Modification of the pyridine moiety of non-peptidyl indole GnRH receptor antagonists
Simeone, Joseph P, Bugianesi, Robert L, Ponpipom, Mitree M, Yang, Yi Tien, Lo, Jane-Ling, Yudkovitz, Joel B, Cui, Jisong, Mount, George R, Ren, Rena Ning, Creighton, Mellissa, Mao, An-Hua, Vincent, Stella H, Cheng, Kang, Goulet, Mark T
Published in Bioorganic & medicinal chemistry letters (18.11.2002)
Published in Bioorganic & medicinal chemistry letters (18.11.2002)
Get full text
Journal Article
Synthesis of chiral β-methyl tryptamine-derived GnRH antagonists
Simeone, Joseph P, Bugianesi, Robert L, Ponpipom, Mitree M, Goulet, Mark T, Levorse, Mark S, Desai, Ranjit C
Published in Tetrahedron letters (10.09.2001)
Published in Tetrahedron letters (10.09.2001)
Get full text
Journal Article
Inhibition of Stromelysin-1 (MMP-3) by P1‘-Biphenylylethyl Carboxyalkyl Dipeptides
Esser, Craig K, Bugianesi, Robert L, Caldwell, Charles G, Chapman, Kevin T, Durette, Philippe L, Girotra, Narindar N, Kopka, Ihor E, Lanza, Thomas J, Levorse, Dorothy A, MacCoss, Malcolm, Owens, Karen A, Ponpipom, Mitree M, Simeone, Joseph P, Harrison, Richard K, Niedzwiecki, Lisa, Becker, Joseph W, Marcy, Alice I, Axel, Melinda G, Christen, Amy J, McDonnell, Joseph, Moore, Vernon L, Olszewski, Julie M, Saphos, Cheryl, Visco, Denise M, Shen, Frank, Colletti, Adria, Krieter, Philip A, Hagmann, William K
Published in Journal of medicinal chemistry (14.03.1997)
Published in Journal of medicinal chemistry (14.03.1997)
Get full text
Journal Article
Biochemical and pharmacological characterization of L-659,989: an extremely potent, selective and competitive receptor antagonist of platelet-activating factor
SAN-BAO HWANG, MY-HANH LAM, ALBERTS, A. W, BUGIANESI, R. L, CHABALA, J. C, PONPIPOM, M. M
Published in The Journal of pharmacology and experimental therapeutics (01.08.1988)
Get full text
Published in The Journal of pharmacology and experimental therapeutics (01.08.1988)
Journal Article
Structure-Activity Relationships of C1 and C6 Side Chains of Zaragozic Acid A Derivatives
Ponpipom, Mitree M., Girotra, Narindar N., Bugianesi, Robert L., Roberts, Cathleen D., Berger, Gregory D., Burk, Robert M., Marquis, Robert W., Parsons, William H., Bartizal, Kenneth F.
Published in Journal of medicinal chemistry (01.11.1994)
Published in Journal of medicinal chemistry (01.11.1994)
Get full text
Journal Article
(±)-Trans-2-(3-methoxy-5-methylsulfonyl-4-propoxyphenyl)-5-(3,4,5-trimethoxyphenyl)tetrahydrofuran (L-659,989), a novel, potent PAF receptor antagonist
Ponpipom, Mitree M., Hwang, San-Bao, Doebber, Thomas W., Acton, John J., Alberts, Alfred W., Biftu, Tesfaye, Brooker, David R., Bugianesi, Robert L., Chabala, John C., Gamble, Nancy L., Graham, Donald W., Lam, My-Hanh, Wu, Margaret S.
Published in Biochemical and biophysical research communications (15.02.1988)
Published in Biochemical and biophysical research communications (15.02.1988)
Get full text
Journal Article
Development, synthesis, and biological evaluation of (-)-trans-(2S,5S)-2-[3-[(2-oxopropyl)sulfonyl]-4-n-propoxy-5-(3-hydroxypropoxy)-phenyl]-5-(3,4,5-trimethoxyphenyl)tetrahydrofuran, a potent orally active platelet-activating factor (PAF) antagonist and its water-soluble prodrug phosphate ester
Girotra, N. N, Biftu, T, Ponpipom, M. M, Acton, J. J, Alberts, A. W, Bach, T. N, Ball, R. G, Bugianesi, R. L, Chabala, J. C
Published in Journal of medicinal chemistry (01.09.1992)
Published in Journal of medicinal chemistry (01.09.1992)
Get full text
Journal Article
Enhanced macrophage uptake of synthetically glycosylated human placental beta-glucocerebrosidase
Doebber, T W, Wu, M S, Bugianesi, R L, Ponpipom, M M, Furbish, F S, Barranger, J A, Brady, R O, Shen, T Y
Published in The Journal of biological chemistry (10.03.1982)
Published in The Journal of biological chemistry (10.03.1982)
Get full text
Journal Article
Rearrangement of zaragozic acid a derivatives
Girotra, Narindar N., Reamer, Robert A., Ponpipom, Mitree M.
Published in Tetrahedron letters (02.07.1993)
Published in Tetrahedron letters (02.07.1993)
Get full text
Journal Article
Structure-activity relationships of kadsurenone analogues
Ponpipom, Mitree M, Bugianesi, Robert L, Brooker, David R, Yue, Bao-zhen, Hwang, San-bao, Shen, Tsung-ying
Published in Journal of medicinal chemistry (01.01.1987)
Published in Journal of medicinal chemistry (01.01.1987)
Get full text
Journal Article
Synthetic Glycopeptide Substrates for Receptor-Mediated Endocytosis by Macrophages
Robbins, James C., Lam, My Hanh, Tripp, Catherine S., Bugianesi, Robert L., Ponpipom, Mitree M., Shen, T. Y.
Published in Proceedings of the National Academy of Sciences - PNAS (01.12.1981)
Published in Proceedings of the National Academy of Sciences - PNAS (01.12.1981)
Get full text
Journal Article
Inhibition of delayed hypersensitivity reactions by cinnamyl 1-thioglycosides
Ponpipom, Mitree M, Bugianesi, Robert L, Blake, Thomas J
Published in Journal of medicinal chemistry (01.04.1987)
Published in Journal of medicinal chemistry (01.04.1987)
Get full text
Journal Article
Glycolipids as host resistance stimulators
Ponpipom, Mitree M, Hagmann, William K, O'Grady, Laura A, Jackson, Jesse J, Wood, David D, Zweerink, Hans J
Published in Journal of medicinal chemistry (01.02.1990)
Published in Journal of medicinal chemistry (01.02.1990)
Get full text
Journal Article
Cell-specific ligands for selective drug delivery to tissues and organs
Ponpipom, Mitree M, Bugianesi, Robert L, Robbins, James C, Doebber, T. W, Shen, T. Y
Published in Journal of medicinal chemistry (01.12.1981)
Published in Journal of medicinal chemistry (01.12.1981)
Get full text
Journal Article
Stability of Carbohydrate-Modified Vesicles in vivo: Comparative Effects of Ceramide and Cholesterol Glycoconjugates
Wu, Po-Shun, Wu, Hsiu-Mei, Tin, George W., Schuh, Joseph R., Croasmun, William R., Baldeschwieler, John D., Shen, T. Y., Ponpipom, M. M.
Published in Proceedings of the National Academy of Sciences - PNAS (01.09.1982)
Published in Proceedings of the National Academy of Sciences - PNAS (01.09.1982)
Get full text
Journal Article