Phase 0 Clinical Trial of the Poly (ADP-Ribose) Polymerase Inhibitor ABT-888 in Patients With Advanced Malignancies
KUMMAR, Shivaani, KINDERS, Robert, MURGO, Anthony J, COLLINS, Jerry, STEINBERG, Seth M, ELIOPOULOS, Helen, GIRANDA, Vincent L, GORDON, Gary, HELMAN, Lee, WILTROUT, Robert, TOMASZEWSKI, Joseph E, DOROSHOW, James H, GUTIERREZ, Martin E, RUBINSTEIN, Larry, PARCHMENT, Ralph E, PHILLIPS, Lawrence R, JIUPING JI, MONKS, Anne, LOW, Jennifer A, CHEN, Alice
Published in Journal of clinical oncology (01.06.2009)
Published in Journal of clinical oncology (01.06.2009)
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Antitumor Benzothiazoles. 8. Synthesis, Metabolic Formation, and Biological Properties of the C- and N-Oxidation Products of Antitumor 2-(4-Aminophenyl)benzothiazoles
Kashiyama, Eiji, Hutchinson, Ian, Chua, Mei-Sze, Stinson, Sherman F, Phillips, Lawrence R, Kaur, Gurmeet, Sausville, Edward A, Bradshaw, Tracey D, Westwell, Andrew D, Stevens, Malcolm F. G
Published in Journal of medicinal chemistry (07.10.1999)
Published in Journal of medicinal chemistry (07.10.1999)
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Deoxyribonucleoside Cyclic N-Acylphosphoramidites as a New Class of Monomers for the Stereocontrolled Synthesis of Oligothymidylyl- and Oligodeoxycytidylyl- Phosphorothioates
Wilk, Andrzej, Grajkowski, Andrzej, Phillips, Lawrence R, Beaucage, Serge L
Published in Journal of the American Chemical Society (15.03.2000)
Published in Journal of the American Chemical Society (15.03.2000)
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Journal Article
Sodium dichloroacetate selectively targets cells with defects in the mitochondrial ETC
Stockwin, Luke H., Yu, Sherry X., Borgel, Suzanne, Hancock, Chad, Wolfe, Tracy L., Phillips, Lawrence R., Hollingshead, Melinda G., Newton, Dianne L.
Published in International journal of cancer (01.12.2010)
Published in International journal of cancer (01.12.2010)
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Journal Article
Liquid Chromatographic Determination of NSC 737664 (ABT-888: An Inhibitor of Poly(ADP-ribose) Polymerase (PARP)) in Plasma and Urine in a Phase 0 Clinical Trial
Phillips, Lawrence R., Hill, Kimberly D., Majerova, Eva
Published in Journal of liquid chromatography & related technologies (01.01.2009)
Published in Journal of liquid chromatography & related technologies (01.01.2009)
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Journal Article
The 3-(N-tert-Butylcarboxamido)-1-propyl Group as an Attractive Phosphate/Thiophosphate Protecting Group for Solid-Phase Oligodeoxyribonucleotide Synthesis
Wilk, Andrzej, Chmielewski, Marcin K, Grajkowski, Andrzej, Phillips, Lawrence R, Beaucage, Serge L
Published in Journal of organic chemistry (06.09.2002)
Published in Journal of organic chemistry (06.09.2002)
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Journal Article
The 4-[N-Methyl-N-(2,2,2-trifluoroacetyl)amino]butyl Group as an Alternative to the 2-Cyanoethyl Group for Phosphate Protection in the Synthesis of Oligodeoxyribonucleotides
Wilk, Andrzej, Grajkowski, Andrzej, Phillips, Lawrence R, Beaucage, Serge L
Published in Journal of organic chemistry (01.10.1999)
Published in Journal of organic chemistry (01.10.1999)
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Journal Article
The automated synthesis of sulfur-containing oligodeoxyribonucleotides using 3H-1,2-benzodithiol-3-one 1,1-dioxide as a sulfur-transfer reagent
Iyer, Radhakrishnan P, Phillips, Lawrence R, Egan, William, Regan, Judith B, Beaucage, Serge L
Published in Journal of organic chemistry (01.07.1990)
Published in Journal of organic chemistry (01.07.1990)
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Journal Article
Modulation of HIV-like Particle Assembly in vitro by Inositol Phosphates
Campbell, Stephen, Fisher, Robert J., Towler, Eric M., Fox, Stephen, Issaq, Haleem J., Wolfe, Tracy, Phillips, Lawrence R., Rein, Alan
Published in Proceedings of the National Academy of Sciences - PNAS (11.09.2001)
Published in Proceedings of the National Academy of Sciences - PNAS (11.09.2001)
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Journal Article
Complete Stereochemistry of Neamphamide A and Absolute Configuration of the β-Methoxytyrosine Residue in Papuamide B
Oku, Naoya, Krishnamoorthy, Ravi, Benson, Alan G, Ferguson, Robert L, Lipton, Mark A, Phillips, Lawrence R, Gustafson, Kirk R, McMahon, James B
Published in Journal of organic chemistry (19.08.2005)
Published in Journal of organic chemistry (19.08.2005)
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Journal Article
Construction of a rhamnose mutation in Bacillus anthracis affects adherence to macrophages but not virulence in guinea pigs
Bozue, Joel A., Parthasarathy, Narayanan, Phillips, Lawrence R., Cote, Christopher K., Fellows, Patricia F., Mendelson, Itai, Shafferman, Avigdor, Friedlander, Arthur M.
