Search Results - "Piatnitski, Evgueni L." :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Arylphthalazines. Part 2: 1-(Isoquinolin-5-yl)-4-arylamino phthalazines as potent inhibitors of VEGF receptors I and II

Arylphthalazines. Part 2: 1-(Isoquinolin-5-yl)-4-arylamino phthalazines as potent inhibitors of VEGF receptors I and II

by Duncton, Matthew A.J., Piatnitski, Evgueni L., Katoch-Rouse, Reeti, Smith, Leon M., Kiselyov, Alexander S., Milligan, Daniel L., Balagtas, Chris, Wong, Wai C., Kawakami, Joel, Doody, Jacqueline F.
Published in Bioorganic & medicinal chemistry letters (15.03.2006)

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Oxadiazole derivatives as a novel class of antimitotic agents: Synthesis, inhibition of tubulin polymerization, and activity in tumor cell lines

Oxadiazole derivatives as a novel class of antimitotic agents: Synthesis, inhibition of tubulin polymerization, and activity in tumor cell lines

by Ouyang, Xiaohu, Piatnitski, Evgueni L., Pattaropong, Vatee, Chen, Xiaoling, He, Hai-Ying, Kiselyov, Alexander S., Velankar, Avdhoot, Kawakami, Joel, Labelle, Marc, Smith, Leon, Lohman, Julia, Lee, Sui Ping, Malikzay, Asra, Fleming, James, Gerlak, Jason, Wang, Ying, Rosler, Robin L., Zhou, Kai, Mitelman, Stan, Camara, Margarita, Surguladze, David, Doody, Jacqueline F., Tuma, M. Carolina
Published in Bioorganic & medicinal chemistry letters (01.03.2006)

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Synthesis and structure–activity relationships of 1,2,4-triazoles as a novel class of potent tubulin polymerization inhibitors

Synthesis and structure–activity relationships of 1,2,4-triazoles as a novel class of potent tubulin polymerization inhibitors

by Ouyang, Xiaohu, Chen, Xiaoling, Piatnitski, Evgueni L., Kiselyov, Alexander S., He, Hai-Ying, Mao, Yunyu, Pattaropong, Vatee, Yu, Yang, Kim, Ki H., Kincaid, John, Smith, Leon, Wong, Wai C., Lee, Sui Ping, Milligan, Daniel L., Malikzay, Asra, Fleming, James, Gerlak, Jason, Deevi, Dhanvanthri, Doody, Jacqueline F., Chiang, Hui-Hsien, Patel, Sheetal N., Wang, Ying, Rolser, Robin L., Kussie, Paul, Labelle, Marc, Tuma, M. Carolina
Published in Bioorganic & medicinal chemistry letters (01.12.2005)

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Arylphthalazines: Identification of a new phthalazine chemotype as inhibitors of VEGFR kinase

Arylphthalazines: Identification of a new phthalazine chemotype as inhibitors of VEGFR kinase

by Piatnitski, Evgueni L., Duncton, Matthew A.J., Kiselyov, Alexander S., Katoch-Rouse, Reeti, Sherman, Dan, Milligan, Daniel L., Balagtas, Chris, Wong, Wai C., Kawakami, Joel, Doody, Jacqueline F.
Published in Bioorganic & medicinal chemistry letters (01.11.2005)

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Novel tricyclic azepine derivatives: Biological evaluation of pyrimido[4,5- b]-1,4-benzoxazepines, thiazepines, and diazepines as inhibitors of the epidermal growth factor receptor tyrosine kinase

Novel tricyclic azepine derivatives: Biological evaluation of pyrimido[4,5- b]-1,4-benzoxazepines, thiazepines, and diazepines as inhibitors of the epidermal growth factor receptor tyrosine kinase

by Smith, Leon, Wong, Wai C., Kiselyov, Alexander S., Burdzovic-Wizemann, Sabina, Mao, Yunyu, Xu, Yongjiang, Duncton, Matthew A.J., Kim, Ki, Piatnitski, Evgueni L., Doody, Jacqueline F., Wang, Ying, Rosler, Robin L., Milligan, Daniel, Columbus, John, Balagtas, Chris, Lee, Sui Ping, Konovalov, Andrey, Hadari, Yaron R.
Published in Bioorganic & medicinal chemistry letters (01.10.2006)

