Glucose 6-phosphate dehydrogenase 6-phosphogluconolactonase: characterization of the Plasmodium vivax enzyme and inhibitor studies
Haeussler, Kristina, Berneburg, Isabell, Jortzik, Esther, Hahn, Julia, Rahbari, Mahsa, Schulz, Norma, Preuss, Janina, Zapol'skii, Viktor A, Bode, Lars, Pinkerton, Anthony B, Kaufmann, Dieter E, Rahlfs, Stefan, Becker, Katja
Published in Malaria journal (25.01.2019)
Published in Malaria journal (25.01.2019)
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An Optimized Dihydrodibenzothiazepine Lead Compound (SBI-0797750) as a Potent and Selective Inhibitor of Plasmodium falciparum and P. vivax Glucose 6-Phosphate Dehydrogenase 6-Phosphogluconolactonase
Berneburg, Isabell, Peddibhotla, Satyamaheshwar, Heimsch, Kim C, Haeussler, Kristina, Maloney, Patrick, Gosalia, Palak, Preuss, Janina, Rahbari, Mahsa, Skorokhod, Oleksii, Valente, Elena, Ulliers, Daniela, Simula, Luigi Felice, Buchholz, Kathrin, Hedrick, Michael P, Hershberger, Paul, Chung, Thomas D Y, Jackson, Michael R, Schwarzer, Evelin, Rahlfs, Stefan, Bode, Lars, Becker, Katja, Pinkerton, Anthony B
Published in Antimicrobial agents and chemotherapy (19.04.2022)
Published in Antimicrobial agents and chemotherapy (19.04.2022)
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Identification and characterization of novel human glucose-6-phosphate dehydrogenase inhibitors
Preuss, Janina, Richardson, Adam D, Pinkerton, Anthony, Hedrick, Michael, Sergienko, Eduard, Rahlfs, Stefan, Becker, Katja, Bode, Lars
Published in Journal of biomolecular screening (01.03.2013)
Published in Journal of biomolecular screening (01.03.2013)
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Glucose-6-phosphate dehydrogenase-6-phosphogluconolactonase: a unique bifunctional enzyme from Plasmodium falciparum
Jortzik, Esther, Mailu, Boniface M, Preuss, Janina, Fischer, Marina, Bode, Lars, Rahlfs, Stefan, Becker, Katja
Published in Biochemical journal (15.06.2011)
Published in Biochemical journal (15.06.2011)
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Plasmodium falciparum glucose‐6‐phosphate dehydrogenase 6‐phosphogluconolactonase is a potential drug target
Allen, Stacey M, Lim, Erin E, Jortzik, Esther, Preuss, Janina, Chua, Hwa Huat, MacRae, James I, Rahlfs, Stefan, Haeussler, Kristina, Downton, Matthew T, McConville, Malcolm J, Becker, Katja, Ralph, Stuart A
Published in The FEBS journal (01.10.2015)
Published in The FEBS journal (01.10.2015)
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High-throughput screening for small-molecule inhibitors of plasmodium falciparum glucose-6-phosphate dehydrogenase 6-phosphogluconolactonase
Preuss, Janina, Hedrick, Michael, Sergienko, Eduard, Pinkerton, Anthony, Mangravita-Novo, Arianna, Smith, Layton, Marx, Carolin, Fischer, Elisabeth, Jortzik, Esther, Rahlfs, Stefan, Becker, Katja, Bode, Lars
Published in Journal of biomolecular screening (01.07.2012)
Published in Journal of biomolecular screening (01.07.2012)
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Discovery of a Plasmodium falciparum Glucose-6-phosphate Dehydrogenase 6‑phosphogluconolactonase Inhibitor (R,Z)‑N‑((1-Ethylpyrrolidin-2-yl)methyl)-2-(2-fluorobenzylidene)-3-oxo-3,4-dihydro‑2H‑benzo[b][1,4]thiazine-6-carboxamide (ML276) That Reduces Parasite Growth in Vitro
Preuss, Janina, Maloney, Patrick, Peddibhotla, Satyamaheshwar, Hedrick, Michael P, Hershberger, Paul, Gosalia, Palak, Milewski, Monika, Li, Yujie Linda, Sugarman, Eliot, Hood, Becky, Suyama, Eigo, Nguyen, Kevin, Vasile, Stefan, Sergienko, Eduard, Mangravita-Novo, Arianna, Vicchiarelli, Michael, McAnally, Danielle, Smith, Layton H, Roth, Gregory P, Diwan, Jena, Chung, Thomas D.Y, Jortzik, Esther, Rahlfs, Stefan, Becker, Katja, Pinkerton, Anthony B, Bode, Lars
Published in Journal of medicinal chemistry (23.08.2012)
Published in Journal of medicinal chemistry (23.08.2012)
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Characterization of tryptophan aminotransferase 1 of Malassezia furfur, the key enzyme in the production of indolic compounds by M. furfur
Preuss, Janina, Hort, Wiebke, Lang, Sarah, Netsch, Anette, Rahlfs, Stefan, Lochnit, Günter, Jortzik, Esther, Becker, Katja, Mayser, Peter A.
Published in Experimental dermatology (01.11.2013)
Published in Experimental dermatology (01.11.2013)
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Characterization of tryptophan aminotransferase 1 of M alassezia furfur , the key enzyme in the production of indolic compounds by M. furfur
Preuss, Janina, Hort, Wiebke, Lang, Sarah, Netsch, Anette, Rahlfs, Stefan, Lochnit, Günter, Jortzik, Esther, Becker, Katja, Mayser, Peter A.
Published in Experimental dermatology (01.11.2013)
Published in Experimental dermatology (01.11.2013)
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Discovery of a Plasmodium falciparum Glucose-6-phosphate Dehydrogenase 6-phosphogluconolactonase Inhibitor ( R , Z )- N -((1-Ethylpyrrolidin-2-yl)methyl)-2-(2-fluorobenzylidene)-3-oxo-3,4-dihydro-2 H -benzo[ b ][1,4]thiazine-6-carboxamide (ML276) That Reduces Parasite Growth in Vitro
Preuss, Janina, Maloney, Patrick, Peddibhotla, Satyamaheshwar, Hedrick, Michael P., Hershberger, Paul, Gosalia, Palak, Milewski, Monika, Li, Yujie Linda, Sugarman, Eliot, Hood, Becky, Suyama, Eigo, Nguyen, Kevin, Vasile, Stefan, Sergienko, Eduard, Mangravita-Novo, Arianna, Vicchiarelli, Michael, McAnally, Danielle, Smith, Layton H., Roth, Gregory P., Diwan, Jena, Chung, Thomas D.Y., Jortzik, Esther, Rahlfs, Stefan, Becker, Katja, Pinkerton, Anthony B., Bode, Lars
Published in Journal of medicinal chemistry (23.08.2012)
Published in Journal of medicinal chemistry (23.08.2012)
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