Effective synthesis of novel dihydrobenzisoxazoles bearing the 2-aminothiazole moiety and evaluation of the antiproliferative activity of their acylated derivatives
Piven, Yuri A, Scherbakov, Alexander M, Yastrebova, Margarita A, Sorokin, Danila V, Shchegolev, Yuri Yu, Matous, Anton E, Zinovich, Veronica G, Khlebnicova, Tatyana S, Lakhvich, Fedor A
Published in Organic & biomolecular chemistry (08.12.2021)
Published in Organic & biomolecular chemistry (08.12.2021)
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Novel O-acylated (E)-3-aryl-6,7-dihydrobenzisoxazol-4(5H)-one oximes targeting HSP90-HER2 axis in breast cancer cells
Piven, Yuri A., Yastrebova, Margarita A., Khamidullina, Alvina I., Scherbakov, Alexander M., Tatarskiy, Victor V., Rusanova, Julia A., Baranovsky, Alexander V., Zinovich, Veronica G., Khlebnicova, Tatyana S., Lakhvich, Fedor A.
Published in Bioorganic & medicinal chemistry (01.01.2022)
Published in Bioorganic & medicinal chemistry (01.01.2022)
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Fluorine-containing lupane triterpenoid acid derivatives: Design, synthesis and biological evaluation as potential anti-inflammatory agents
Khlebnicova, Tatyana S., Piven, Yuri A., Baranovsky, Alexander V., Lakhvich, Fedor A., Sorokina, Iryna V., Tolstikova, Tatyana G.
Published in Steroids (01.07.2019)
Published in Steroids (01.07.2019)
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Computer-aided design, synthesis and evaluation of new SARS-CoV-2 Mpro inhibitors based on 1,5,6,7-tetrahydro-4H-indazol-4-one scaffold
Piven, Yuri A., Zinovich, Veronica G., Shcherbakov, Dmitriy N., Chirkova, Varvara Yu, Belenkaya, Svetlana V., Puzanau, Raman M., Khlebnicova, Tatyana S., Lakhvich, Fedor A.
Published in Medicinal chemistry research (2024)
Published in Medicinal chemistry research (2024)
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Synthesis of novel lupane triterpenoid-indazolone hybrids with oxime ester linkage
Khlebnicova, Tatyana S., Piven, Yuri A., Baranovsky, Alexander V., Lakhvich, Fedor A., Shishkina, Svetlana V., Zicāne, Daina, Tetere, Zenta, Rāviņa, Irisa, Kumpiņš, Viktors, Rijkure, Inese, Mieriņa, Inese, Peipiņš, Uldis, Turks, Māris
Published in Steroids (01.01.2017)
Published in Steroids (01.01.2017)
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A facile synthesis of 4-acylamino-tetrahydroindazoles via the Ritter reaction
Turks, Māris, Strakova, Inta, Gorovojs, Kirils, Belyakov, Sergey, Piven, Yuri A., Khlebnicova, Tatyana S., Lakhvich, Fedor A.
Published in Tetrahedron (05.08.2012)
Published in Tetrahedron (05.08.2012)
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