Bicyclic heteroarylpiperazines as selective brain penetrant 5-HT 6 receptor antagonists
Ahmed, Mahmood, Briggs, Michael A., Bromidge, Steven M., Buck, Tania, Campbell, Lorraine, Deeks, Nigel J., Garner, Ashley, Gordon, Laurie, Hamprecht, Dieter W., Holland, Vicky, Johnson, Christopher N., Medhurst, Andrew D., Mitchell, Darren J., Moss, Stephen F., Powles, Jenifer, Seal, Jon T., Stean, Tania O., Stemp, Geoffrey, Thompson, Mervyn, Trail, Brenda, Upton, Neil, Winborn, Kim, Witty, David R.
Published in Bioorganic & medicinal chemistry letters (01.11.2005)
Published in Bioorganic & medicinal chemistry letters (01.11.2005)
Get full text
Journal Article
Structure-guided design of pyrazolo[1,5- a]pyrimidines as inhibitors of human cyclin-dependent kinase 2
Williamson, Douglas S., Parratt, Martin J., Bower, Justin F., Moore, Jonathan D., Richardson, Christine M., Dokurno, Pawel, Cansfield, Andrew D., Francis, Geraint L., Hebdon, Richard J., Howes, Rob, Jackson, Philip S., Lockie, Andrea M., Murray, James B., Nunns, Claire L., Powles, Jenifer, Robertson, Alan, Surgenor, Allan E., Torrance, Christopher J.
Published in Bioorganic & medicinal chemistry letters (15.02.2005)
Published in Bioorganic & medicinal chemistry letters (15.02.2005)
Get full text
Journal Article
Bicyclic heteroarylpiperazines as selective brain penetrant 5-HT6 receptor antagonists
AHMED, Mahmood, BRIGGS, Michael A, JOHNSON, Christopher N, MEDHURST, Andrew D, MITCHELL, Darren J, MOSS, Stephen F, POWLES, Jenifer, SEAL, Jon T, STEAN, Tania O, STEMP, Geoffrey, THOMPSON, Mervyn, TRAIL, Brenda, BROMIDGE, Steven M, UPTON, Neil, WINBORN, Kim, WITTY, David R, BUCK, Tania, CAMPBELL, Lorraine, DEEKS, Nigel J, GARNER, Ashley, GORDON, Laurie, HAMPRECHT, Dieter W, HOLLAND, Vicky
Published in Bioorganic & medicinal chemistry letters (01.11.2005)
Published in Bioorganic & medicinal chemistry letters (01.11.2005)
Get full text
Journal Article
Structure-based design of agents targeting the bacterial ribosome
Bower, Justin, Drysdale, Martin, Hebdon, Richard, Jordan, Allan, Lentzen, Georg, Matassova, Natalia, Murchie, Alastair, Powles, Jenifer, Roughley, Stephen
Published in Bioorganic & medicinal chemistry letters (04.08.2003)
Published in Bioorganic & medicinal chemistry letters (04.08.2003)
Get full text
Journal Article
8-piperazinyl-2,3-dihydropyrrolo[3,2-g]isoquinolines : Potent, selective, orally bioavailable 5-HT1 receptor ligands
HEIGHTMAN, Tom D, GASTER, Laramie M, GORDON, Laurie J, HOLLAND, Vicky A, POWLES, Jenifer, RILEY, Graham J, STEAN, Tania O, TRAIL, Brenda K, UPTON, Neil, AUSTIN, Nigel E, AYRTON, Andrew D, COLEMAN, Tanya, PARDOE, Sarah L, CUTLER, Leanne, PILLEUX, Jean-Pierre, HADLEY, Michael S, MIDDLEMISS, Derek N, PRICE, Gary W, ROBERTS, Claire, SCOTT, Claire M, WATSON, Jeannette M
Published in Bioorganic & medicinal chemistry letters (01.10.2005)
Published in Bioorganic & medicinal chemistry letters (01.10.2005)
Get full text
Journal Article
WITHDRAWN: Bicyclic heteroarylpiperazines as selective brain penetrant 5-HT6 receptor antagonists
Ahmed, Mahmood, Briggs, Michael A., Bromidge, Steven M., Buck, Tania, Campbell, Lorraine, Deeks, Nigel J., Garner, Ashley, Gordon, Laurie, Hamprecht, Dieter W., Holland, Vicky, Johnson, Christopher N., Medhurst, Andrew D., Mitchell, Darren J., Moss, Stephen F., Powles, Jenifer, Seal, Jon T., Stean, Tania O., Stemp, Geoffrey, Thompson, Mervyn, Trail, Brenda, Upton, Neil, Winborn, Kim, Witty, David R.
Published in Bioorganic & medicinal chemistry (01.07.2005)
Published in Bioorganic & medicinal chemistry (01.07.2005)
Get full text
Journal Article
8-Piperazinyl-2,3-dihydropyrrolo[3,2- g]isoquinolines: Potent, selective, orally bioavailable 5-HT 1 receptor ligands
Heightman, Tom D., Gaster, Laramie M., Pardoe, Sarah L., Pilleux, Jean-Pierre, Hadley, Michael S., Middlemiss, Derek N., Price, Gary W., Roberts, Claire, Scott, Claire M., Watson, Jeannette M., Gordon, Laurie J., Holland, Vicky A., Powles, Jenifer, Riley, Graham J., Stean, Tania O., Trail, Brenda K., Upton, Neil, Austin, Nigel E., Ayrton, Andrew D., Coleman, Tanya, Cutler, Leanne
Published in Bioorganic & medicinal chemistry letters (2005)
Published in Bioorganic & medicinal chemistry letters (2005)
Get full text
Journal Article
Structure-Based Design of Agents Targeting the Bacterial Ribosome
Bower, Justin, Drysdale, Martin, Hebdon, Richard, Jordan, Allan, Lentzen, Georg, Matassova, Natalia, Murchie, Alastair, Powles, Jenifer, Roughley, Stephen
Published in ChemInform (28.10.2003)
Published in ChemInform (28.10.2003)
Get full text
Journal Article