Chemical Synthesis and Biological Evaluation of 3-Substituted Estrone/Estradiol Derivatives as 17β-Hydroxysteroid Dehydrogenase Type 1 Inhibitors Acting via a Reverse Orientation of the Natural Substrate Estrone
Ngueta, Adrien Djiemeny, Roy, Jenny, Maltais, René, Poirier, Donald
Published in Molecules (Basel, Switzerland) (07.01.2023)
Published in Molecules (Basel, Switzerland) (07.01.2023)
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Synthesis and characterization of some new Cu(II), Ni(II) and Zn(II) complexes with salicylidene thiosemicarbazones: antibacterial, antifungal and in vitro antileukemia activity
Pahontu, Elena, Fala, Valeriu, Gulea, Aurelian, Poirier, Donald, Tapcov, Victor, Rosu, Tudor
Published in Molecules (Basel, Switzerland) (24.07.2013)
Published in Molecules (Basel, Switzerland) (24.07.2013)
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Induction of Endoplasmic Reticulum Stress-Mediated Apoptosis by Aminosteroid RM-581 Efficiently Blocks the Growth of PC-3 Cancer Cells and Tumors Resistant or Not to Docetaxel
Maltais, René, Roy, Jenny, Perreault, Martin, Sato, Sachiko, Lévesque, Julie-Christine, Poirier, Donald
Published in International journal of molecular sciences (17.10.2021)
Published in International journal of molecular sciences (17.10.2021)
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Synthesis and Characterization of Novel Cu(II), Pd(II) and Pt(II) Complexes with 8-Ethyl-2-hydroxytricyclo(7.3.1.0(2,7))tridecan-13-one-thiosemicarbazone: Antimicrobial and in Vitro Antiproliferative Activity
Pahonțu, Elena, Paraschivescu, Codruța, Ilieș, Diana-Carolina, Poirier, Donald, Oprean, Camelia, Păunescu, Virgil, Gulea, Aurelian, Roșu, Tudor, Bratu, Ovidiu
Published in Molecules (Basel, Switzerland) (21.05.2016)
Published in Molecules (Basel, Switzerland) (21.05.2016)
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Comparison between Hippocampus-Synthesized and Circulation-Derived Sex Steroids in the Hippocampus
Hojo, Yasushi, Higo, Shimpei, Ishii, Hirotaka, Ooishi, Yuuki, Mukai, Hideo, Murakami, Gen, Kominami, Toshihiro, Kimoto, Tetsuya, Honma, Seijiro, Poirier, Donald, Kawato, Suguru
Published in Endocrinology (Philadelphia) (01.11.2009)
Published in Endocrinology (Philadelphia) (01.11.2009)
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An Improved Synthesis of Glucuronide Metabolites of Hindered Phenolic Xenoestrogens
Sancéau, Jean-Yves, Bélanger, Patrick, Maltais, René, Poirier, Donald
Published in Current organic synthesis (01.01.2022)
Published in Current organic synthesis (01.01.2022)
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Molecular therapy of breast cancer: progress and future directions
Chen, Jiong, Poirier, Donald, Lin, Sheng-Xiang, Zhou, Ming, Wang, Cheng, Azzi, Arezki, Mazumdar, Mausumi
Published in Nature reviews. Endocrinology (01.09.2010)
Published in Nature reviews. Endocrinology (01.09.2010)
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Investigation of the In Vitro and In Vivo efficiency of RM-532-105, a 17β-hydroxysteroid dehydrogenase type 3 inhibitor, in LAPC-4 prostate cancer cell and tumor models
Kenmogne, Lucie Carolle, Roy, Jenny, Maltais, René, Rouleau, Mélanie, Neveu, Bertrand, Pouliot, Frédéric, Poirier, Donald
Published in PloS one (09.02.2017)
Published in PloS one (09.02.2017)
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Parallel Solid-Phase Synthesis using a New Diethylsilylacetylenic Linker and Leading to Mestranol Derivatives with Potent Antiproliferative Activities on Multiple Cancer Cell Lines
Dutour, Raphaël, Maltais, René, Perreault, Martin, Roy, Jenny, Poirier, Donald
Published in Anti-cancer agents in medicinal chemistry (01.01.2018)
Published in Anti-cancer agents in medicinal chemistry (01.01.2018)
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Regiospecificity and stereospecificity of human UDP-glucuronosyltransferases in the glucuronidation of estriol, 16-epiestriol, 17-epiestriol, and 13-epiestradiol
Sneitz, Nina, Vahermo, Mikko, Mosorin, Johanna, Laakkonen, Liisa, Poirier, Donald, Finel, Moshe
Published in Drug metabolism and disposition (01.03.2013)
Published in Drug metabolism and disposition (01.03.2013)
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Journal Article
Aminosteroid RM-581 Decreases Cell Proliferation of All Breast Cancer Molecular Subtypes, Alone and in Combination with Breast Cancer Treatments
Burguin, Anna, Roy, Jenny, Ouellette, Geneviève, Maltais, René, Bherer, Juliette, Diorio, Caroline, Poirier, Donald, Durocher, Francine
Published in Journal of clinical medicine (24.06.2023)
Published in Journal of clinical medicine (24.06.2023)
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Journal Article
Development of New Resolvin D1 Analogues for Osteoarthritis Therapy: Acellular and Computational Approaches to Study Their Antioxidant Activities
Kariminezhad, Zahra, Rahimi, Mahdi, Fernandes, Julio, Maltais, René, Sancéau, Jean-Yves, Poirier, Donald, Fahmi, Hassan, Benderdour, Mohamed
Published in Antioxidants (01.04.2024)
Published in Antioxidants (01.04.2024)
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