Novel orally available salvinorin A analog PR-38 inhibits gastrointestinal motility and reduces abdominal pain in mouse models mimicking irritable bowel syndrome
Sałaga, M, Polepally, P R, Sobczak, M, Grzywacz, D, Kamysz, W, Sibaev, A, Storr, M, Do Rego, J C, Zjawiony, J K, Fichna, J
Published in The Journal of pharmacology and experimental therapeutics (01.07.2014)
Published in The Journal of pharmacology and experimental therapeutics (01.07.2014)
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Journal Article
Salvinorin A analogues PR‐37 and PR‐38 attenuate compound 48/80‐induced itch responses in mice
Salaga, M, Polepally, P R, Zielinska, M, Marynowski, M, Fabisiak, A, Murawska, N, Sobczak, K, Sacharczuk, M, Do Rego, J C, Roth, B L, Zjawiony, J K, Fichna, J
Published in British journal of pharmacology (01.09.2015)
Published in British journal of pharmacology (01.09.2015)
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Journal Article
New C(2)-sulfonyl ester-type Salvinorin A ligands to the kappa-opioid receptor
Polepally, PR, Keasling, A, White, K, Vardy, E, Roth, BL, Zjawiony, JK
Published in Planta Medica (09.04.2015)
Published in Planta Medica (09.04.2015)
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Conference Proceeding
High affinity C(2)-thiocarbonate and thioacetate-type salvinorin A ligands to the kappa-opioid receptor
Polepally, PR, Keasling, A, White, K, Vardy, E, Mosier, PD, Roth, BL, Zjawiony, JK
Published in Planta Medica (09.04.2015)
Published in Planta Medica (09.04.2015)
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Conference Proceeding
New Michael Acceptor-type of Salvinorin A Ligands to Kappa-Opioid Receptor
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Conference Proceeding
Synthesis and In Vitro Biological Evaluation of New Dicarboxylic Ester-type Salvinorin A Analogs
Polepally, PR, Roth, BL, White, K, Ferreira, D, Zjawiony, JK
Published in Planta Medica (22.03.2013)
Published in Planta Medica (22.03.2013)
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Conference Proceeding
New salvinorin A – Derived ligands to opioid receptors
Polepally, PR, Setola, V, Vardy, E, Roth, BL, Mosier, PD, Zjawiony, JK
Published in Planta Medica (19.07.2012)
Published in Planta Medica (19.07.2012)
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Conference Proceeding
Michael Acceptor Approach to the Design of New Salvinorin A- Based High Affinity Ligands to the Kappa-Opioid Receptor
Polepally, PR, Setola, V, Vardy, E, Roth, BL, Mosier, PD, Zjawiony, J
Published in Planta Medica (01.04.2012)
Published in Planta Medica (01.04.2012)
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Conference Proceeding