Search Results - "Poli, Gregory B" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

A β-tryptase inhibitor with a tropanylamide scaffold to improve in vitro stability and to lower hERG channel binding affinity

A β-tryptase inhibitor with a tropanylamide scaffold to improve in vitro stability and to lower hERG channel binding affinity

by Liang, Guyan, Choi-Sledeski, Yong Mi, Shum, Patrick, Chen, Xin, Poli, Gregory B., Kumar, Vasant, Minnich, Anne, Wang, Qingping, Tsay, Joseph, Sides, Keith, Kang, Jiesheng, Zhang, Ying
Published in Bioorganic & medicinal chemistry letters (15.02.2012)

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Journal Article

PRODRUGS OF [4[4-(5-AMINOMETHYL-2-FLUORO-PHENYL)-PIPERIDIN-1-YL]-(1H-PYRROLO-PYRIDIN-YL)-METHANONES AND SYNTHESIS THEREOF

PRODRUGS OF [4[4-(5-AMINOMETHYL-2-FLUORO-PHENYL)-PIPERIDIN-1-YL]-(1H-PYRROLO-PYRIDIN-YL)-METHANONES AND SYNTHESIS THEREOF

by POLI GREGORY B, CHOI SLEDESKI YONG MI
Year of Publication 26.09.2012

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Patent

Development of a novel series of (2-quinolinylmethoxy)phenyl-containing compounds as high-affinity leukotriene D4 receptor antagonists. 4. Addition of chromone moiety enhances leukotriene D4 receptor binding affinity

Development of a novel series of (2-quinolinylmethoxy)phenyl-containing compounds as high-affinity leukotriene D4 receptor antagonists. 4. Addition of chromone moiety enhances leukotriene D4 receptor binding affinity

by Huang, Fu Chih, Galemmo, Robert A, Poli, Gregory B, Learn, Keith S, Morrissette, Mathew M, Johnson, William H, Dankulich, William P, Campbell, Henry F, Carnathan, Gilbert W, Van Inwegen, Richard G
Published in Journal of medicinal chemistry (01.05.1991)

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Journal Article

A SUBSTITUTED PYRIMIDINE AS A PROSTAGLANDIN D2 RECEPTOR ANTAGONIST

A SUBSTITUTED PYRIMIDINE AS A PROSTAGLANDIN D2 RECEPTOR ANTAGONIST

by REILING STEPHAN, HARRIS KEITH JOHN, AGUIAR JOACY C, POLI GREGORY B, STOKLOSA GREGORY T, ZHAO ZHICHENG, CHOI SLEDESKI YONG MI, SHUM PATRICK WAI KWOK
Year of Publication 21.01.2013

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Patent

4[4-(5-AMINOMETHYL-2-FLUORO-PHENYL)-PIPERIDIN-1-YL]-(1H-PYRROLO-PYRIDIN-YL)-METHANONES AND SYNTHESIS THEREOF

4[4-(5-AMINOMETHYL-2-FLUORO-PHENYL)-PIPERIDIN-1-YL]-(1H-PYRROLO-PYRIDIN-YL)-METHANONES AND SYNTHESIS THEREOF

by NIEDUZAK THADDEUS R, POLI GREGORY B, STOKLOSA GREGORY T, ZHAO ZHICHENG, CHOI SLEDESKI YONG MI, SHUM PATRICK WAI KWOK
Year of Publication 11.10.2012

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Patent

INDOLYL-PIPERIDINYL BENZYLAMINES AS BETA-TRYPTASE INHIBITORS

INDOLYL-PIPERIDINYL BENZYLAMINES AS BETA-TRYPTASE INHIBITORS

by NIEDUZAK THADDEUS R, POLI GREGORY B, STOKLOSA GREGORY T, ZHAO ZHICHENG, LIANG GUYAN, CHOI SLEDESKI YONG MI, SHUM PATRICK WAI KWOK
Year of Publication 03.09.2012

