Quantitative, Wide-Spectrum Kinase Profiling in Live Cells for Assessing the Effect of Cellular ATP on Target Engagement
Vasta, James D., Corona, Cesear R., Wilkinson, Jennifer, Zimprich, Chad A., Hartnett, James R., Ingold, Morgan R., Zimmerman, Kristopher, Machleidt, Thomas, Kirkland, Thomas A., Huwiler, Kristin G., Ohana, Rachel Friedman, Slater, Michael, Otto, Paul, Cong, Mei, Wells, Carrow I., Berger, Benedict-Tilman, Hanke, Thomas, Glas, Carina, Ding, Ke, Drewry, David H., Huber, Kilian V.M., Willson, Timothy M., Knapp, Stefan, Müller, Susanne, Meisenheimer, Poncho L., Fan, Frank, Wood, Keith V., Robers, Matthew B.
Published in Cell chemical biology (15.02.2018)
Published in Cell chemical biology (15.02.2018)
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Journal Article
Engineered Luciferase Reporter from a Deep Sea Shrimp Utilizing a Novel Imidazopyrazinone Substrate
Hall, Mary P, Unch, James, Binkowski, Brock F, Valley, Michael P, Butler, Braeden L, Wood, Monika G, Otto, Paul, Zimmerman, Kristopher, Vidugiris, Gediminas, Machleidt, Thomas, Robers, Matthew B, Benink, Hélène A, Eggers, Christopher T, Slater, Michael R, Meisenheimer, Poncho L, Klaubert, Dieter H, Fan, Frank, Encell, Lance P, Wood, Keith V
Published in ACS chemical biology (16.11.2012)
Published in ACS chemical biology (16.11.2012)
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Journal Article
Quantifying CDK inhibitor selectivity in live cells
Wells, Carrow I., Vasta, James D., Corona, Cesear R., Wilkinson, Jennifer, Zimprich, Chad A., Ingold, Morgan R., Pickett, Julie E., Drewry, David H., Pugh, Kathryn M., Schwinn, Marie K., Hwang, Byounghoon (Brian), Zegzouti, Hicham, Huber, Kilian V. M., Cong, Mei, Meisenheimer, Poncho L., Willson, Timothy M., Robers, Matthew B.
Published in Nature communications (02.06.2020)
Published in Nature communications (02.06.2020)
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Journal Article
An Improved, Practical, and Scalable Five-Step Synthesis of Psilocybin
Sherwood, Alexander M., Meisenheimer, Poncho, Tarpley, Gary, Kargbo, Robert B.
Published in Synthesis (Stuttgart) (03.03.2020)
Published in Synthesis (Stuttgart) (03.03.2020)
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Journal Article
DELs enable the development of BRET probes for target engagement studies in cells
Teske, Kelly A, Su, Wenji, Corona, Cesear R, Wen, Jing, Deng, Jason, Ping, Yan, Zhang, Zaihong, Zhang, Qi, Wilkinson, Jennifer, Beck, Michael T, Nealey, Kendra R, Vasta, James D, Cong, Mei, Meisenheimer, Poncho L, Kuai, Letian, Robers, Matthew B
Published in Cell chemical biology (17.08.2023)
Published in Cell chemical biology (17.08.2023)
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Journal Article
Novel Heterocyclic Analogues of Firefly Luciferin
Woodroofe, Carolyn C, Meisenheimer, Poncho L, Klaubert, Dieter H, Kovic, Yumi, Rosenberg, Justin C, Behney, Curran E, Southworth, Tara L, Branchini, Bruce R
Published in Biochemistry (Easton) (11.12.2012)
Published in Biochemistry (Easton) (11.12.2012)
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Journal Article
Direct Phosphorylation of Psilocin Enables Optimized cGMP Kilogram-Scale Manufacture of Psilocybin
Kargbo, Robert B, Sherwood, Alexander, Walker, Andrew, Cozzi, Nicholas V, Dagger, Raymond E, Sable, Jessica, O’Hern, Kelsey, Kaylo, Kristi, Patterson, Tura, Tarpley, Gary, Meisenheimer, Poncho
Published in ACS omega (14.07.2020)
Published in ACS omega (14.07.2020)
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Journal Article
Proluciferin Acetals as Bioluminogenic Substrates for Cytochrome P450 Activity and Probes for CYP3A Inhibition
