Allosteric Small Molecules Unveil a Role of an Extracellular E2/Transmembrane Helix 7 Junction for G Protein-coupled Receptor Activation
Jäger, Dorothea, Schmalenbach, Caroline, Prilla, Stefanie, Schrobang, Jasmin, Kebig, Anna, Sennwitz, Matthias, Heller, Eberhard, Tränkle, Christian, Holzgrabe, Ulrike, Höltje, Hans-Dieter, Mohr, Klaus
Published in The Journal of biological chemistry (30.11.2007)
Published in The Journal of biological chemistry (30.11.2007)
Get full text
Journal Article
Critical Amino Acid Residues of the Common Allosteric Site on the M2 Muscarinic Acetylcholine Receptor: More Similarities than Differences between the Structurally Divergent Agents Gallamine and Bis(ammonio)alkane-Type Hexamethylene-bis-[dimethyl-(3-phthalimidopropyl)ammonium]dibromide
Huang, Xi-Ping, Prilla, Stefanie, Mohr, Klaus, Ellis, John
Published in Molecular pharmacology (01.09.2005)
Published in Molecular pharmacology (01.09.2005)
Get full text
Journal Article
Allosteric Interactions with Muscarinic Acetylcholine Receptors: Complex Role of the Conserved Tryptophan M2422Trp in a Critical Cluster of Amino Acids for Baseline Affinity, Subtype Selectivity, and Cooperativity
Prilla, Stefanie, Schrobang, Jasmin, Ellis, John, Höltje, Hans-Dieter, Mohr, Klaus
Published in Molecular pharmacology (01.07.2006)
Published in Molecular pharmacology (01.07.2006)
Get full text
Journal Article
European Medicines Agency review of post-authorisation studies with implications for the European Network of Centres for Pharmacoepidemiology and Pharmacovigilance
Blake, Kevin V., Prilla, Stefanie, Accadebled, Sophie, Guimier, Marie, Biscaro, Monica, Persson, Ingemar, Arlett, Peter, Blackburn, Stella, Fitt, Henry
Published in Pharmacoepidemiology and drug safety (01.10.2011)
Published in Pharmacoepidemiology and drug safety (01.10.2011)
Get full text
Journal Article
Critical Amino Acid Residues of the Common Allosteric Site on the M 2 Muscarinic Acetylcholine Receptor: More Similarities than Differences between the Structurally Divergent Agents Gallamine and Bis(ammonio)alkane-Type Hexamethylene- bis -[dimethyl-(3-phthalimidopropyl)ammonium]dibromide
Huang, Xi-Ping, Prilla, Stefanie, Mohr, Klaus, Ellis, John
Published in Molecular pharmacology (01.09.2005)
Published in Molecular pharmacology (01.09.2005)
Get full text
Journal Article
Critical Amino Acid Residues of the Common Allosteric Site on the M sub(2) Muscarinic Acetylcholine Receptor: More Similarities than Differences between the Structurally Divergent Agents Gallamine and Bis(ammonio)alkane-Type Hexamethylene-bis-[dimethyl-(3-phthalimidopropyl)ammonium]dibromid e
Huang, Xi-Ping, Prilla, Stefanie, Mohr, Klaus, Ellis, John
Published in Molecular pharmacology (01.09.2005)
Get full text
Published in Molecular pharmacology (01.09.2005)
Journal Article
Allosteric Interactions with Muscarinic Acetylcholine Receptors: Complex Role of the Conserved Tryptophan M 2 422 Trp in a Critical Cluster of Amino Acids for Baseline Affinity, Subtype Selectivity, and Cooperativity
Prilla, Stefanie, Schrobang, Jasmin, Ellis, John, Höltje, Hans-Dieter, Mohr, Klaus
Published in Molecular pharmacology (01.07.2006)
Published in Molecular pharmacology (01.07.2006)
Get full text
Journal Article