Structure activity relationship of 3-nitro-2-(trifluoromethyl)-2H-chromene derivatives as P2Y6 receptor antagonists
Jung, Young-Hwan, Jain, Shanu, Gopinatth, Varun, Phung, Ngan B., Gao, Zhan-Guo, Jacobson, Kenneth A.
Published in Bioorganic & medicinal chemistry letters (01.06.2021)
Published in Bioorganic & medicinal chemistry letters (01.06.2021)
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Journal Article
P2Y 14 receptor inhibition reverses mechanical sensitivity in a mouse model of chronic neuropathic pain
Mufti, Fatma, Jung, Young-Hwan, Giancotti, Luigino A, Yu, Jinha, Chen, Zhoumou, Phung, Ngan B, Jacobson, Kenneth A, Salvemini, Daniela
Published in The FASEB journal (01.05.2022)
Published in The FASEB journal (01.05.2022)
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Journal Article
Structure-activity relationships of pyrimidine nucleotides containing a 5′-α,β-methylene diphosphonate at the P2Y6 receptor
Oliva, Paola, Scortichini, Mirko, Dobelmann, Clemens, Jain, Shanu, Gopinatth, Varun, Toti, Kiran S., Phung, Ngan B., Junker, Anna, Jacobson, Kenneth A.
Published in Bioorganic & medicinal chemistry letters (01.08.2021)
Published in Bioorganic & medicinal chemistry letters (01.08.2021)
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Journal Article
Bridged Piperidine Analogues of a High Affinity Naphthalene-Based P2Y14R Antagonist
Wen, Zhiwei, Salmaso, Veronica, Jung, Young-Hwan, Phung, Ngan B, Gopinatth, Varun, Shah, Qasim, Patterson, Alexandra T, Randle, John C. R, Chen, Zhoumou, Salvemini, Daniela, Lieberman, David I, Whitehead, Gregory S, Karcz, Tadeusz P, Cook, Donald N, Jacobson, Kenneth A
Published in Journal of medicinal chemistry (24.02.2022)
Published in Journal of medicinal chemistry (24.02.2022)
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Journal Article
Bridged Piperidine Analogues of a High Affinity Naphthalene-Based P2Y 14 R Antagonist
Wen, Zhiwei, Salmaso, Veronica, Jung, Young-Hwan, Phung, Ngan B, Gopinatth, Varun, Shah, Qasim, Patterson, Alexandra T, Randle, John C R, Chen, Zhoumou, Salvemini, Daniela, Lieberman, David I, Whitehead, Gregory S, Karcz, Tadeusz P, Cook, Donald N, Jacobson, Kenneth A
Published in Journal of medicinal chemistry (24.02.2022)
Published in Journal of medicinal chemistry (24.02.2022)
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Journal Article
Structure-Activity Relationship of Heterocyclic P2Y 14 Receptor Antagonists: Removal of the Zwitterionic Character with Piperidine Bioisosteres
Jung, Young-Hwan, Salmaso, Veronica, Wen, Zhiwei, Bennett, John M, Phung, Ngan B, Lieberman, David I, Gopinatth, Varun, Randle, John C R, Chen, Zhoumou, Salvemini, Daniela, Karcz, Tadeusz P, Cook, Donald N, Jacobson, Kenneth A
Published in Journal of medicinal chemistry (22.04.2021)
Published in Journal of medicinal chemistry (22.04.2021)
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Journal Article
Structure–Activity Relationship of Heterocyclic P2Y14 Receptor Antagonists: Removal of the Zwitterionic Character with Piperidine Bioisosteres
Jung, Young-Hwan, Salmaso, Veronica, Wen, Zhiwei, Bennett, John M, Phung, Ngan B, Lieberman, David I, Gopinatth, Varun, Randle, John C. R, Chen, Zhoumou, Salvemini, Daniela, Karcz, Tadeusz P, Cook, Donald N, Jacobson, Kenneth A
Published in Journal of medicinal chemistry (22.04.2021)
Published in Journal of medicinal chemistry (22.04.2021)
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Journal Article
Exploration of Alternative Scaffolds for P2Y14 Receptor Antagonists Containing a Biaryl Core
Jung, Young-Hwan, Yu, Jinha, Wen, Zhiwei, Salmaso, Veronica, Karcz, Tadeusz P, Phung, Ngan B, Chen, Zhoumou, Duca, Sierra, Bennett, John M, Dudas, Steven, Salvemini, Daniela, Gao, Zhan-Guo, Cook, Donald N, Jacobson, Kenneth A
Published in Journal of medicinal chemistry (10.09.2020)
Published in Journal of medicinal chemistry (10.09.2020)
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Journal Article
Exploration of Alternative Scaffolds for P2Y 14 Receptor Antagonists Containing a Biaryl Core
Jung, Young-Hwan, Yu, Jinha, Wen, Zhiwei, Salmaso, Veronica, Karcz, Tadeusz P, Phung, Ngan B, Chen, Zhoumou, Duca, Sierra, Bennett, John M, Dudas, Steven, Salvemini, Daniela, Gao, Zhan-Guo, Cook, Donald N, Jacobson, Kenneth A
Published in Journal of medicinal chemistry (10.09.2020)
Published in Journal of medicinal chemistry (10.09.2020)
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Journal Article
P2Y14 Receptor Antagonists Reverse Chronic Neuropathic Pain in a Mouse Model
Mufti, Fatma, Jung, Young-Hwan, Giancotti, Luigino Antonio, Yu, Jinha, Chen, Zhoumou, Phung, Ngan B, Jacobson, Kenneth A, Salvemini, Daniela
Published in ACS medicinal chemistry letters (11.06.2020)
Published in ACS medicinal chemistry letters (11.06.2020)
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Journal Article
Structure activity relationship of 3-nitro-2-(trifluoromethyl)-2H-chromene derivatives as P2Y(6) receptor antagonists
Jung, Young-Hwan, Jain, Shanu, Gopinatth, Varun, Phung, Ngan B., Gao, Zhan-Guo, Jacobson, Kenneth A.
