A simple, modular synthesis of C4-substituted tryptophan derivatives
Bartoccini, F., Bartolucci, S., Mari, M., Piersanti, G.
Published in Organic & biomolecular chemistry (01.01.2016)
Published in Organic & biomolecular chemistry (01.01.2016)
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5-(2-Ethyl-phenyl)-3-(3-methoxy-phenyl)-1H-[1,2,4]triazole (DL-111-IT) and related compounds induce apoptotic patterns in cultures of human tumor cell lines
Burattini, S, Luchetti, F, Battistelli, M, Della Felice, M, Papa, S, Piersanti, G, Tarzia, G, Falcieri, E
Published in Journal of biological regulators and homeostatic agents (01.10.2003)
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Published in Journal of biological regulators and homeostatic agents (01.10.2003)
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Cyclohexylcarbamic Acid 3‘- or 4‘-Substituted Biphenyl-3-yl Esters as Fatty Acid Amide Hydrolase Inhibitors: Synthesis, Quantitative Structure−Activity Relationships, and Molecular Modeling Studies
Mor, Marco, Rivara, Silvia, Lodola, Alessio, Plazzi, Pier Vincenzo, Tarzia, Giorgio, Duranti, Andrea, Tontini, Andrea, Piersanti, Giovanni, Kathuria, Satish, Piomelli, Daniele
Published in Journal of medicinal chemistry (07.10.2004)
Published in Journal of medicinal chemistry (07.10.2004)
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2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine and analogues as A(2A) adenosine receptor antagonists. Design, synthesis, and pharmacological characterization
Minetti, P, Tinti, MO, Carminati, P, Castorina, M, Di Cesare, MA, Di Serio, S, Gallo, G, Ghirardi, O, Giorgi, F, Giorgi, L, Piersanti, G, Bartoccini, F, Tarzia, G
Published in Journal of medicinal chemistry (03.11.2005)
Published in Journal of medicinal chemistry (03.11.2005)
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Design, Synthesis, and Structure−Activity Relationships of Alkylcarbamic Acid Aryl Esters, a New Class of Fatty Acid Amide Hydrolase Inhibitors
Tarzia, Giorgio, Duranti, Andrea, Tontini, Andrea, Piersanti, Giovanni, Mor, Marco, Rivara, Silvia, Plazzi, Pier Vincenzo, Park, Chris, Kathuria, Satish, Piomelli, Daniele
Published in Journal of medicinal chemistry (05.06.2003)
Published in Journal of medicinal chemistry (05.06.2003)
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Journal Article
collisional behavior of ESI-generated protonated molecules of some carbamate FAAH inhibitors isosteres and its relationships with biological activity
Valitutti, Giovanni, Duranti, Andrea, Mor, Marco, Piersanti, Giovanni, Piomelli, Daniele, Rivara, Silvia, Tontini, Andrea, Tarzia, Giorgio, Traldi, Pietro
Published in Journal of mass spectrometry. (01.04.2009)
Published in Journal of mass spectrometry. (01.04.2009)
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Tricyclic Alkylamides as Melatonin Receptor Ligands with Antagonist or Inverse Agonist Activity
Lucini, Valeria, Pannacci, Marilou, Scaglione, Francesco, Fraschini, Franco, Rivara, Sivia, Mor, Marco, Bordi, Fabrizio, Plazzi, Pier Vincenzo, Spadoni, Gilberto, Bedini, Annalida, Piersanti, Giovanni, Diamantini, Giuseppe, Tarzia, Giorgio
Published in Journal of medicinal chemistry (12.08.2004)
Published in Journal of medicinal chemistry (12.08.2004)
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A Trans-Stereoselective Synthesis of 3-Halo-4-alkyl(aryl)-NH-azetidin-2-ones
Bandini, Elisa, Favi, Gianfranco, Martelli, Giorgio, Panunzio, Mauro, Piersanti, Giovanni
Published in Organic letters (20.04.2000)
Published in Organic letters (20.04.2000)
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Stereochemical Aspects of a Two-Step Staudinger Reaction − Asymmetric Synthesis of Chiral Azetidine-2-ones
Bongini, Alessandro, Panunzio, Mauro, Piersanti, Giovanni, Bandini, Elisa, Martelli, Giorgio, Spunta, Giuseppe, Venturini, Alessandro
Published in European journal of organic chemistry (01.07.2000)
Published in European journal of organic chemistry (01.07.2000)
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2-n-Butyl-9-mrthyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine and Analogues as A sub(2A) Adenosine Receptor Antagonists. Design, Synthesis, and Pharmacological Characterization
Minetti, P, Tinti, MO, Carminati, P, Castorina, M, Di Cesare, MA, Di Serio, S, Gallo, G, Ghirardi, O, Giorgi, F, Giorgi, L, Piersanti, G, Bartoccini, F, Tarzia, G
Published in Journal of medicinal chemistry (03.11.2005)
Published in Journal of medicinal chemistry (03.11.2005)
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An efficient synthesis of the cyclic form of scalemic 2,4-di- epi-polyoxamic acid exploiting the hetero Diels-Alder approach
Bandini, Elisa, Martelli, Giorgio, Spunta, Giuseppe, Bongini, Alessandro, Panunzio, Mauro, Piersanti, Giovanni
Published in Tetrahedron: asymmetry (27.11.1997)
Published in Tetrahedron: asymmetry (27.11.1997)
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