Effect of several 5-hydroxytryptamine(1A) receptor ligands on the micturition reflex in rats: comparison with WAY 100635
Testa, R, Guarneri, L, Poggesi, E, Angelico, P, Velasco, C, Ibba, M, Cilia, A, Motta, G, Riva, C, Leonardi, A
Published in The Journal of pharmacology and experimental therapeutics (01.09.1999)
Get full text
Published in The Journal of pharmacology and experimental therapeutics (01.09.1999)
Journal Article
Effect of different 5‐hydroxytryptamine receptor subtype antagonists on the micturition reflex in rats
Testa, R., Guarneri, L., Angelico, P., Velasco, C., Poggesi, E., Cilia, A., Leonardi, A.
Published in BJU international (01.02.2001)
Published in BJU international (01.02.2001)
Get full text
Journal Article
Pharmacological characterization of the uroselective alpha-1 antagonist Rec 15/2739 (SB 216469): role of the alpha-1L adrenoceptor in tissue selectivity, part I
Leonardi, A, Hieble, J P, Guarneri, L, Naselsky, D P, Poggesi, E, Sironi, G, Sulpizio, A C, Testa, R
Published in The Journal of pharmacology and experimental therapeutics (01.06.1997)
Get full text
Published in The Journal of pharmacology and experimental therapeutics (01.06.1997)
Journal Article
Pharmacological characterization of the uroselective alpha-1 antagonist Rec 15/2739 (SB 216469): role of the alpha-1L adrenoceptor in tissue selectivity, part II
Testa, R, Guarneri, L, Angelico, P, Poggesi, E, Taddei, C, Sironi, G, Colombo, D, Sulpizio, A C, Naselsky, D P, Hieble, J P, Leonardi, A
Published in The Journal of pharmacology and experimental therapeutics (01.06.1997)
Get full text
Published in The Journal of pharmacology and experimental therapeutics (01.06.1997)
Journal Article
N-[2-[4-(2-Methoxyphenyl)-1-piperazinyl]ethyl]-N-(2-nitrophenyl) Cyclohexanecarboxamide: A Novel Pre- and Postsynaptic 5-Hydroxytryptamine1A Receptor Antagonist Active on the Lower Urinary Tract
A. Leonardi, L. Guarneri, E. Poggesi, P. Angelico, C. Velasco, A. Cilia, R. Testa
Published in The Journal of pharmacology and experimental therapeutics (01.12.2001)
Get full text
Published in The Journal of pharmacology and experimental therapeutics (01.12.2001)
Journal Article
Mediation of noradrenaline‐induced contractions of rat aorta by the (α1B‐adrenoceptor subtype
Testa, R., Guarneri, L., Poggesi, E., Simonazzi, I., Taddei, C., Leonardi, A.
Published in British journal of pharmacology (01.02.1995)
Published in British journal of pharmacology (01.02.1995)
Get full text
Journal Article
Functional antagonistic activity of Rec 15/2739, a novel alpha-1 antagonist selective for the lower urinary tract, on noradrenaline-induced contraction of human prostate and mesenteric artery
Testa, R, Guarneri, L, Taddei, C, Poggesi, E, Angelico, P, Sartani, A, Leonardi, A, Gofrit, O N, Meretyk, S, Caine, M
Published in The Journal of pharmacology and experimental therapeutics (01.06.1996)
Get full text
Published in The Journal of pharmacology and experimental therapeutics (01.06.1996)
Journal Article
Searching for cyclazosin analogues as α1B-adrenoceptor antagonists
GIARDINA, Dario, POLIMANTI, O, SAGRATINI, G, ANGELI, P, GULINI, U, MARUCCI, G, MELCHIORRE, C, POGGESI, E, LEONARDI, A
Published in Farmaco (Società chimica italiana : 1989) (01.07.2003)
Published in Farmaco (Società chimica italiana : 1989) (01.07.2003)
Get full text
Journal Article
Synthesis, screening, and molecular modeling of new potent and selective antagonists at the alpha(1d) adrenergic receptor
Leonardi, A, Barlocco, D, Montesano, F, Cignarella, G, Motta, G, Testa, R, Poggesi, E, Seeber, M, De Benedetti, PG, Fanelli, F
Published in Journal of medicinal chemistry (08.04.2004)
Published in Journal of medicinal chemistry (08.04.2004)
Get full text
Journal Article
Prazosin-related compounds. Effect of transforming the piperazinylquinazoline moiety into an aminomethyltetrahydroacridine system on the affinity for alpha(1)-adrenoreceptors
Rosini, M, Antonello, A, Cavalli, A, Bolognesi, ML, Minarini, A, Marucci, G, Poggesi, E, Leonardi, A, Melchiorre, C
Published in Journal of medicinal chemistry (06.11.2003)
Published in Journal of medicinal chemistry (06.11.2003)
