Development of an Efficient Pd-Catalyzed Coupling Process for Axitinib
Chekal, Brian P, Guinness, Steven M, Lillie, Brett M, McLaughlin, Robert W, Palmer, Charles W, Post, Ronald J, Sieser, Janice E, Singer, Robert A, Sluggett, Gregory W, Vaidyanathan, Rajappa, Withbroe, Gregory J
Published in Organic process research & development (17.01.2014)
Published in Organic process research & development (17.01.2014)
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The Evolution of High-Throughput Experimentation in Pharmaceutical Development and Perspectives on the Future
Mennen, Steven M, Alhambra, Carolina, Allen, C. Liana, Barberis, Mario, Berritt, Simon, Brandt, Thomas A, Campbell, Andrew D, Castañón, Jesús, Cherney, Alan H, Christensen, Melodie, Damon, David B, Eugenio de Diego, J, García-Cerrada, Susana, García-Losada, Pablo, Haro, Rubén, Janey, Jacob, Leitch, David C, Li, Ling, Liu, Fangfang, Lobben, Paul C, MacMillan, David W. C, Magano, Javier, McInturff, Emma, Monfette, Sebastien, Post, Ronald J, Schultz, Danielle, Sitter, Barbara J, Stevens, Jason M, Strambeanu, Iulia I, Twilton, Jack, Wang, Ke, Zajac, Matthew A
Published in Organic process research & development (21.06.2019)
Published in Organic process research & development (21.06.2019)
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Palbociclib Commercial Manufacturing Process Development. Part III. Deprotection Followed by Crystallization for API Particle Property Control
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Published in Organic process research & development (15.07.2016)
Published in Organic process research & development (15.07.2016)
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Chemoselective Saponification in the Synthesis of Danuglipron Facilitated with Trifluoroethanol
Han, Lu, Li, Bryan, Wang, Ke, Damon, David B., Magano, Javier, Maloney, Mark T., Mustakis, Jason, Post, Ronald J., Li, Ruizhi, Nguyen, Truong
Published in Organic process research & development (19.07.2024)
Published in Organic process research & development (19.07.2024)
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5-[(3-Nitropyrid-2-yl)amino]indoles: Novel Serotonin Agonists with Selectivity for the 5-HT1D Receptor. Variation of the C3 Substituent on the Indole Template Leads to Increased 5-HT1D Receptor Selectivity
Macor, John E, Blank, David H, Fox, Carol B, Lebel, Lorraine A, Newman, Michael E, Post, Ronald J, Ryan, Kevin, Schmidt, Anne W, Schulz, David W, Koe, B. Kenneth
Published in Journal of medicinal chemistry (01.08.1994)
Published in Journal of medicinal chemistry (01.08.1994)
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Journal Article
5-cyano-1-[3-(N-methylpyrrolidin-2R-ylmethyl)indol-5-yl] benzimidazole (CP-161,242): A potent, centrally active 5-HT1D receptor agonist and benzodiazepine partial agonist
Macor, John E, Blank, David H, Desai, Kishor, Fox, Carol B, Kenneth Koe, B, Lebel, Lorraine A, Post, Ronald J, Schmidt, Anne W, Schulz, David W, Seymour, Patricia A
Published in Bioorganic & medicinal chemistry letters (19.10.1995)
Published in Bioorganic & medicinal chemistry letters (19.10.1995)
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Journal Article
Synthesis and reactivity of pyrrolo[3,2-e]indole: Removal of a N-BOM group from an unactivated indole
Macor, John E., Forman, James T., Post, Ronald J., Ryan, Kevin
Published in Tetrahedron letters (10.03.1997)
Published in Tetrahedron letters (10.03.1997)
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Journal Article
The discovery of a novel and potent benzodiazepine receptor pharmacophore
Macor, John E., Blake, James F., Desai, Kishor, Post, Ronald J., Schmidt, Anne W.
Published in Bioorganic & medicinal chemistry letters (19.10.1995)
Published in Bioorganic & medicinal chemistry letters (19.10.1995)
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Journal Article
5-cyano-1-[3-(N-methylpyrrolidin-2R-ylmethyl)indol-5-yl] benzimidazole (CP-161,242): A potent, centrally active 5-HT 1D receptor agonist and benzodiazepine partial agonist
Macor, John E, Blank, David H, Desai, Kishor, Fox, Carol B, Kenneth Koe, B, Lebel, Lorraine A, Post, Ronald J, Schmidt, Anne W, Schulz, David W, Seymour, Patricia A
Published in Bioorganic & medicinal chemistry letters (1995)
Published in Bioorganic & medicinal chemistry letters (1995)
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Journal Article
Process for the preparation of pyrazolopyridine tartrates
BUSCH FRANK R.,CHIU CHARLES K.,MELTZ CLIFFORD N.,POST RONALD J.,ROSE PETER R
Year of Publication 27.09.2006
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Year of Publication 27.09.2006
Patent
Process for preparing growth hormone secretagogues
Busch, Frank R, Chiu, Charles K, Meltz, Clifford N, Post, Ronald J, Rose, Peter R
Year of Publication 06.01.2004
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Year of Publication 06.01.2004
Patent
Process for preparing growth hormone secretagogues
ROSE PETER R, CHIU CHARLES K, MELTZ CLIFFORD N, POST RONALD J, BUSCH FRANK R
Year of Publication 06.01.2004
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Year of Publication 06.01.2004
Patent
Process for preparing growth hormone secretagogues
ROSE PETER R, CHIU CHARLES K, MELTZ CLIFFORD N, POST RONALD J, BUSCH FRANK R
Year of Publication 21.08.2003
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Year of Publication 21.08.2003
Patent
Process for preparing growth hormone secretagogues
Busch, Frank R, Chiu, Charles K, Meltz, Clifford N, Post, Ronald J, Rose, Peter R
Year of Publication 01.04.2003
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Year of Publication 01.04.2003
Patent
Process for preparing growth hormone secretagogues
ROSE PETER R, CHIU CHARLES K, MELTZ CLIFFORD N, POST RONALD J, BUSCH FRANK R
Year of Publication 01.04.2003
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Year of Publication 01.04.2003
Patent