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ortho-Substituted azoles as selective and dual inhibitors of VEGF receptors 1 and 2

ortho-Substituted azoles as selective and dual inhibitors of VEGF receptors 1 and 2

by Kiselyov, Alexander S., Piatnitski, Evgueni L., Samet, Alexander V., Kisliy, Victor P., Semenov, Victor V.
Published in Bioorganic & medicinal chemistry letters (01.03.2007)

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1-(Azolyl)-4-(aryl)-phthalazines: Novel Potent Inhibitors of VEGF Receptors I and II

1-(Azolyl)-4-(aryl)-phthalazines: Novel Potent Inhibitors of VEGF Receptors I and II

by Kiselyov, Alexander S., Semenova, Marina, Semenov, Victor V., Piatnitski, Evgueni L.
Published in Chemical biology & drug design (01.11.2006)

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Synthesis of Polysubstituted 4-Fluoroquinolinones

Synthesis of Polysubstituted 4-Fluoroquinolinones

by Kiselyov, Alexander S, Piatnitski, Evgueni L, Doody, Jacqueline
Published in Organic letters (28.10.2004)

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Tricyclic azepine derivatives: Pyrimido[4,5-b]-1,4-benzoxazepines as a novel class of epidermal growth factor receptor kinase inhibitors

Tricyclic azepine derivatives: Pyrimido[4,5-b]-1,4-benzoxazepines as a novel class of epidermal growth factor receptor kinase inhibitors

by Smith, Leon, Piatnitski, Evgueni L., Kiselyov, Alexander S., Ouyang, Xiaohu, Chen, Xiaoling, Burdzovic-Wizemann, Sabina, Xu, Yongjiang, Wang, Ying, Rosler, Robin L., Patel, Sheetal N., Chiang, Hui-Hsien, Milligan, Daniel L., Columbus, John, Wong, Wai C., Doody, Jacqueline F., Hadari, Yaron R.
Published in Bioorganic & medicinal chemistry letters (15.03.2006)

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Hemicarceplexes That Release Guests upon Irradiation

Hemicarceplexes That Release Guests upon Irradiation

by Piatnitski, Evgueni L., Deshayes, Kurt D.
Published in Angewandte Chemie International Edition (20.04.1998)

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Design and Synthesis of Foldamers Based on an Anthracene Diels-Alder Adduct We thank Professor Samuel H. Gellman (University of Wisconsin) and Professors William F. DeGrado and Stanley J. Opella (University of Pennsylvania) for valuable discussions. We also thank Ms. Lori Krim and Mr. Daniel Macks for their experimental and computational contributions to the early stages of this work. Generous financial support from Boehringer-Ingelheim and Alfred P. Bader (J.K.: Alfred E. Bader Fellow, 1996-199

Design and Synthesis of Foldamers Based on an Anthracene Diels-Alder Adduct We thank Professor Samuel H. Gellman (University of Wisconsin) and Professors William F. DeGrado and Stanley J. Opella (University of Pennsylvania) for valuable discussions. We also thank Ms. Lori Krim and Mr. Daniel Macks for their experimental and computational contributions to the early stages of this work. Generous financial support from Boehringer-Ingelheim and Alfred P. Bader (J.K.: Alfred E. Bader Fellow, 1996-199

by Winkler, Jeffrey D., Piatnitski, Evgueni L., Mehlmann, John, Kasparec, Jiri, Axelsen, Paul H.
Published in Angewandte Chemie International Edition (16.02.2001)

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Arylphthalazines: Identification of a New Phthalazine Chemotype as Inhibitors of VEGFR Kinase

Arylphthalazines: Identification of a New Phthalazine Chemotype as Inhibitors of VEGFR Kinase

by Piatnitski, Evgueni L., Duncton, Matthew A. J., Kiselyov, Alexander S., Katoch-Rouse, Reeti, Sherman, Dan, Miligan, Daniel L., Balagtas, Chris, Wong, Wai C., Kawakami, Joel, Doody, Jacqueline F.
Published in ChemInform (24.01.2006)