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Patent

DISUBSTITUTED [4-(5-AMINOMETHYL-PHENYL)-PIPERIDIN-1-YL]-1H-INDOL-3-YL]-METHANONES

DISUBSTITUTED [4-(5-AMINOMETHYL-PHENYL)-PIPERIDIN-1-YL]-1H-INDOL-3-YL]-METHANONES

by POLI GREGORY B, STOKLOSA GREGORY T, ZHAO ZHICHENG, LIANG GUYAN, CHOI SLEDESKI YONG MI, GARDNER CHARLES J, SHUM PATRICK WAI KWOK
Year of Publication 20.06.2012

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Patent

SUBSTITUTED PYRIMIDINES AS PROSTAGLANDIN D2 RECEPTOR ANTAGONISTS

SUBSTITUTED PYRIMIDINES AS PROSTAGLANDIN D2 RECEPTOR ANTAGONISTS

by HARRIS KEITH J, REILING STEPHAN, STEFANY DAVID, AGUIAR JOACY C, POLI GREGORY B, GARDNER CHARLES, STOKLOSA GREGORY, ZHAO ZHICHENG, CHOI SLEDESKI YONG MI, SHUM PATRICK WAI KWOK
Year of Publication 25.02.2013

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Patent

Structure-based design, synthesis, and profiling of a β-tryptase inhibitor with a spiro-piperidineamide scaffold, benzylamine P1 group, and a substituted indole P4 group

Structure-based design, synthesis, and profiling of a β-tryptase inhibitor with a spiro-piperidineamide scaffold, benzylamine P1 group, and a substituted indole P4 group

by Liang, Guyan, Choi-Sledeski, Yong Mi, Poli, Gregory B., Chen, Xin, Minnich, Anne, Wang, Qingping, Tsay, Joseph, Sides, Keith, Vaz, Roy J.
Published in MedChemComm (01.08.2011)

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Journal Article

Development of a novel series of (2-quinolinylmethoxy)phenyl-containing compounds as high-affinity leukotriene D4 receptor antagonists. 2. Effects of an additional phenyl ring on receptor affinity

Development of a novel series of (2-quinolinylmethoxy)phenyl-containing compounds as high-affinity leukotriene D4 receptor antagonists. 2. Effects of an additional phenyl ring on receptor affinity

by Huang, Fu Chih, Galemmo, Robert A, Johnson, William H, Poli, Gregory B, Morrissette, Matthew M, Mencel, James J, Warus, James D, Campbell, Henry F, Nuss, George W
Published in Journal of medicinal chemistry (01.04.1990)

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Journal Article

Prodrugs of [4[4-(5-aminomethyl-2-fluoro-phenyl)-piperidin-1-yl]-(1H-pyrrolo-pyridin-yl)-methanones and synthesis thereof

Prodrugs of [4[4-(5-aminomethyl-2-fluoro-phenyl)-piperidin-1-yl]-(1H-pyrrolo-pyridin-yl)-methanones and synthesis thereof

by POLI, GREGORY B, CHOI-SLEDESKI, YONG MI
Year of Publication 14.07.2016

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Patent

PRODRUGS OF [4[4-(5-AMINOMETHYL-2-FLUORO-PHENYL)-PIPERIDIN-1-YL]-(1H-PYRROLO-PYRIDIN-YL)-METHANONES AND SYNTHESIS THEREOF

PRODRUGS OF [4[4-(5-AMINOMETHYL-2-FLUORO-PHENYL)-PIPERIDIN-1-YL]-(1H-PYRROLO-PYRIDIN-YL)-METHANONES AND SYNTHESIS THEREOF

by POLI, GREGORY B, CHOI-SLEDESKI, YONG-MI
Year of Publication 31.12.2015

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Patent

Quaternary substituted PDE4 inhibitors I: The synthesis and in vitro evaluation of a novel series of oxindoles

Quaternary substituted PDE4 inhibitors I: The synthesis and in vitro evaluation of a novel series of oxindoles

by Hulme, Christopher, Poli, Gregory B., Fu-Chih Huang, Souness, John E., Djuric, Stevan W.
Published in Bioorganic & medicinal chemistry letters (20.01.1998)

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Journal Article

PRODRUGS OF [4[4-(5-AMINOMETHYL-2-FLUORO-PHENYL)-PIPERIDIN-1-YL]-(1H-PYRROLO-PYRIDIN-YL)-METHANONES AND SYNTHESIS THEREOF

