Discovery and Development of TMPRSS6 Inhibitors Modulating Hepcidin Levels in Human Hepatocytes
Béliveau, François, Tarkar, Aarti, Dion, Sébastien P, Désilets, Antoine, Ghinet, Mariana Gabriela, Boudreault, Pierre-Luc, St-Georges, Catherine, Marsault, Éric, Paone, Daniel, Collins, Jon, Macphee, Colin H, Campobasso, Nino, Groy, Arthur, Cottom, Josh, Ouellette, Michael, Pope, Andrew J, Leduc, Richard
Published in Cell chemical biology (21.11.2019)
Published in Cell chemical biology (21.11.2019)
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High-throughput screening: new technology for the 21st century
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Book Review
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Cell-Based Selection Expands the Utility of DNA-Encoded Small-Molecule Library Technology to Cell Surface Drug Targets: Identification of Novel Antagonists of the NK3 Tachykinin Receptor
Wu, Zining, Graybill, Todd L, Zeng, Xin, Platchek, Michael, Zhang, Jean, Bodmer, Vera Q, Wisnoski, David D, Deng, Jianghe, Coppo, Frank T, Yao, Gang, Tamburino, Alex, Scavello, Genaro, Franklin, G. Joseph, Mataruse, Sibongile, Bedard, Katie L, Ding, Yun, Chai, Jing, Summerfield, Jennifer, Centrella, Paolo A, Messer, Jeffrey A, Pope, Andrew J, Israel, David I
Published in ACS combinatorial science (14.12.2015)
Published in ACS combinatorial science (14.12.2015)
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Inhibitors of LexA Autoproteolysis and the Bacterial SOS Response Discovered by an Academic–Industry Partnership
Mo, Charlie Y, Culyba, Matthew J, Selwood, Trevor, Kubiak, Jeffrey M, Hostetler, Zachary M, Jurewicz, Anthony J, Keller, Paul M, Pope, Andrew J, Quinn, Amy, Schneck, Jessica, Widdowson, Katherine L, Kohli, Rahul M
Published in ACS infectious diseases (09.03.2018)
Published in ACS infectious diseases (09.03.2018)
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Development and validation of reagents and assays for EZH2 peptide and nucleosome high-throughput screens
Diaz, Elsie, Machutta, Carl A, Chen, Stephanie, Jiang, Yong, Nixon, Christopher, Hofmann, Glenn, Key, Danielle, Sweitzer, Sharon, Patel, Mehul, Wu, Zining, Creasy, Caretha L, Kruger, Ryan G, LaFrance, Louis, Verma, Sharad K, Pappalardi, Melissa B, Le, Baochau, Van Aller, Glenn S, McCabe, Michael T, Tummino, Peter J, Pope, Andrew J, Thrall, Sara H, Schwartz, Benjamin, Brandt, Martin
Published in Journal of biomolecular screening (01.12.2012)
Published in Journal of biomolecular screening (01.12.2012)
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Journal Article
Single-molecule detection technologies in miniaturized high-throughput screening: fluorescence intensity distribution analysis
Haupts, Ulrich, Rüdiger, Martin, Ashman, Stephen, Turconi, Sandra, Bingham, Ryan, Wharton, Charlotte, Hutchinson, Jonathan, Carey, Charlotte, Moore, Keith J, Pope, Andrew J
Published in Journal of biomolecular screening (01.02.2003)
Published in Journal of biomolecular screening (01.02.2003)
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Journal Article
Identification via a Parallel Hit Progression Strategy of Improved Small Molecule Inhibitors of the Malaria Purine Uptake Transporter that Inhibit Plasmodium falciparum Parasite Proliferation
Sosa, Yvett, Deniskin, Roman, Frame, I. J, Steiginga, Matthew S, Bandyopadhyay, Deepak, Graybill, Todd L, Kallal, Lorena A, Ouellette, Michael T, Pope, Andrew J, Widdowson, Katherine L, Young, Robert J, Akabas, Myles H
Published in ACS infectious diseases (11.10.2019)
Published in ACS infectious diseases (11.10.2019)
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Journal Article
A novel approach applying a chemical biology strategy in phenotypic screening reveals pathway-selective regulators of histone 3 K27 tri-methylation
Liu, Yan, Platchek, Michael, Kement, Burcu, Bee, Weilin T, Truong, Maggie, Zeng, Xin, Hung, Sunny, Lin, Hong, Morrow, Dwight, Kallal, Lorena A, Xie, Qing, Agarwal, Pankaj, Pope, Andrew J, Wu, Zining
Published in Molecular bioSystems (01.02.2014)
Published in Molecular bioSystems (01.02.2014)
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A High-Content Imaging Screen for Cellular Regulators of β-Catenin Protein Abundance
Zeng, Xin, Montoute, Monica, Bee, Tiger W, Lin, Hong, Kallal, Lorena A, Liu, Yan, Agarwal, Pankaj, Wang, Dayuan, Lu, Quinn, Morrow, Dwight, Pope, Andrew J, Wu, Zining
Published in Journal of biomolecular screening (01.03.2016)
Published in Journal of biomolecular screening (01.03.2016)
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Journal Article
Perspectives on the discovery of small-molecule modulators for epigenetic processes
Lu, Quinn, Quinn, Amy M, Patel, Mehul P, Semus, Simon F, Graves, Alan P, Bandyopadhyay, Deepak, Pope, Andrew J, Thrall, Sara H
Published in Journal of biomolecular screening (01.06.2012)
Published in Journal of biomolecular screening (01.06.2012)
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Journal Article
SB-219383, a Novel Tyrosyl tRNA Synthetase Inhibitor from a Micromonospora sp: I. Fermentation, Isolation and Properties
STEFANSKA, ANNA L, COATES, NIGEL J., MENSAH, LUCY M., POPE, ANDREW J., READY, SARAH J., WARR, STEPHEN. R.