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Design and Synthesis of Foldamers Based on an Anthracene Diels-Alder Adduct

Design and Synthesis of Foldamers Based on an Anthracene Diels-Alder Adduct

by Winkler, Jeffrey D., Piatnitski, Evgueni L., Mehlmann, John, Kasparec, Jiri, Axelsen, Paul H.
Published in Angewandte Chemie International Edition (16.02.2001)

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Research Article: 1-(Azolyl)-4-(aryl)-phthalazines: Novel Potent Inhibitors of VEGF Receptors I and II

Research Article: 1-(Azolyl)-4-(aryl)-phthalazines: Novel Potent Inhibitors of VEGF Receptors I and II

by Kiselyov, Alexander S, Semenova, Marina, Semenov, Victor V, Piatnitski, Evgueni L
Published in Chemical biology & drug design (01.11.2006)

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Highly Organized Spherical Hosts That Bind Organic Guests in Aqueous Solution with Micromolar Affinity: Microcalorimetry Studies

Highly Organized Spherical Hosts That Bind Organic Guests in Aqueous Solution with Micromolar Affinity: Microcalorimetry Studies

by Piatnitski, Evgueni L., Flowers II, Robert A., Deshayes, Kurt
Published in Chemistry : a European journal (17.03.2000)

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Corrigendum to “Tricyclic azepine derivatives: Pyrimido[4,5- b]-1,4-benzoxazepines as a novel class of epidermal growth factor receptor kinase inhibitors” [Bioorg. Med. Chem. Lett. 16 (2006) 1643–1646]

Corrigendum to “Tricyclic azepine derivatives: Pyrimido[4,5- b]-1,4-benzoxazepines as a novel class of epidermal growth factor receptor kinase inhibitors” [Bioorg. Med. Chem. Lett. 16 (2006) 1643–1646]

by Smith, Leon, Piatnitski, Evgueni L., Kiselyov, Alexander S., Ouyang, Xiaohu, Chen, Xiaoling, Burdzovic-Wizemann, Sabina, Xu, Yongjiang, Pan, Weitao, Chen, Xin, Wang, Ying, Rosler, Robin L., Patel, Sheetal N., Chiang, Hui-Hsien, Milligan, Daniel L., Columbus, John, Wong, Wai C., Doody, Jacqueline F., Hadari, Yaron R.
Published in Bioorganic & medicinal chemistry letters (15.07.2006)

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ortho-Substituted azoles as selective and dual inhibitors of VEGF receptors 1 and 2

ortho-Substituted azoles as selective and dual inhibitors of VEGF receptors 1 and 2

by KISELYOV, Alexander S, PIATNITSKI, Evgueni L, SAMET, Alexander V, KISLIY, Victor P, SEMENOV, Victor V
Published in Bioorganic & medicinal chemistry letters (2007)

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Design and Synthesis of Foldamers Based on an Anthracene Diels-Alder Adduct

Design and Synthesis of Foldamers Based on an Anthracene Diels-Alder Adduct

by Winkler, Jeffrey D., Piatnitski, Evgueni L., Mehlmann, John, Kasparec, Jiri, Axelsen, Paul H.
Published in Angewandte Chemie (16.02.2001)

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Tricyclic Azepine Derivatives: Pyrimido[4,5-b]-1,4-benzoxazepines as a Novel Class of Epidermal Growth Factor Receptor Kinase Inhibitors

Tricyclic Azepine Derivatives: Pyrimido[4,5-b]-1,4-benzoxazepines as a Novel Class of Epidermal Growth Factor Receptor Kinase Inhibitors

by Piatnitski, Evgueni L., ., et al
Published in ChemInform (06.06.2006)

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Synthesis of Polysubstituted 4-Fluoroquinolinones

Synthesis of Polysubstituted 4-Fluoroquinolinones

by Kiselyov, Alexander S., Piatnitski, Evgueni L., Doody, Jacqueline
Published in ChemInform (08.02.2005)

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