MEISENHEIMER, Poncho L, TETSUO UYEDA, H, DONGPING MA, SOBOL, Mary, MCDOUGALL, Mark G, CORONA, Cesear, SIMPSON, Dan, KLAUBERT, Dieter H, CALI, James J
Published in Drug metabolism and disposition (01.12.2011)
Published in Drug metabolism and disposition (01.12.2011)
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Journal Article
N-Alkylated 6′-Aminoluciferins Are Bioluminescent Substrates for Ultra-Glo and QuantiLum Luciferase: New Potential Scaffolds for Bioluminescent Assays
Woodroofe, Carolyn C, Shultz, John W, Wood, Monika G, Osterman, Jean, Cali, James J, Daily, William J, Meisenheimer, Poncho L, Klaubert, Dieter H
Published in Biochemistry (Easton) (30.09.2008)
Published in Biochemistry (Easton) (30.09.2008)
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Journal Article
Self-Immolative Bioluminogenic Quinone Luciferins for NAD(P)H Assays and Reducing Capacity-Based Cell Viability Assays
Zhou, Wenhui, Leippe, Donna, Duellman, Sarah, Sobol, Mary, Vidugiriene, Jolanta, O'Brien, Martha, Shultz, John W., Kimball, Joshua J., DiBernardo, Céline, Moothart, Leonard, Bernad, Laurent, Cali, James, Klaubert, Dieter H., Meisenheimer, Poncho
Published in Chembiochem : a European journal of chemical biology (21.03.2014)
Published in Chembiochem : a European journal of chemical biology (21.03.2014)
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Journal Article
Synthesis and Biological Evaluation of Tryptamines Found in Hallucinogenic Mushrooms: Norbaeocystin, Baeocystin, Norpsilocin, and Aeruginascin
Sherwood, Alexander M, Halberstadt, Adam L, Klein, Adam K, McCorvy, John D, Kaylo, Kristi W, Kargbo, Robert B, Meisenheimer, Poncho
Published in Journal of natural products (Washington, D.C.) (28.02.2020)
Published in Journal of natural products (Washington, D.C.) (28.02.2020)
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Journal Article
Psilocybin: crystal structure solutions enable phase analysis of prior art and recently patented examples
Kaduk, James, Sherwood, Alexander, Kargbo, Robert, Kaylo, Kristi, Meisenheimer, Poncho, Cozzi, Nicholas
Published in Acta crystallographica. Section A, Foundations and advances (29.07.2022)
Published in Acta crystallographica. Section A, Foundations and advances (29.07.2022)
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Journal Article
Bioluminescent, Nonlytic, Real-Time Cell Viability Assay and Use in Inhibitor Screening
Duellman, Sarah J, Zhou, Wenhui, Meisenheimer, Poncho, Vidugiris, Gediminas, Cali, James J, Gautam, Prson, Wennerberg, Krister, Vidugiriene, Jolanta
Published in Assay and drug development technologies (01.10.2015)
Published in Assay and drug development technologies (01.10.2015)
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Journal Article
Novel No-Wash Luminogenic Probes for the Detection of Transporter Uptake Activity
Mustafa, Dana, Ma, Dongping, Zhou, Wenhui, Meisenheimer, Poncho, Cali, James J
Published in Bioconjugate chemistry (20.01.2016)
Published in Bioconjugate chemistry (20.01.2016)
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Journal Article
Psilocybin: crystal structure solutions enable phase analysis of prior art and recently patented examples
Sherwood, Alexander M., Kargbo, Robert B., Kaylo, Kristi W., Cozzi, Nicholas V., Meisenheimer, Poncho, Kaduk, James A.
Published in Acta crystallographica. Section C, Crystal structure communications (01.01.2022)
Published in Acta crystallographica. Section C, Crystal structure communications (01.01.2022)
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