Published in Journal of antibiotics (01.04.2000)
Published in Journal of antibiotics (01.04.2000)
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Development of phenotypic screening assays for γ-globin induction using primary human bone marrow day 7 erythroid progenitor cells
Li, Hu, Xie, Wensheng, Gore, Elizabeth R, Montoute, Monica N, Bee, Weilin Tiger, Zappacosta, Francesca, Zeng, Xin, Wu, Zining, Kallal, Lorena, Ames, Robert S, Pope, Andrew J, Benowitz, Andrew, Erickson-Miller, Connie L
Published in Journal of biomolecular screening (01.12.2013)
Published in Journal of biomolecular screening (01.12.2013)
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Journal Article
Synthesis and Activity of Analogues of SB-219383: Novel Potent Inhibitors of Bacterial Tyrosyl tRNA Synthetase
BERGE, JOHN M., BROOM, NIGEL J. P., HOUGE-FRYDRYCH, CATHERINE S. V., JARVEST, RICHARD L., MENSAH, LUCY, MCNAIR, DAVID J., O'HANLON, PETER J., POPE, ANDREW J., RITTENHOUSE, STEPHEN
Published in Journal of antibiotics (01.11.2000)
Published in Journal of antibiotics (01.11.2000)
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The antimicrobial natural product chuangxinmycin and Some synthetic analogues are potent and selective inhibitors of bacterial tryptophanyl tRNA synthetase
Brown, Murray J., Carter, Paul S., Fenwick, Ashley E., Fosberry, Andrew P., Hamprecht, Dieter W., Hibbs, Martin J., Jarvest, Richard L., Mensah, Lucy, Milner, Peter H., O'Hanlon, Peter J., Pope, Andrew J., Richardson, Christine M., West, Andrew, Witty, David R.
Published in Bioorganic & medicinal chemistry letters (04.11.2002)
Published in Bioorganic & medicinal chemistry letters (04.11.2002)
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Homogeneous fluorescence readouts for miniaturized high-throughput screening: theory and practice
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Book Review
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Nanomolar Inhibitors of Staphylococcus aureus Methionyl tRNA Synthetase with Potent Antibacterial Activity against Gram-Positive Pathogens
JARVEST, Richard L., BERGE, John M., BERRY, Valerie, BOYD, Helen F., BROWN, Murray J., ELDER, John S., FORREST, Andrew K., FOSBERRY, Andrew P., GENTRY, Daniel R., HIBBS, Martin J., JAWORSKI, Deborah D., O'HANLON, Peter J., POPE, Andrew J., RITTENHOUSE, Stephen, SHEPPARD, Robert J., SLATER-RADOSTI, Courtney, WORBY, Angela
Published in Journal of medicinal chemistry (09.05.2002)
Published in Journal of medicinal chemistry (09.05.2002)
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Journal Article
Rational Design of Femtomolar Inhibitors of Isoleucyl tRNA Synthetase from a Binding Model for Pseudomonic Acid-A
Brown, Murray J. B, Mensah, Lucy M, Doyle, Michael L, Broom, Nigel J. P, Osbourne, Neal, Forrest, Andrew K, Richardson, Christine M, O'Hanlon, Peter J, Pope, Andrew J
Published in Biochemistry (Easton) (23.05.2000)
Published in Biochemistry (Easton) (23.05.2000)
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Developments in fluorescence lifetime-based analysis for ultra-HTS
Turconi, Sandra, Bingham, Ryan P., Haupts, Ulrich, Pope, Andrew J.
Published in Drug Discovery Today (2001)
Published in Drug Discovery Today (2001)
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Book Review
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Fluorescence correlation spectroscopy: lead discovery by miniaturized HTS
Auer, Manfred, Moore, Keith J, Meyer-Almes, Franz J, Guenther, Rolf, Pope, Andrew J, Stoeckli, Kurt A
Published in Drug discovery today (01.10.1998)
Published in Drug discovery today (01.10.1998)
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