Published in Bioorganic & medicinal chemistry letters (01.06.2021)
Published in Bioorganic & medicinal chemistry letters (01.06.2021)
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Journal Article
Exploration of Alternative Scaffolds for P2Y(14) Receptor Antagonists Containing a Biaryl Core
Jung, Young-Hwan, Yu, Jinha, Wen, Zhiwei, Salmaso, Veronica, Karcz, Tadeusz P., Phung, Ngan B., Chen, Zhoumou, Duca, Sierra, Bennett, John M., Dudas, Steven, Salvemini, Daniela, Gao, Zhan-Guo, Cook, Donald N., Jacobson, Kenneth A.
Published in Journal of medicinal chemistry (10.09.2020)
Published in Journal of medicinal chemistry (10.09.2020)
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Journal Article
P2Y(14) Receptor Antagonists Reverse Chronic Neuropathic Pain in a Mouse Model
Mufti, Fatma, Jung, Young-Hwan, Giancotti, Luigino Antonio, Yu, Jinha, Chen, Zhoumou, Phung, Ngan B., Jacobson, Kenneth A., Salvemini, Daniela
Published in ACS medicinal chemistry letters (11.06.2020)
Published in ACS medicinal chemistry letters (11.06.2020)
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Journal Article
Structure-activity relationships of pyrimidine nucleotides containing a 5 '-alpha,beta-methylene diphosphonate at the P2Y(6) receptor
Oliva, Paola, Scortichini, Mirko, Dobelmann, Clemens, Jain, Shanu, Gopinatth, Varun, Toti, Kiran S., Phung, Ngan B., Junker, Anna, Jacobson, Kenneth A.
Published in Bioorganic & medicinal chemistry letters (01.08.2021)
Published in Bioorganic & medicinal chemistry letters (01.08.2021)
Get full text
Journal Article
Structure-Activity Relationship of Heterocyclic P2Y(14) Receptor Antagonists: Removal of the Zwitterionic Character with Piperidine Bioisosteres
Jung, Young-Hwan, Salmaso, Veronica, Wen, Zhiwei, Bennett, John M., Phung, Ngan B., Lieberman, David, Gopinatth, Varun, Randle, John C. R., Chen, Zhoumou, Salvemini, Daniela, Karcz, Tadeusz P., Cook, Donald N., Jacobson, Kenneth A.
Published in Journal of medicinal chemistry (22.04.2021)
Published in Journal of medicinal chemistry (22.04.2021)
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Journal Article
P2Y 14 Receptor Antagonists Reverse Chronic Neuropathic Pain in a Mouse Model
Mufti, Fatma, Jung, Young-Hwan, Giancotti, Luigino Antonio, Yu, Jinha, Chen, Zhoumou, Phung, Ngan B., Jacobson, Kenneth A., Salvemini, Daniela
Published in ACS medicinal chemistry letters (11.06.2020)
Published in ACS medicinal chemistry letters (11.06.2020)
Get full text
Journal Article
Structure activity relationship of 3-nitro-2-(trifluoromethyl)-2H-chromene derivatives as P2Y 6 receptor antagonists
Jung, Young-Hwan, Jain, Shanu, Gopinatth, Varun, Phung, Ngan B, Gao, Zhan-Guo, Jacobson, Kenneth A
Published in Bioorganic & medicinal chemistry letters (01.06.2021)
Get full text
Published in Bioorganic & medicinal chemistry letters (01.06.2021)
Journal Article
Structure-activity relationships of pyrimidine nucleotides containing a 5'-α,β-methylene diphosphonate at the P2Y 6 receptor
Oliva, Paola, Scortichini, Mirko, Dobelmann, Clemens, Jain, Shanu, Gopinatth, Varun, Toti, Kiran S, Phung, Ngan B, Junker, Anna, Jacobson, Kenneth A
Published in Bioorganic & medicinal chemistry letters (01.08.2021)
Get full text
Published in Bioorganic & medicinal chemistry letters (01.08.2021)
Journal Article