primofiore, Giampaolo, Da Settimo, Federico, Taliani, Sabrina, Simorini, Francesca, Patrizi, Maria Paola, Novellino, Ettore, Greco, Giovanni, Abignente, Enrico, Costa, Barbara, Chelli, Beatrice, Martini, Claudia
Published in Journal of medicinal chemistry (25.03.2004)

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SYNTHESIS AND EVALUATION OF AMINOADAMANTANE DERIVATIVES FOR IN-VITRO ANTI-HIV AND ANTITUMOR ACTIVITIES

SYNTHESIS AND EVALUATION OF AMINOADAMANTANE DERIVATIVES FOR IN-VITRO ANTI-HIV AND ANTITUMOR ACTIVITIES

by DASETTIMO, A, MARINI, AM, PRIMOFIORE, G, DASETTIMO, F
Published in Farmaco (Società chimica italiana : 1989) (01.05.1995)

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Novel, Highly Potent Adenosine Deaminase Inhibitors Containing the Pyrazolo[3,4-d]pyrimidine Ring System. Synthesis, Structure−Activity Relationships, and Molecular Modeling Studies

Novel, Highly Potent Adenosine Deaminase Inhibitors Containing the Pyrazolo[3,4-d]pyrimidine Ring System. Synthesis, Structure−Activity Relationships, and Molecular Modeling Studies

by Da Settimo, Federico, Primofiore, Giampaolo, La Motta, Concettina, Taliani, Sabrina, Simorini, Francesca, Marini, Anna Maria, Mugnaini, Laura, Lavecchia, Antonio, Novellino, Ettore, Tuscano, Daniela, Martini, Claudia
Published in Journal of medicinal chemistry (11.08.2005)

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2-(Benzimidazol-2-yl)quinoxalines: A novel class of selective antagonists at human A(1) and A(3) adenosine receptors designed by 3D database searching

2-(Benzimidazol-2-yl)quinoxalines: A novel class of selective antagonists at human A(1) and A(3) adenosine receptors designed by 3D database searching

by Novellino, E, Cosimelli, B, Ehlardo, M, Greco, G, Iadanza, M, Lavecchia, A, Rimoli, MG, Sala, A, Da Settimo, A, Primofiore, G, Da Settimo, F, Taliani, S, La Motta, C, Klotz, KN, Tuscano, D, Trincavelli, ML, Martini, C
Published in Journal of medicinal chemistry (29.12.2005)

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Naphtho[1,2-d]isothiazole Acetic Acid Derivatives as a Novel Class of Selective Aldose Reductase Inhibitors

Naphtho[1,2-d]isothiazole Acetic Acid Derivatives as a Novel Class of Selective Aldose Reductase Inhibitors

by Da Settimo, Federico, Primofiore, Giampaolo, La Motta, Concettina, Sartini, Stefania, Taliani, Sabrina, Simorini, Francesca, Marini, Anna Maria, Lavecchia, Antonio, Novellino, Ettore, Boldrini, Enrico
Published in Journal of medicinal chemistry (03.11.2005)

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Synthesis and benzodiazepine receptor activity of some 4,5-dihydro-1H-pyrazolo[4,3-c][1,8]naphthyridine derivatives

Synthesis and benzodiazepine receptor activity of some 4,5-dihydro-1H-pyrazolo[4,3-c][1,8]naphthyridine derivatives

by Da Settimo, A, Primofiore, G, Da Settimo, F, Simorini, F, Barili, P L, Senatore, G, Martini, C, Lucacchini, A
Published in Drug design and discovery (01.06.1994)

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Acid derivatives of benzisothiazole-1,1-dioxide as inhibitors of rat lens aldose reductase

Acid derivatives of benzisothiazole-1,1-dioxide as inhibitors of rat lens aldose reductase

by DaSettimo, A, Primofiore, G, LaMotta, C, DaSettimo, F, Simorini, F, Boldrini, E, Bianchini, P
Published in Farmaco (Società chimica italiana : 1989) (01.04.1996)

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Spirohydantoin derivatives of thiopyrano[2,3- b]pyridin-4(4 H)-one as potent in vitro and in vivo aldose reductase inhibitors

Spirohydantoin derivatives of thiopyrano[2,3- b]pyridin-4(4 H)-one as potent in vitro and in vivo aldose reductase inhibitors

by Da Settimo, Federico, Primofiore, Giampaolo, La Motta, Concettina, Salerno, Silvia, Novellino, Ettore, Greco, Giovanni, Lavecchia, Antonio, Laneri, Sonia, Boldrini, Enrico
Published in Bioorganic & medicinal chemistry (17.01.2005)

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Isosteric replacement of amide by ester function. Synthesis and benzodiazepine receptor affinity of indol-3-ylglyoxylyl ester derivatives

Isosteric replacement of amide by ester function. Synthesis and benzodiazepine receptor affinity of indol-3-ylglyoxylyl ester derivatives

by DaSettimo, A, Primofiore, G, Marini, AM, DaSettimo, F, Nuti, Martini, C, Trincavelli, L, Lucacchini, A
Published in Farmaco (Società chimica italiana : 1989) (01.06.1997)

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3-aryl[1,2,4]triazino[4,3-alpha]benzimidazol-4(10H)-ones: A new class of selective A(1) adenosine receptor antagonists

3-aryl[1,2,4]triazino[4,3-alpha]benzimidazol-4(10H)-ones: A new class of selective A(1) adenosine receptor antagonists

by Da Settimo, F, Primofiore, G, Taliani, S, Marini, AM, La Motta, C, Novellino, E, Greco, G, Lavecchia, A, Trincavelli, L, Martini, C
Published in Journal of medicinal chemistry (01.02.2001)

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