Discovery of Aminothiazole Inhibitors of Cyclin-Dependent Kinase 2: Synthesis, X-ray Crystallographic Analysis, and Biological Activities
Kim, Kyoung Soon, Kimball, S. David, Misra, Raj N, Rawlins, David B, Hunt, John T, Xiao, Hai-Yun, Lu, Songfeng, Qian, Ligang, Han, Wen-Ching, Shan, Weifang, Mitt, Toomas, Cai, Zhen-Wei, Poss, Michael A, Zhu, Hong, Sack, John S, Tokarski, John S, Chang, Chieh Ying, Pavletich, Nikola, Kamath, Amrita, Humphreys, William G, Marathe, Punit, Bursuker, Isia, Kellar, Kristen A, Roongta, Urvashi, Batorsky, Roberta, Mulheron, Janet G, Bol, David, Fairchild, Craig R, Lee, Francis Y, Webster, Kevin R
Published in Journal of medicinal chemistry (29.08.2002)
Published in Journal of medicinal chemistry (29.08.2002)
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Identification of chemokine receptor CCR4 antagonist
Purandare, Ashok V., Gao, Aiming, Wan, Honghe, Somerville, John, Burke, Christine, Seachord, Carrie, Vaccaro, Wayne, Wityak, John, Poss, Michael A.
Published in Bioorganic & medicinal chemistry letters (16.05.2005)
Published in Bioorganic & medicinal chemistry letters (16.05.2005)
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Identification of purine inhibitors of phosphodiesterase 7 (PDE7)
Pitts, William J., Vaccaro, Wayne, Huynh, Tram, Leftheris, Katerina, Roberge, Jacques Y., Barbosa, Joseph, Guo, Junqing, Brown, Baerbel, Watson, Andrew, Donaldson, Karen, Starling, Gary C., Kiener, Peter A., Poss, Michael A., Dodd, John H., Barrish, Joel C.
Published in Bioorganic & medicinal chemistry letters (07.06.2004)
Published in Bioorganic & medicinal chemistry letters (07.06.2004)
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Pyrrolopyridazine MEK inhibitors
Chen, Zhong, Kim, Soong-Hoon, Barbosa, Stephanie A., Huynh, Tram, Tortolani, David R., Leavitt, Kenneth J., Wei, Donna D., Manne, Veeraswamy, Ricca, Carolyn S., Gullo-Brown, Johnni, Poss, Michael A., Vaccaro, Wayne, Salvati, Mark E.
Published in Bioorganic & medicinal chemistry letters (01.02.2006)
Published in Bioorganic & medicinal chemistry letters (01.02.2006)
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Aminotriazine 5-HT7 antagonists
MATTSON, Ronald J, DENHART, Derek J, PURANDARE, Ashok, TORTOLANI, David, YUFEN ZHAO, HUA YANG, YEOLA, Suresh, PALMER, Jane, TORRENTE, John, STARK, Arlene, JOHNSON, Graham, CATT, John D, DEE, Michael F, DESKUS, Jeffrey A, DITTA, Jonathan L, EPPERSON, James, KING, H. Dalton, AIMING GAO, POSS, Michael A
Published in Bioorganic & medicinal chemistry letters (16.08.2004)
Published in Bioorganic & medicinal chemistry letters (16.08.2004)
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Discovery and initial SAR of imidazoquinoxalines as inhibitors of the Src-family kinase p56(Lck)
Chen, Ping, Norris, Derek, Iwanowicz, Edwin J, Spergel, Steven H, Lin, James, Gu, Henry H, Shen, Zhongqi, Wityak, John, Lin, Tai-An, Pang, Suhong, De Fex, Henry F, Pitt, Sidney, Shen, Ding Ren, Doweyko, Arthur M, Bassolino, Donna A, Roberge, Jacques Y, Poss, Michael A, Chen, Bang-Chi, Schieven, Gary L, Barrish, Joel C
Published in Bioorganic & medicinal chemistry letters (20.05.2002)
Published in Bioorganic & medicinal chemistry letters (20.05.2002)
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Diaminopyrimidine and diaminopyridine 5-HT7 ligands
DENHART, Derek J, PURANDARE, Ashok V, MATTSON, Ronald J, CATT, John D, KING, H. Dalton, AIMING GAO, DESKUS, Jeffrey A, POSS, Michael A, STARK, Arlene D, TORRENTE, John R, JOHNSON, Graham
Published in Bioorganic & medicinal chemistry letters (16.08.2004)
Published in Bioorganic & medicinal chemistry letters (16.08.2004)
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A general synthesis of dioxolenone prodrug moieties
Sun, CQ, Cheng, PTW, Stevenson, J, Dejneka, T, Brown, B, Wang, TC, Robl, JA, Poss, MA
Published in Tetrahedron letters (11.02.2002)
Published in Tetrahedron letters (11.02.2002)
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BMS‐180560, an insurmountable inhibitor of angiotensin II‐stimulated responses: comparison with losartan and EXP3174
Dickinson, K.E.J., Cohen, R.B., Skwish, S., Delaney, C.L., Serafino, R.P., Poss, M.A., Gu, Z., Ryono, D.E., Moreland, S., Powell, J.R.
Published in British journal of pharmacology (01.09.1994)
Published in British journal of pharmacology (01.09.1994)
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Diastereoselective Reaction of a Grignard Reagent with Chiral Imides: A Practical Preparation of a Key Intermediate in the Synthesis of Ifetroban Sodium
Mueller, Richard H, Wang, Shaopeng, Pansegrau, Paul D, Jannotti, Joy Q, Poss, Michael A, Thottathil, John K, Singh, Janak, Humora, Michael J, Kissick, Thomas P, Boyhan, Brenda
Published in Organic process research & development (01.01.1997)
Published in Organic process research & development (01.01.1997)
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