PRODRUGS OF [4[4-(5-AMINOMETHYL-2-FLUORO-PHENYL)-PIPERIDIN-1-YL]-(1H-PYRROLO-PYRIDIN-YL)-METHANONES AND SYNTHESIS THEREOF

by POLI, GREGORY B, CHOI-SLEDESKI, YONG MI
Year of Publication 31.12.2014

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Patent

PRODRUGS OF [4[4-(5-AMINOMETHYL-2-FLUORO-PHENYL)-PIPERIDIN-1-YL]-(1H-PYRROLO-PYRIDIN-YL)-METHANONES AND SYNTHESIS THEREOF

PRODRUGS OF [4[4-(5-AMINOMETHYL-2-FLUORO-PHENYL)-PIPERIDIN-1-YL]-(1H-PYRROLO-PYRIDIN-YL)-METHANONES AND SYNTHESIS THEREOF

by POLI, GREGORY B, CHOI-SLEDESKI, YONG MI
Year of Publication 31.10.2014

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Patent

PRODRUGS OF [4[4-(5-AMINOMETHYL-2-FLUORO-PHENYL)-PIPERIDIN-1-YL]-(1H-PYRROLO-PYRIDIN-YL)-METHANONES AND SYNTHESIS THEREOF

PRODRUGS OF [4[4-(5-AMINOMETHYL-2-FLUORO-PHENYL)-PIPERIDIN-1-YL]-(1H-PYRROLO-PYRIDIN-YL)-METHANONES AND SYNTHESIS THEREOF

by POLI, GREGORY B, CHOI-SLEDESKI, YONG MI
Year of Publication 26.09.2014

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Patent

PRODRUGS OF Š4Š4-(5-AMINOMETHYL-2-FLUORO-PHENYL)-PIPERIDIN-1-YL -(1H-PYRROLO-PYRIDIN-YL)-METHANONES AND SYNTHESIS THEREOF

PRODRUGS OF Š4Š4-(5-AMINOMETHYL-2-FLUORO-PHENYL)-PIPERIDIN-1-YL -(1H-PYRROLO-PYRIDIN-YL)-METHANONES AND SYNTHESIS THEREOF

by POLI GREGORY B, CHOI-SLEDESKI YONG MI
Year of Publication 29.08.2014

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Patent

PRO-DRUGS AF [4[4-(5-AMINOMETHYL-2-FLUOR-PHENYL)-PIPERIDIN-1-YL]-(1H-PYRROLO-PYRIDIN-YL)-METHANONER OG SYNTESE DERAF

PRO-DRUGS AF [4[4-(5-AMINOMETHYL-2-FLUOR-PHENYL)-PIPERIDIN-1-YL]-(1H-PYRROLO-PYRIDIN-YL)-METHANONER OG SYNTESE DERAF

by POLI, GREGORY B, CHOI-SLEDESKI, YONG MI
Year of Publication 11.08.2014

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Patent

PRODRUGS OF [4[4-(5-AMINOMETHYL-2-FLUORO-PHENYL)-PIPERIDIN-1-YL]-(1H-PYRROLO-PYRIDIN-YL)-METHANONES AND SYNTHESIS THEREOF

PRODRUGS OF [4[4-(5-AMINOMETHYL-2-FLUORO-PHENYL)-PIPERIDIN-1-YL]-(1H-PYRROLO-PYRIDIN-YL)-METHANONES AND SYNTHESIS THEREOF

by YONG MI CHOI-SLEDESKI, GREGORY B. POLI
Year of Publication 18.07.2014

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Patent

PRODRUGS OF [4[4-(5-AMINOMETHYL-2-FLUORO-PHENYL)-PIPERIDIN-1-YL]-(1H-PYRROLO-PYRIDIN-YL)-METHANONES AND SYNTHESIS THEREOF

PRODRUGS OF [4[4-(5-AMINOMETHYL-2-FLUORO-PHENYL)-PIPERIDIN-1-YL]-(1H-PYRROLO-PYRIDIN-YL)-METHANONES AND SYNTHESIS THEREOF

by POLI, GREGORY B, CHOI-SLEDESKI, YONG MI
Year of Publication 14.05.2014

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Patent

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