Published in Microbial pathogenesis (2005)
Published in Microbial pathogenesis (2005)
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Journal Article
The 2-(N-Formyl-N-methyl)aminoethyl Group as a Potential Phosphate/Thiophosphate Protecting Group in Solid-Phase Oligodeoxyribonucleotide Synthesis
Grajkowski, Andrzej, Wilk, Andrzej, Chmielewski, Marcin K, Phillips, Lawrence R, Beaucage, Serge L
Published in Organic letters (03.05.2001)
Published in Organic letters (03.05.2001)
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Journal Article
Identification of the major metabolite of 2,5-bis(5-hydroxymethyl-2-thienyl)furan (NSC 652287), an antitumor agent, in the S9 subcellular fraction of dog liver cells
Phillips, Lawrence R, Jorden, Jean L, Rivera, Maria I, Upadhyay, Kaye, Wolfe, Tracy L, Stinson, Sherman F
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (05.02.2002)
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (05.02.2002)
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Journal Article
Synthesis of (2-Deoxy-α- and -β-d-erythro-pentofuranosyl)(thymin-1-yl)alkanes and Their Incorporation into Oligodeoxyribonucleotides. Effect of Nucleobase−Sugar Linker Flexibility on the Formation of DNA−DNA and DNA−RNA Hybrids
Boal, Jila H, Wilk, Andrzej, Scremin, Carlo L, Gray, Glenn N, Phillips, Lawrence R, Beaucage, Serge L
Published in Journal of organic chemistry (29.11.1996)
Published in Journal of organic chemistry (29.11.1996)
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Journal Article
3-(N-tert-butylcarboxamido)-1-propyl and 4-oxopentyl groups for phosphate/thiophosphate protection in oligodeoxyribonucleotide synthesis
Wilk, Andrzej, Chmielewski, Marcin K, Grajkowski, Andrzej, Beaucage, Serge L, Phillips, Lawrence R
Published in Current protocols in nucleic acid chemistry (01.02.2003)
Published in Current protocols in nucleic acid chemistry (01.02.2003)
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1-(2-Deoxy-α- and β-D-erythro-pentofuranosyl)-2-(thymin-1-yl)ethane derivatives as conformational probes for altDNA oligonucleotides
Scremin, Carlo L., Boal, Jila H., Wilk, Andrzej, Phillips, Lawrence R., Zhou, Liang, Beaucage, Serge L.
Published in Tetrahedron letters (01.12.1995)
Published in Tetrahedron letters (01.12.1995)
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Journal Article
Solid-phase synthesis, separation, and stereochemical aspects of P-chiral methane- and 4,4'-dimethoxytriphenylmethanephosphonate analogs of oligodeoxyribonucleotides
Stec, Wojciech J, Zon, Gerald, Egan, William, Byrd, R. Andrew, Phillips, Lawrence R, Gallo, Kathleen A
Published in Journal of organic chemistry (01.10.1985)
Published in Journal of organic chemistry (01.10.1985)
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Journal Article
Deoxyribonucleoside phosphoramidites
Wilk, A, Grajkowski, A, Chmielewski, M K, Beaucage, S L, Phillips, L R
Published in Current protocols in nucleic acid chemistry (01.04.2001)
Published in Current protocols in nucleic acid chemistry (01.04.2001)
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