Total Synthesis and Configurational Assignment of (−)-Dictyostatin, a Microtubule-Stabilizing Macrolide of Marine Sponge Origin
Paterson, Ian, Britton, Robert, Delgado, Oscar, Meyer, Arndt, Poullennec, Karine G.
Published in Angewandte Chemie (International ed.) (06.09.2004)
Published in Angewandte Chemie (International ed.) (06.09.2004)
Get full text
Journal Article
Enantioselective Total Synthesis of (+)-Dibromophakellstatin
Poullennec, Karine G, Romo, Daniel
Published in Journal of the American Chemical Society (28.05.2003)
Published in Journal of the American Chemical Society (28.05.2003)
Get full text
Journal Article
Discovery of a Potent and Orally Bioavailable Cyclophilin Inhibitor Derived from the Sanglifehrin Macrocycle
Mackman, Richard L, Steadman, Victoria A, Dean, David K, Jansa, Petr, Poullennec, Karine G, Appleby, Todd, Austin, Carol, Blakemore, Caroline A, Cai, Ruby, Cannizzaro, Carina, Chin, Gregory, Chiva, Jean-Yves C, Dunbar, Neil A, Fliri, Hans, Highton, Adrian J, Hui, Hon, Ji, Mingzhe, Jin, Haolun, Karki, Kapil, Keats, Andrew J, Lazarides, Linos, Lee, Yu-Jen, Liclican, Albert, Mish, Michael, Murray, Bernard, Pettit, Simon B, Pyun, Peter, Sangi, Michael, Santos, Rex, Sanvoisin, Jonathan, Schmitz, Uli, Schrier, Adam, Siegel, Dustin, Sperandio, David, Stepan, George, Tian, Yang, Watt, Gregory M, Yang, Hai, Schultz, Brian E
Published in Journal of medicinal chemistry (08.11.2018)
Published in Journal of medicinal chemistry (08.11.2018)
Get full text
Journal Article
Discovery of Potent Cyclophilin Inhibitors Based on the Structural Simplification of Sanglifehrin A
Steadman, Victoria A, Pettit, Simon B, Poullennec, Karine G, Lazarides, Linos, Keats, Andrew J, Dean, David K, Stanway, Steven J, Austin, Carol A, Sanvoisin, Jonathan A, Watt, Gregory M, Fliri, Hans G, Liclican, Albert C, Jin, Debi, Wong, Melanie H, Leavitt, Stephanie A, Lee, Yu-Jen, Tian, Yang, Frey, Christian R, Appleby, Todd C, Schmitz, Uli, Jansa, Petr, Mackman, Richard L, Schultz, Brian E
Published in Journal of medicinal chemistry (09.02.2017)
Published in Journal of medicinal chemistry (09.02.2017)
Get full text
Journal Article
Synthesis and biological evaluation of novel analogues of dictyostatin
Paterson, Ian, Gardner, Nicola M., Poullennec, Karine G., Wright, Amy E.
Published in Bioorganic & medicinal chemistry letters (01.05.2007)
Published in Bioorganic & medicinal chemistry letters (01.05.2007)
Get full text
Journal Article
Synthesis and Biological Evaluation of 10,11-Dihydrodictyostatin, a Potent Analogue of the Marine Anticancer Agent Dictyostatin
Paterson, Ian, Gardner, Nicola M, Poullennec, Karine G, Wright, Amy E
Published in Journal of natural products (Washington, D.C.) (01.03.2008)
Published in Journal of natural products (Washington, D.C.) (01.03.2008)
Get full text
Journal Article
ASSESSMENT OF GAS COOLED FAST REACTOR WITH INDIRECT SUPERCRITICAL $CO_2$ CYCLE
Hejzlar, P, Dostal, V, Driscoll, M.J, Dumaz, P, Poullennec, G, Alpy, N
Published in Nuclear engineering and technology (2006)
Get full text
Published in Nuclear engineering and technology (2006)
Journal Article
Planned and unplanned halogenations in route to selected oroidin alkaloids
Wang, Shaohui, Dilley, Anja S., Poullennec, Karine G., Romo, Daniel
Published in Tetrahedron (24.07.2006)
Published in Tetrahedron (24.07.2006)
Get full text
Journal Article
Total synthesis of (-)-dictyostatin, a microtubule-stabilising anticancer macrolide of marine sponge origin: 2009 Tetrahedron Prize for Creativity in Organic Chemistry: Adventures in Organic Synthesis: Steven V. Ley
PATERSON, Ian, BRITTON, Robert, DELGADO, Oscar, GARDNER, Nicola M, MEYER, Arndt, NAYLOR, Guy J, POULLENNEC, Karine G