Get full text
Journal Article
1,3-dioxolane-based ligands as a novel class of alpha(1)-adrenoceptor antagonists
Brasili, L, Sorbi, C, Franchini, S, Manicardi, M, Angeli, P, Marucci, G, Leonardi, A, Poggesi, E
Published in Journal of medicinal chemistry (10.04.2003)
Published in Journal of medicinal chemistry (10.04.2003)
Get full text
Journal Article
Structure-activity relationships in 1,4-benzodioxan-related compounds. 7. Selectivity of 4-phenylchroman analogues for alpha(1)-adrenoreceptor subtypes
Quaglia, W, Pigini, M, Piergentili, A, Giannella, M, Gentili, F, Marucci, G, Carrieri, A, Carotti, A, Poggesi, E, Leonardi, A, Melchiorre, C
Published in Journal of medicinal chemistry (11.04.2002)
Published in Journal of medicinal chemistry (11.04.2002)
Get full text
Journal Article
Effects of some antidepressants on the volume-induced reflex contractions of the rat urinary bladder: lack of correlation with muscarinic receptors affinity
Pietra, C, Poggesi, E, Angelico, P, Guarneri, L, Testa, R
Published in Pharmacological research (01.07.1990)
Published in Pharmacological research (01.07.1990)
Get more information
Journal Article
Structure-activity relationships in 1,4-benzodioxan-related compounds. 8. {2-[2-(4-chlorobenzyloxy)phenoxy]ethyl}-[2-(2,6-dimethoxyphenoxy)ethyl]amine (clopenphendioxan) as a tool to highlight the involvement of alpha(1D)- and alpha(1B)-adrenoreceptor subtypes in the regulation of human PC-3 prostate cancer cell apoptosis and proliferation
Quaglia, W, Santoni, G, Pigini, M, Piergentili, A, Gentili, F, Buccioni, A, Mosca, M, Lucciarini, R, Amantini, C, Nabissi, MI, Ballarini, P, Poggesi, E, Leonardi, A, Giannella, M
Published in Journal of medicinal chemistry (01.12.2005)
Published in Journal of medicinal chemistry (01.12.2005)
Get full text
Journal Article
Reduction in the number of serotonin receptors in the brainstem of morphine dependent rats: relation to blockade of naloxone precipitated jumping by serotonin agonists
Samanin, R, Cervo, L, Rochat, C, Poggesi, E, Mennini, T
Published in Life sciences (1973) (29.09.1980)
Published in Life sciences (1973) (29.09.1980)
Get more information
Journal Article
New potential uroselective NO-Donor alpha(1)-antagonists
Boschi, D, Tron, GC, Di Stilo, A, Fruttero, R, Gasco, A, Poggesi, E, Motta, G, Leonardi, A
Published in Journal of medicinal chemistry (14.08.2003)
Published in Journal of medicinal chemistry (14.08.2003)
Get full text
Journal Article
Synthesis and Structure−Activity Relationships of 1-Aralkyl-4-Benzylpiperidine and 1-Aralkyl-4-Benzylpiperazine Derivatives as Potent σ Ligands
Costantino, Luca, Gandolfi, Francesca, Sorbi, Claudia, Franchini, Silvia, Prezzavento, Orazio, Vittorio, Franco, Ronsisvalle, Giuseppe, Leonardi, Amedeo, Poggesi, Elena, Brasili, Livio
Published in Journal of medicinal chemistry (13.01.2005)
Published in Journal of medicinal chemistry (13.01.2005)
Get full text
Journal Article
Trans-4-[4-(methoxyphenyl)cyclohexyll-1-arylpiperazines: A new class of potent and selective 5-HT1A receptor ligands as conformationally constrained analogues of 4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]-1-arylpiperazines
Perrone, R, Berardi, F, Colabufo, NA, Leopoldo, M, Lacivita, E, Tortorella, Leonardi, A, Poggesi, E, Testa, R
Published in Journal of medicinal chemistry (06.12.2001)
Published in Journal of medicinal chemistry (06.12.2001)
Get full text
Journal Article
Structure-activity relationships in 1,4-benzodioxan-related compounds. 6. Role of the dioxane unit on selectivity for alpha(1)-adrenoreceptor subtypes
Quaglia, W, Pigini, M, Piergentili, A, Giannella, M, Marucci, G, Poggesi, E, Leonardi, A, Melchiorre, C
Published in Journal of medicinal chemistry (29.07.1999)
Published in Journal of medicinal chemistry (29.07.1999)
Get full text
Journal Article
Changes in Serotonin, but Not Catecholamine, Receptor Binding in the Brain of Morphine-Dependent Rats
Mennini, T, Poggesi, E, Cotecchia, S, De Blasi, A, Samanin, R
Published in Molecular pharmacology (01.09.1981)
Get full text
Published in Molecular pharmacology (01.09.1981)
Journal Article