Published in Tetrahedron (2010)
Get full text
Published in Tetrahedron (2010)
Journal Article
Synthesis and Biological Evaluation of 10,11-Dihydrodictyostatin, a Potent Analogue of the Marine Anticancer Agent Dictyostatin super([section])
Gardner, Nicola M, Paterson, Ian, Wright, Amy E, Poullennec, Karine G
Published in Journal of natural products (Washington, D.C.) (01.01.2008)
Published in Journal of natural products (Washington, D.C.) (01.01.2008)
Get full text
Journal Article
MACROCYCLIC INHIBITORS OF FLAVIVIRIDAE VIRUSES
LINOS LAZARIDES, GREG WATT, RICHARD L. MACKMAN, KARINE G. POULLENNEC, DUSTIN SCOTT SIEGEL, VICTORIA ALEXANDRA STEADMAN, JEAN YVES CHIVA, ANDREW JOHN KEATS, PETR JANSA, CAROLINE ACIRO, ADRIAN JOHN HIGHTON, DAVID KENNETH DEAN, ADAM JAMES SCHRIER
Year of Publication 12.06.2018
Get full text
Year of Publication 12.06.2018
Patent
MACROCYCLIC INHIBITORS OF FLAVIVIRIDAE VIRUSES
KAPIL KUMAR KARKI, RICHARD MACKMAN, LINOS LAZARIDES, KARINE G. POULLENNEC, DUSTIN SCOTT SIEGEL, VICTORIA ALEXANDRA STEADMAN, SIMON NEIL PETTIT, NEIL ANDREW DUNBAR, ANDREW JOHN KEATS, PETR JANSA, CAROLINE ACIRO, DAVID KENNETH DEAN, ADRIAN JOHN HIGHTON, ADAM JAMES SCHRIER
Year of Publication 18.01.2018
Get full text
Year of Publication 18.01.2018
Patent
inibidores macrocíclicos do vírus flaviviridae
ANDREW J. KEATS, GREGORY M. WATT, JONATHAN SANVOISIN, LINOS LAZARIDES, HANS G. FLIRI, RICHARD L. MACKMAN, KARINE G. POULLENNEC, TODD APPLEBY, VICTORIA A. STEADMAN, SIMON N. PETTIT
Year of Publication 13.09.2016
Get full text
Year of Publication 13.09.2016
Patent
MACROCYCLIC INHIBITORS OF FLAVIVIRIDAE VIRUSES
KAPIL KUMAR KARKI, RICHARD MACKMAN, LINOS LAZARIDES, KARINE G. POULLENNEC, DUSTIN SCOTT SIEGEL, VICTORIA ALEXANDRA STEADMAN, JEAN YVES CHIVA, SIMON NEIL PETTIT, NEIL ANDREW DUNBAR, ANDREW JOHN KEATS, PETR JANSA, CAROLINE ACIRO, DAVID KENNETH DEAN, ADRIAN JOHN HIGHTON, ADAM JAMES SCHRIER
Year of Publication 05.05.2017
Get full text
Year of Publication 05.05.2017
Patent
MACROCYCLIC INHIBITORS OF FLAVIVIRIDAE VIRUSES
ANDREW J. KEATS, JONATHAN SANVOISIN, GREGORY M. WATT, LINOS LAZARIDES, HANS G. FLIRI, RICHARD L. MACKMAN, KARINE G. POULLENNEC, TODD APPLEBY, VICTORIA A. STEADMAN, SIMON N. PETTIT
Year of Publication 02.06.2015
Get full text
Year of Publication 02.06.2015
Patent
MACROCYCLIC INHIBITORS OF FLAVIVIRIDAE VIRUSES
Victoria Alexandra Steadman, David Kenneth Dean, Karine G. Poullennec, Petr Jansa, Adam James Schrier, Richard Mackman, Adrian John Highton, Dustin Scott Siegel, Caroline Aciro, Gregory Watt, Andrew John Keats, Linos Lazarides, Jean Yves Chiva
Year of Publication 27.01.2016
Get full text
Year of Publication 27.01.2016
Patent
MACROCYCLIC INHIBITORS OF FLAVIVIRIDAE VIRUSES
ANDREW J. KEATS, JONATHAN SANVOISIN, GREGORY M. WATT, LINOS LAZARIDES, HANS G. FLIRI, RICHARD L. MACKMAN, KARINE G. POULLENNEC, TODD APPLEBY, VICTORIA A. STEADMAN, SIMON N. PETTIT
Year of Publication 18.07.2014
Get full text
Year of Publication 18.07.2014
Patent
Cover Picture: Total Synthesis and Configurational Assignment of (−)-Dictyostatin, a Microtubule-Stabilizing Macrolide of Marine Sponge Origin / Total Synthesis of (−)-Dictyostatin: Confirmation of Relative and Absolute Configurations (Angew. Chem. Int. Ed. 35/2004)
Paterson, Ian, Britton, Robert, Delgado, Oscar, Meyer, Arndt, Poullennec, Karine G., Shin, Youseung, Fournier, Jean-Hugues, Fukui, Yoshikazu, Brückner, Arndt M., Curran, Dennis P.
Published in Angewandte Chemie (International ed.) (06.09.2004)
Published in Angewandte Chemie (International ed.) (06.09.2004)
Get full text
Journal Article